| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM50060080 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_53572 (CHEMBL663592) |
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| Ki | 191±n/a nM |
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| Citation |  Liao, S; Lin, J; Shenderovich, MD; Han, Y; Hasohata, K; Davis, P; Qiu, W; Porreca, F; Yamamura, HI; Hruby, VJ The stereochemical requirements of the novel δ-opioid selective dipeptide antagonist TMT-Tic Bioorg Med Chem Lett7:3049-3052 (1997) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40577.25 |
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| Organism: | MOUSE |
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| Description: | P32300 |
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| Residue: | 372 |
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| Sequence: | MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTAC
TPSDGPGGGAAA
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|
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| BDBM50060080 |
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| n/a |
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| Name | BDBM50060080 |
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| Synonyms: | 2-({2-[(R)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-propionic acid | CHEMBL485576 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H20N2O4 |
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| Mol. Mass. | 340.3731 |
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| SMILES | N[C@@H](Cc1ccc(O)cc1)C(=O)N1Cc2ccccc2C[C@H]1C(O)=O |r| |
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| Structure | 
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