| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Mitogen-activated protein kinase 13 |
|---|
| Ligand | BDBM60589 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_774372 (CHEMBL1908589) |
|---|
| Kd | >10000±n/a nM |
|---|
| Citation |  Davis, MI; Hunt, JP; Herrgard, S; Ciceri, P; Wodicka, LM; Pallares, G; Hocker, M; Treiber, DK; Zarrinkar, PP Comprehensive analysis of kinase inhibitor selectivity. Nat Biotechnol29:1046-51 (2011) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Mitogen-activated protein kinase 13 |
|---|
| Name: | Mitogen-activated protein kinase 13 |
|---|
| Synonyms: | MAP kinase p38 delta | MAPK13 | MK13_HUMAN | Mitogen-activated protein kinase 13 | Mitogen-activated protein kinase 13 (MAPK13) | Mitogen-activated protein kinase p38 | Mitogen-activated protein kinase p38 delta | PRKM13 | SAPK4 | Stress-activated protein kinase 4 | p38 delta/gamma |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 42097.16 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | O15264 |
|---|
| Residue: | 365 |
|---|
| Sequence: | MSLIRKKGFYKQDVNKTAWELPKTYVSPTHVGSGAYGSVCSAIDKRSGEKVAIKKLSRPF
QSEIFAKRAYRELLLLKHMQHENVIGLLDVFTPASSLRNFYDFYLVMPFMQTDLQKIMGM
EFSEEKIQYLVYQMLKGLKYIHSAGVVHRDLKPGNLAVNEDCELKILDFGLARHADAEMT
GYVVTRWYRAPEVILSWMHYNQTVDIWSVGCIMAEMLTGKTLFKGKDYLDQLTQILKVTG
VPGTEFVQKLNDKAAKSYIQSLPQTPRKDFTQLFPRASPQAADLLEKMLELDVDKRLTAA
QALTHPFFEPFRDPEEETEAQQPFDDSLEHEKLTVDEWKQHIYKEIVNFSPIARKDSRRR
SGMKL
|
|
|
|---|
| BDBM60589 |
|---|
| n/a |
|---|
| Name | BDBM60589 |
|---|
| Synonyms: | 6-{[6-(1-methyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline (4) | BDBM50355498 |
|---|
| Type | n/a |
|---|
| Emp. Form. | C18H13N7S |
|---|
| Mol. Mass. | 359.408 |
|---|
| SMILES | Cn1cc(cn1)-c1ccc2nnc(Sc3ccc4ncccc4c3)n2n1 |
|---|
| Structure | 
|
|---|
Search and Browse
