| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Casein kinase I isoform gamma-1 |
|---|
| Ligand | BDBM24654 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_774608 (CHEMBL1908825) |
|---|
| Kd | >10000±n/a nM |
|---|
| Citation |  Davis, MI; Hunt, JP; Herrgard, S; Ciceri, P; Wodicka, LM; Pallares, G; Hocker, M; Treiber, DK; Zarrinkar, PP Comprehensive analysis of kinase inhibitor selectivity. Nat Biotechnol29:1046-51 (2011) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Casein kinase I isoform gamma-1 |
|---|
| Name: | Casein kinase I isoform gamma-1 |
|---|
| Synonyms: | CKI-gamma 1 | CSNK1G1 | Casein kinase I | Casein kinase I gamma 1 isoform | Casein kinase I isoform gamma-1 | KC1G1_HUMAN |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 48530.93 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_774608 |
|---|
| Residue: | 422 |
|---|
| Sequence: | MDHPSREKDERQRTTKPMAQRSAHCSRPSGSSSSSGVLMVGPNFRVGKKIGCGNFGELRL
GKNLYTNEYVAIKLEPIKSRAPQLHLEYRFYKQLGSAGEGLPQVYYFGPCGKYNAMVLEL
LGPSLEDLFDLCDRTFTLKTVLMIAIQLLSRMEYVHSKNLIYRDVKPENFLIGRQGNKKE
HVIHIIDFGLAKEYIDPETKKHIPYREHKSLTGTARYMSINTHLGKEQSRRDDLEALGHM
FMYFLRGSLPWQGLKADTLKERYQKIGDTKRNTPIEALCENFPEEMATYLRYVRRLDFFE
KPDYEYLRTLFTDLFEKKGYTFDYAYDWVGRPIPTPVGSVHVDSGASAITRESHTHRDRP
SQQQPLRNQVVSSTNGELNVDDPTGAHSNAPITAHAEVEVVEEAKCCCFFKRKRKKTAQR
HK
|
|
|
|---|
| BDBM24654 |
|---|
| n/a |
|---|
| Name | BDBM24654 |
|---|
| Synonyms: | 4-N-(2,6-dichlorobenzene)-3-N-(piperidin-4-yl)-1H-pyrazole-3,4-diamido | AT7519 | JMC514986 Compound 33 | pyrazole diamide, 33 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C16H17Cl2N5O2 |
|---|
| Mol. Mass. | 382.244 |
|---|
| SMILES | Clc1cccc(Cl)c1C(=O)Nc1cn[nH]c1C(=O)NC1CCNCC1 |
|---|
| Structure | 
|
|---|
Search and Browse
