| Reaction Details |
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 | Report a problem with these data |
| Target | Substance-K receptor |
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| Ligand | BDBM50366377 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_142711 |
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| IC50 | 0.079000±n/a nM |
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| Citation |  Horwell, DC; Naylor, D; Willems, HM 2,3-Substituted 2-azanorbornanes as polar -turn mimetics Bioorg Med Chem Lett7:31-36 (1997) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Substance-K receptor |
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| Name: | Substance-K receptor |
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| Synonyms: | NK2R_MESAU | Neurokinin 2 receptor | Neurokinin NK2 | TAC2R | TACR2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 43436.75 |
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| Organism: | HAMSTER |
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| Description: | P51144 |
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| Residue: | 384 |
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| Sequence: | MGGRAIVTDTNIFSGLESNTTGVTAFSMPAWQLALWATAYLGLVLVAVTGNATVIWIILA
HERMRTVTNYFIINLALADLCMAAFNATFNFVYASHNIWYFGRAFCYFQNLFPITAMFVS
IYSMTAIAADRYMAIVHPFQPRLSAPITKATIAGIWLVALALASPQCFYSTITVDQGATK
CVVAWPNDNGGKMLLLYHLVVFVLVYFLPLVVMFVAYSVIGLTLWKRAVPRHQAHGANLR
HLHAKKKFVKAMVLVVLTFAICWLPYHLYFILGSFQKDIYYRKFIQQVYLALFWLAMSST
MYNPIIYCCLNHRFRSGFRLAFRCCPWVTPTEEDRLELTRTPSLSRRVNRCHTKETLFMT
ADMTHSEATNGQVGSPQDVEPAAP
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| BDBM50366377 |
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| n/a |
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| Name | BDBM50366377 |
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| Synonyms: | CHEMBL334721 | MEN-10627 |
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| Type | Small organic molecule |
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| Emp. Form. | C38H48N8O7S |
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| Mol. Mass. | 760.902 |
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| SMILES | CSCC[C@@H]1NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]2CNC(=O)C[C@H](NC1=O)C(=O)N[C@@H](Cc1c[nH]c3ccccc13)C(=O)N[C@@H](Cc1ccccc1)C(=O)N2 |
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| Structure | 
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