| Reaction Details |
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 | Report a problem with these data |
| Target | Vasopressin V1a receptor |
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| Ligand | BDBM50108499 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_214566 |
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| Ki | 7.6±n/a nM |
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| Citation |  Kakefuda, A; Tsukada, J; Kusayama, T; Tahara, A; Tsukamoto, S N-Methylbenzanilide derivatives as a novel class of selective V(1A) receptor antagonists. Bioorg Med Chem Lett12:229-32 (2001) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Vasopressin V1a receptor |
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| Name: | Vasopressin V1a receptor |
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| Synonyms: | Avpr1a | V1AR_RAT | VASOPRESSIN V1A | Vasopressin V1 receptor | Vasopressin V1a receptor | Vasopressin receptor |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 47674.81 |
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| Organism: | RAT |
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| Description: | VASOPRESSIN V1A AVPR1A RAT::P30560 |
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| Residue: | 424 |
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| Sequence: | MSFPRGSQDRSVGNSSPWWPLTTEGSNGSQEAARLGEGDSPLGDVRNEELAKLEIAVLAV
IFVVAVLGNSSVLLALHRTPRKTSRMHLFIRHLSLADLAVAFFQVLPQLCWDITYRFRGP
DWLCRVVKHLQVFAMFASAYMLVVMTADRYIAVCHPLKTLQQPARRSRLMIATSWVLSFI
LSTPQYFIFSVIEIEVNNGTKTQDCWATFIQPWGTRAYVTWMTSGVFVAPVVVLGTCYGF
ICYHIWRNIRGKTASSRHSKGDKGSGEAVGPFHKGLLVTPCVSSVKSISRAKIRTVKMTF
VIVSAYILCWAPFFIVQMWSVWDENFIWTDSENPSITITALLASLNSCCNPWIYMFFSGH
LLQDCVQSFPCCHSMAQKFAKDDSDSMSRRQTSYSNNRSPTNSTGMWKDSPKSSKSIRFI
PVST
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| BDBM50108499 |
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| n/a |
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| Name | BDBM50108499 |
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| Synonyms: | 1N-methyl-1N-{4-methyl-2-[4-(4-methylhexahydro-1-pyrazinylcarbonyl)benzyloxy]phenyl}-4-[2-(2-ethyl-1H-1-imidazolyl)phenylcarboxamido]benzamide | CHEMBL75489 |
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| Type | Small organic molecule |
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| Emp. Form. | C40H42N6O4 |
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| Mol. Mass. | 670.7993 |
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| SMILES | CCc1nccn1-c1ccccc1C(=O)Nc1ccc(cc1)C(=O)N(C)c1ccc(C)cc1OCc1ccc(cc1)C(=O)N1CCN(C)CC1 |
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| Structure | 
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