| Reaction Details |
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 | Report a problem with these data |
| Target | Glutamyl aminopeptidase |
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| Ligand | BDBM50036824 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_32828 (CHEMBL646206) |
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| Ki | 140±n/a nM |
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| Citation |  Chauvel, EN; Coric, P; Llorens-Cortès, C; Wilk, S; Roques, BP; Fournié-Zaluski, MC Investigation of the active site of aminopeptidase A using a series of new thiol-containing inhibitors. J Med Chem37:1339-46 (1994) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Glutamyl aminopeptidase |
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| Name: | Glutamyl aminopeptidase |
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| Synonyms: | AMPE_HUMAN | AP-A | Aminopeptidase A | CD_antigen=CD249 | Differentiation antigen gp160 | EAP | ENPEP | Glutamyl aminopeptidase |
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| Type: | PROTEIN |
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| Mol. Mass.: | 109226.47 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_32829 |
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| Residue: | 957 |
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| Sequence: | MNFAEREGSKRYCIQTKHVAILCAVVVGVGLIVGLAVGLTRSCDSSGDGGPGTAPAPSHL
PSSTASPSGPPAQDQDICPASEDESGQWKNFRLPDFVNPVHYDLHVKPLLEEDTYTGTVS
ISINLSAPTRYLWLHLRETRITRLPELKRPSGDQVQVRRCFEYKKQEYVVVEAEEELTPS
SGDGLYLLTMEFAGWLNGSLVGFYRTTYTENGQVKSIVATDHEPTDARKSFPCFDEPNKK
ATYTISITHPKEYGALSNMPVAKEESVDDKWTRTTFEKSVPMSTYLVCFAVHQFDSVKRI
SNSGKPLTIYVQPEQKHTAEYAANITKSVFDYFEEYFAMNYSLPKLDKIAIPDFGTGAME
NWGLITYRETNLLYDPKESASSNQQRVATVVAHELVHQWFGNIVTMDWWEDLWLNEGFAS
FFEFLGVNHAETDWQMRDQMLLEDVLPVQEDDSLMSSHPIIVTVTTPDEITSVFDGISYS
KGSSILRMLEDWIKPENFQKGCQMYLEKYQFKNAKTSDFWAALEEASRLPVKEVMDTWTR
QMGYPVLNVNGVKNITQKRFLLDPRANPSQPPSDLGYTWNIPVKWTEDNITSSVLFNRSE
KEGITLNSSNPSGNAFLKINPDHIGFYRVNYEVATWDSIATALSLNHKTFSSADRASLID
DAFALARAQLLDYKVALNLTKYLKREENFLPWQRVISAVTYIISMFEDDKELYPMIEEYF
QGQVKPIADSLGWNDAGDHVTKLLRSSVLGFACKMGDREALNNASSLFEQWLNGTVSLPV
NLRLLVYRYGMQNSGNEISWNYTLEQYQKTSLAQEKEKLLYGLASVKNVTLLSRYLDLLK
DTNLIKTQDVFTVIRYISYNSYGKNMAWNWIQLNWDYLVNRYTLNNRNLGRIVTIAEPFN
TELQLWQMESFFAKYPQAGAGEKPREQVLETVKNNIEWLKQHRNTIREWFFNLLESG
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| BDBM50036824 |
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| n/a |
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| Name | BDBM50036824 |
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| Synonyms: | (S)-3-Carboxy-1-mercaptomethyl-propyl-ammonium | (S)-4-Amino-5-mercapto-pentanoic acid | CHEMBL28124 |
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| Type | Small organic molecule |
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| Emp. Form. | C5H11NO2S |
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| Mol. Mass. | 149.211 |
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| SMILES | N[C@H](CS)CCC(O)=O |
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| Structure | 
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