Reaction Details |
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Target | P2Y purinoceptor 2 |
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Ligand | BDBM50371704 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_463988 (CHEMBL929975) |
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IC50 | >100000±n/a nM |
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Citation | Weyler, S; Baqi, Y; Hillmann, P; Kaulich, M; Hunder, AM; Müller, IA; Müller, CE Combinatorial synthesis of anilinoanthraquinone derivatives and evaluation as non-nucleotide-derived P2Y2 receptor antagonists. Bioorg Med Chem Lett18:223-7 (2008) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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P2Y purinoceptor 2 |
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Name: | P2Y purinoceptor 2 |
Synonyms: | ATP receptor | P2RY2_MOUSE | P2U purinoceptor 1 | P2U1 | P2Y purinoceptor 2 | P2Y2 | P2ru1 | P2ry2 | Purinergic receptor | Purinergic receptor P2Y2 |
Type: | PROTEIN |
Mol. Mass.: | 42202.78 |
Organism: | Mus musculus |
Description: | ChEMBL_587770 |
Residue: | 373 |
Sequence: | MAADLEPWNSTINGTWEGDELGYKCRFNEDFKYVLLPVSYGVVCVLGLCLNVVALYIFLC
RLKTWNASTTYMFHLAVSDSLYAASLPLLVYYYARGDHWPFSTVLCKLVRFLFYTNLYCS
ILFLTCISVHRCLGVLRPLHSLRWGRARYARRVAAVVWVLVLACQAPVLYFVTTSVRGTR
ITCHDTSARELFSHFVAYSSVMLGLLFAVPFSVILVCYVLMARRLLKPAYGTTGGLPRAK
RKSVRTIALVLAVFALCFLPFHVTRTLYYSFRSLDLSCHTLNAINMAYKITRPLASANSC
LDPVLYFLAGQRLVRFARDAKPPTEPTPSPQARRKLGLHRPNRTVRKDLSVSSDDSRRTE
STPAGSETKDIRL
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BDBM50371704 |
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n/a |
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Name | BDBM50371704 |
Synonyms: | CHEMBL270415 |
Type | Small organic molecule |
Emp. Form. | C14H7BrNO5S |
Mol. Mass. | 381.179 |
SMILES | Nc1c2C(=O)c3ccccc3C(=O)c2c(Br)cc1S([O-])(=O)=O |
Structure |
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