| Reaction Details |
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 | Report a problem with these data |
| Target | Protein-tyrosine-phosphatase |
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| Ligand | BDBM50379184 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_810616 (CHEMBL2015667) |
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| IC50 | 18000±n/a nM |
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| Citation |  He, Y; Zeng, LF; Yu, ZH; He, R; Liu, S; Zhang, ZY Bicyclic benzofuran and indole-based salicylic acids as protein tyrosine phosphatase inhibitors. Bioorg Med Chem20:1940-6 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Protein-tyrosine-phosphatase |
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| Name: | Protein-tyrosine-phosphatase |
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| Synonyms: | Secreted effector protein | Secreted protein-tyrosine phosphatase |
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| Type: | PROTEIN |
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| Mol. Mass.: | 50881.86 |
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| Organism: | Yersinia pestis |
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| Description: | ChEMBL_810616 |
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| Residue: | 468 |
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| Sequence: | MNLSLSDLHRQVSRLVQQESGDCTGKLRGNVAANKETTFQGLTIASGARESEKVFAQTVL
SHVANVVLTQEDTAKLLQSTVKHNLNNYDLRSVGNGNSVLVSLRSDQMTLQDAKVLLEAA
LRQESGARGHVSSHSHSALHAPGTPVREGLRSHLDPRTPPLPPRERPHTSGHHGAGEARA
TAPSTVSPYGPEARAELSSRLTTLRNTLAPATNDPRYLQACGGEKLNRFRDIQCCRQTAV
RADLNANYIQVGNTRTIACQYPLQSQLESHFRMLAENRTPVLAVLASSSEIANQRFGMPD
YFRQSGTYGSITVESKMTQQVGLGDGIMADMYTLTIREAGQKTISVPVVHVGNWPDQTAV
SSEVTKALASLVDQTAETKRNMYESKGSSAVGDDSKLRPVIHCRAGVGRTAQLIGAMCMN
DSRNSQLSVEDMVSQMRVQRNGIMVQKDEQLDVLIKLAEGQGRPLLNS
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| BDBM50379184 |
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| n/a |
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| Name | BDBM50379184 |
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| Synonyms: | CHEMBL2010868 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H8O4 |
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| Mol. Mass. | 204.1788 |
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| SMILES | OC(=O)c1cc2cccc(O)c2cc1O |
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| Structure | 
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