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TargetD(2) dopamine receptor
LigandBDBM50010618
Substrate/Competitorn/a
Meas. Tech.ChEMBL_61139 (CHEMBL670072)
IC50 230±n/a nM
Citation Seri-Levy, A; West, S; Richards, WG Molecular similarity, quantitative chirality, and QSAR for chiral drugs. J Med Chem37:1727-32 (1994) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
D(2) dopamine receptor
Name:D(2) dopamine receptor
Synonyms:DOPAMINE D2 | DOPAMINE D2 Long | DOPAMINE D2 Short | DRD2_RAT | Dopamine D2 receptor | Dopamine2-like | Drd2
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:50931.60
Organism:Rattus norvegicus (rat)
Description:P61169
Residue:444
Sequence:
MDPLNLSWYDDDLERQNWSRPFNGSEGKADRPHYNYYAMLLTLLIFIIVFGNVLVCMAVS
REKALQTTTNYLIVSLAVADLLVATLVMPWVVYLEVVGEWKFSRIHCDIFVTLDVMMCTA
SILNLCAISIDRYTAVAMPMLYNTRYSSKRRVTVMIAIVWVLSFTISCPLLFGLNNTDQN
ECIIANPAFVVYSSIVSFYVPFIVTLLVYIKIYIVLRKRRKRVNTKRSSRAFRANLKTPL
KGNCTHPEDMKLCTVIMKSNGSFPVNRRRMDAARRAQELEMEMLSSTSPPERTRYSPIPP
SHHQLTLPDPSHHGLHSNPDSPAKPEKNGHAKIVNPRIAKFFEIQTMPNGKTRTSLKTMS
RRKLSQQKEKKATQMLAIVLGVFIICWLPFFITHILNIHCDCNIPPVLYSAFTWLGYVNS
AVNPIIYTTFNIEFRKAFMKILHC
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  Blast E-value cutoff:
BDBM50010618
n/a
NameBDBM50010618
Synonyms:(+)-3-(1-Propyl-piperidin-3-yl)-phenol | 3-((R)-1-Propyl-piperidin-3-yl)-phenol | 3-(1-Propyl-piperidin-3-yl)-phenol | 3PPP,(-) | CHEMBL7393 | cid_202478
TypeSmall organic molecule
Emp. Form.C14H21NO
Mol. Mass.219.3226
SMILESCCCN1CCC[C@@H](C1)c1cccc(O)c1
Structure
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