| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Hrh3 protein |
|---|
| Ligand | BDBM85412 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 3.4±n/a nM |
|---|
| Comments | PDSP_908 |
|---|
| Citation |  Yates, SL; Phillips, JG; Gregory, R; Pawlowski, GP; Fadnis, L; Khan, MA; Ali, SM; Tedford, CE Identification and pharmacological characterization of a series of new 1H-4-substituted-imidazoyl histamine H3 receptor ligands. J Pharmacol Exp Ther289:1151-9 (1999) [PubMed] |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Hrh3 protein |
|---|
| Name: | Hrh3 protein |
|---|
| Synonyms: | HISTAMINE H3 | HRH3 | Hrh3 protein |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 37860.96 |
|---|
| Organism: | RAT |
|---|
| Description: | Q5PPG3 |
|---|
| Residue: | 344 |
|---|
| Sequence: | MERAPPDGLMNASGTLAGEAAAAGGARGFSAAWTAVLAALMALLIVATVLGNALVMLAFV
ADSSLRTQNNFFLLNLAISDFLVGAFCIPLYVPYVLTGRWTFGRGLCKLWLVVDYLLCAS
SVFNIVLISYDRFLSVTRAVSYRAQQGDTRRAVRKMALVWVLAFLLYGPAILSWEYLSGG
SSIPEGHCYAEFFYNWYFLITASTLEFFTPFLSVTFFNLSIYLNIQRRTRLRLDGGREAG
PEPPPDAQPSPPPAPPSCWGCWPKGHGEAMPLHRGSKPSASSASLEKRMKMVSQSITQRF
RLSRDKKVAKSLAIIVSIFGLCWAPYTLLMIIRAACHGRCIPDY
|
|
|
|---|
| BDBM85412 |
|---|
| n/a |
|---|
| Name | BDBM85412 |
|---|
| Synonyms: | GT 2287 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C16H24N2 |
|---|
| Mol. Mass. | 244.3752 |
|---|
| SMILES | C(CC#CCCc1cnc[nH]1)CC1CCCCC1 |
|---|
| Structure | 
|
|---|
Search and Browse
