| Reaction Details |
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 | Report a problem with these data |
| Target | Alpha-2A adrenergic receptor |
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| Ligand | BDBM81979 |
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| Substrate/Competitor | n/a |
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| Ki | 57.54±n/a nM |
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| Comments | PDSP_914 |
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| Citation |  Brink, CB; Wade, SM; Neubig, RR Agonist-directed trafficking of porcine alpha(2A)-adrenergic receptor signaling in Chinese hamster ovary cells: l-isoproterenol selectively activates G(s). J Pharmacol Exp Ther294:539-47 (2000) [PubMed] |
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| More Info.: | Get all data from this article |
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| Alpha-2A adrenergic receptor |
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| Name: | Alpha-2A adrenergic receptor |
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| Synonyms: | Alpha-2A adrenergic receptor | adrenergic Alpha2 | adrenergic Alpha2A |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 48998.96 |
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| Organism: | PIG |
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| Description: | adrenergic Alpha2 0 PIG::P18871 |
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| Residue: | 450 |
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| Sequence: | MGSLQPEAGNASWNGTEAPGGGARATPYSLQVTLTLVCLAGLLMLFTVFGNVLVIIAVFT
SRALKAPQNLFLVSLASADILVATLVIPFSLANEVMGYWYFGKAWCEIYLALDVLFCTSS
IVHLCAISLDRYWSITQAIEYNLKRTPRRIKAIIVTVWVISAVISFPPLISIEKKAGGGG
QQPAEPRCEINDQKWYVISSCIGSFFAPCLIMILVYVRIYQIAKRRTRVPPSRRGPDAAA
ALPGGAERRPNGLGPERGVGRVGAEAEPLPVQLNGAPGEPAPAGPRDADGLDLEESSSSE
HAERPPGPRRSERGPRAKSKARASQVKPGDSLPRRGPGAPGPGAPATGAGEERGGVAKAS
RWRGRQNREKRFTFVLAVVIGVFVVCWFPFFFTYTLTAVGCSVPPTLFKFFFWFGYCNSS
LNPVIYTIFNHDFRRAFKKILCRGDRKRIV
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| BDBM81979 |
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| n/a |
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| Name | BDBM81979 |
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| Synonyms: | CAS_5051-62-7 | CAS_65636 | Fluprofylline | Guanabenz | NSC_3517 | NSC_65636 |
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| Type | Small organic molecule |
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| Emp. Form. | C8H8Cl2N4 |
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| Mol. Mass. | 231.082 |
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| SMILES | [#7]\[#6](-[#7])=[#7]\[#7]=[#6]-c1c(Cl)cccc1Cl |w:5.5| |
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| Structure | 
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