| Reaction Details |
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 | Report a problem with these data |
| Target | Gamma-aminobutyric acid receptor subunit rho-3 |
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| Ligand | BDBM24183 |
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| Substrate/Competitor | n/a |
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| Ki | 580±n/a nM |
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| Comments | PDSP_867 |
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| Citation |  Chang, Y; Covey, DF; Weiss, DS Correlation of the apparent affinities and efficacies of gamma-aminobutyric acid(C) receptor agonists. Mol Pharmacol58:1375-80 (2000) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Gamma-aminobutyric acid receptor subunit rho-3 |
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| Name: | Gamma-aminobutyric acid receptor subunit rho-3 |
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| Synonyms: | GABA B rho 1 | GABRR3 | GBRR3_HUMAN | Gamma-aminobutyric acid receptor subunit rho-3 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 54281.08 |
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| Organism: | Homo sapiens (Human) |
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| Description: | GABA B rho 1 0 HUMAN::A8MPY1 |
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| Residue: | 467 |
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| Sequence: | MVLAFQLVSFTYIWIILKPNVCAASNIKMTHQRCSSSMKQTCKQETRMKKDDSTKARPQK
YEQLLHIEDNDFAMRPGFGGSPVPVGIDVHVESIDSISETNMDFTMTFYLRHYWKDERLS
FPSTANKSMTFDHRLTRKIWVPDIFFVHSKRSFIHDTTMENIMLRVHPDGNVLLSLRITV
SAMCFMDFSRFPLDTQNCSLELESYAYNEDDLMLYWKHGNKSLNTEEHMSLSQFFIEDFS
ASSGLAFYSSTGWYNRLFINFVLRRHVFFFVLQTYFPAILMVMLSWVSFWIDRRAVPARV
SLGITTVLTMSTIITAVSASMPQVSYLKAVDVYLWVSSLFVFLSVIEYAAVNYLTTVEER
KQFKKTGKISRMYNIDAVQAMAFDGCYHDSEIDMDQTSLSLNSEDFMRRKSICSPSTDSS
RIKRRKSLGGHVGRIILENNHVIDTYSRILFPIVYILFNLFYWGVYV
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| BDBM24183 |
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| n/a |
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| Name | BDBM24183 |
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| Synonyms: | 4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic acid | Aminalon | CHEMBL96 | GABA | Gamma-Aminobutyric acid | [3H]GABA | cid_119 |
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| Type | Radiolabeled ligand |
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| Emp. Form. | C4H9NO2 |
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| Mol. Mass. | 103.1198 |
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| SMILES | NCCCC(O)=O |
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| Structure | 
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