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TargetPeptidyl-prolyl cis-trans isomerase H
LigandBDBM92913
Substrate/Competitorn/a
Meas. Tech.PPIase Assay
pH7.8±n/a
Temperature278.15±n/a K
Ki>1.00e+5±n/a nM
Commentsextracted
Citation Daum, SSchumann, MMathea, SAumüller, TBalsley, MAConstant, SLde Lacroix, BFKruska, FBraun, MSchiene-Fischer, C Isoform-specific inhibition of cyclophilins. Biochemistry48:6268-77 (2009) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Peptidyl-prolyl cis-trans isomerase H
Name:Peptidyl-prolyl cis-trans isomerase H
Synonyms:CYP20 | CYPH | PPIH | PPIH_HUMAN | Peptidyl-prolyl cis-trans isomerase H (USA-Cyp) | Small nuclear ribonucleoprotein particle-specific cyclophilin H
Type:Protein
Mol. Mass.:19211.45
Organism:Homo sapiens (Human)
Description:O43447
Residue:177
Sequence:
MAVANSSPVNPVVFFDVSIGGQEVGRMKIELFADVVPKTAENFRQFCTGEFRKDGVPIGY
KGSTFHRVIKDFMIQGGDFVNGDGTGVASIYRGPFADENFKLRHSAPGLLSMANSGPSTN
GCQFFITCSKCDWLDGKHVVFGKIIDGLLVMRKIENVPTGPNNKPKLPVVISQCGEM
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BDBM92913
n/a
NameBDBM92913
Synonyms:Aryl 1-indanylketone, 2
TypeSmall molecule
Emp. Form.C22H18FNO3
Mol. Mass.363.3816
SMILESNc1cc(F)cc(-c2ccc(O)c(c2)C(=O)C2CCc3ccccc23)c1O
Structure
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