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TargetTrace amine-associated receptor 1
LigandBDBM106645
Substrate/Competitorn/a
Meas. Tech.Binding Assay
Temperature277.15±0 K
Ki 1±n/a nM
Citation Galley, GGoergler, AZbinden, KGNorcross, RStalder, H Aminomethyl-4-imidazoles US Patent US8586617 Publication Date 11/19/2013
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Trace amine-associated receptor 1
Name:Trace amine-associated receptor 1
Synonyms:TAAR1_MOUSE | Ta1 | Taar1 | Tar1 | Trace amine receptor 1 (TARR1) | Trace amine-associated receptor 1 (TAAR1) | Trace amine-associated receptor1 | Trar1
Type:Protein
Mol. Mass.:37635.41
Organism:Mus musculus (Mouse)
Description:Q923Y8
Residue:332
Sequence:
MHLCHAITNISHRNSDWSREVQASLYSLMSLIILATLVGNLIVIISISHFKQLHTPTNWL
LHSMAIVDFLLGCLIMPCSMVRTVERCWYFGEILCKVHTSTDIMLSSASIFHLAFISIDR
YCAVCDPLRYKAKINISTILVMILVSWSLPAVYAFGMIFLELNLKGVEELYRSQVSDLGG
CSPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRTNVQVGLEGKSQAPQ
SKETKAAKTLGIMVGVFLVCWCPFFLCTVLDPFLGYVIPPSLNDALYWFGYLNSALNPMV
YAFFYPWFRRALKMVLLGKIFQKDSSRSKLFL
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  Blast E-value cutoff:
BDBM106645
n/a
NameBDBM106645
Synonyms:US8586617, 242
TypeSmall organic molecule
Emp. Form.C13H16BrN3
Mol. Mass.294.19
SMILESCC(C)N(Cc1cnc[nH]1)c1cccc(Br)c1
Structure
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