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TargetVascular endothelial growth factor A
LigandBDBM107697
Substrate/Competitorn/a
Meas. Tech.ELISA Assay
EC50>1.00e+5±n/a nM
Citation Kawamoto, RMWu, SWarshakoon, NCEvdokimov, AGGreis, KDBoyer, AS Prolyl hydroxylase inhibitors and methods of use US Patent US8598210 Publication Date 12/3/2013
More Info.:Get all data from this article,  Assay Method
 
Vascular endothelial growth factor A
Name:Vascular endothelial growth factor A
Synonyms:VEGF | VEGF-A | VEGFA | VEGFA_HUMAN | VPF | Vascular endothelial growth factor (VEGF) | Vascular endothelial growth factor A (VEGF) | Vascular endothelial growth factor A (VEGF2) | Vascular permeability factor
Type:Protein
Mol. Mass.:27063.81
Organism:Homo sapiens (Human)
Description:P15692
Residue:395
Sequence:
MTDRQTDTAPSPSYHLLPGRRRTVDAAASRGQGPEPAPGGGVEGVGARGVALKLFVQLLG
CSRFGGAVVRAGEAEPSGAARSASSGREEPQPEEGEEEEEKEEERGPQWRLGARKPGSWT
GEAAVCADSAPAARAPQALARASGRGGRVARRGAEESGPPHSPSRRGSASRAGPGRASET
MNFLLSWVHWSLALLLYLHHAKWSQAAPMAEGGGQNHHEVVKFMDVYQRSYCHPIETLVD
IFQEYPDEIEYIFKPSCVPLMRCGGCCNDEGLECVPTEESNITMQIMRIKPHQGQHIGEM
SFLQHNKCECRPKKDRARQEKKSVRGKGKGQKRKRKKSRYKSWSVPCGPCSERRKHLFVQ
DPQTCKCSCKNTDSRCKARQLELNERTCRCDKPRR
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  Blast E-value cutoff:
BDBM107697
n/a
NameBDBM107697
Synonyms:US8598210, Table XV, 3 | US8722895, 3: {[5-(4-Cyano-phenyl)-3-hydroxy-pyridine-2- carbonyl]-amino}-acetic acid methyl ester
TypeSmall organic molecule
Emp. Form.C16H13N3O4
Mol. Mass.311.2921
SMILESCOC(=O)CNC(=O)c1ncc(cc1O)-c1ccc(cc1)[N+]#[C-]
Structure
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