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TargetVascular endothelial growth factor A
LigandBDBM107707
Substrate/Competitorn/a
Meas. Tech.ELISA Assay
EC50 1.5e+4±n/a nM
Citation Kawamoto, RMWu, SWarshakoon, NCEvdokimov, AGGreis, KDBoyer, AS Prolyl hydroxylase inhibitors and methods of use US Patent US8598210 Publication Date 12/3/2013
More Info.:Get all data from this article,  Assay Method
 
Vascular endothelial growth factor A
Name:Vascular endothelial growth factor A
Synonyms:VEGF | VEGF-A | VEGFA | VEGFA_HUMAN | VPF | Vascular endothelial growth factor (VEGF) | Vascular endothelial growth factor A (VEGF) | Vascular endothelial growth factor A (VEGF2) | Vascular permeability factor
Type:Protein
Mol. Mass.:27063.81
Organism:Homo sapiens (Human)
Description:P15692
Residue:395
Sequence:
MTDRQTDTAPSPSYHLLPGRRRTVDAAASRGQGPEPAPGGGVEGVGARGVALKLFVQLLG
CSRFGGAVVRAGEAEPSGAARSASSGREEPQPEEGEEEEEKEEERGPQWRLGARKPGSWT
GEAAVCADSAPAARAPQALARASGRGGRVARRGAEESGPPHSPSRRGSASRAGPGRASET
MNFLLSWVHWSLALLLYLHHAKWSQAAPMAEGGGQNHHEVVKFMDVYQRSYCHPIETLVD
IFQEYPDEIEYIFKPSCVPLMRCGGCCNDEGLECVPTEESNITMQIMRIKPHQGQHIGEM
SFLQHNKCECRPKKDRARQEKKSVRGKGKGQKRKRKKSRYKSWSVPCGPCSERRKHLFVQ
DPQTCKCSCKNTDSRCKARQLELNERTCRCDKPRR
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BDBM107707
n/a
NameBDBM107707
Synonyms:US11426393, Compound Table XV.13 | US8598210, Table XV, 13 | US8722895, 13: {[5-(4-Isopropylphenyl)-3-hydroxypyridine- 2-carbonyl]amino}-acetic acid | US9598370, Example 00138 | USRE47437, Example {[5-(4-Isopropylphenyl)-3-hydroxypyridine-2-carbonyl]amino}-acetic acid
TypeSmall organic molecule
Emp. Form.C17H18N2O4
Mol. Mass.314.3358
SMILESCC(C)c1ccc(cc1)-c1cnc(C(=O)NCC(O)=O)c(O)c1
Structure
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