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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Glycogen phosphorylase, muscle form | ||
| Ligand | BDBM50246619 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Inhibition Assay | ||
| pH | 7.2±n/a | ||
| Temperature | 295.15±n/a K | ||
| IC50 | 4.610e+5±n/a nM | ||
| Comments | extracted | ||
| Citation |  Zhang, L; Jia, X; Dong, J; Chen, D; Liu, J; Zhang, L; Wen, X Synthesis and evaluation of novel oleanolic acid derivatives as potential antidiabetic agents. Chem Biol Drug Des83:297-305 (2014) [PubMed] Article | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Glycogen phosphorylase, muscle form | |||
| Name: | Glycogen phosphorylase, muscle form | ||
| Synonyms: | Glycogen Phosphorylase (PYGM) | Glycogen phosphorylase a (RMGPa) | Glycogen phosphorylase, muscle form | Myophosphorylase | PYGM | PYGM_RABIT | ||
| Type: | Enzyme | ||
| Mol. Mass.: | 97296.32 | ||
| Organism: | Oryctolagus cuniculus (rabbit) | ||
| Description: | Phosphorylation of Ser-15 converts phosphorylase B (unphosphorylated) to phosphorylase A. | ||
| Residue: | 843 | ||
| Sequence: |
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| BDBM50246619 | |||
| n/a | |||
| Name | BDBM50246619 | ||
| Synonyms: | (4aS,6aS,6bR,8aR,10S,12aR,12bR,14bS)-benzyl 10-hydroxy-2,2,6a,6b,9,9,12a-heptamethyl-1,2,3,4,4a,5,6,6a,6b,7,8,8a,9,10,11,12,12a,12b,13,14b-icosahydropicene-4a-carboxylate | CHEMBL445301 | benzyl (4aS,6aS,6bR,8aR,10S,12aR,12bR,14bS)-10- hydroxy-2,2,6a,6b,9,9,12a-heptamethyl- 1,3,4,5,6,7,8,8a,10,11,12,12b,13,14b- tetradecahydropicene-4a-carboxylate (Compound 4) | ||
| Type | Small organic molecule | ||
| Emp. Form. | C37H54O3 | ||
| Mol. Mass. | 546.8229 | ||
| SMILES | CC1(C)CC[C@@]2(CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]2C1)C(=O)OCc1ccccc1 |r,c:10| | ||
| Structure | 
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