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TargetTrace amine-associated receptor 7b
LigandBDBM129420
Substrate/Competitorn/a
Meas. Tech.Radioligand Binding
pH7.4±n/a
Temperature310.15±n/a K
Ki 9.4±n/a nM
Commentsextracted
Citation Galley, GNorcross, RDPflieger, P Heterocyclic amine derivatives US Patent US8802673 Publication Date 8/12/2014
More Info.:Get all data from this article,  Assay Method
 
Trace amine-associated receptor 7b
Name:Trace amine-associated receptor 7b
Synonyms:TAA7B_RAT | Ta12 | Taar7b | Tar12 | Trace amine-associated receptor 1 (TAAR1) | Trar12
Type:Enzyme
Mol. Mass.:40296.65
Organism:Rattus norvegicus (Rat)
Description:Q923X8
Residue:358
Sequence:
MATDDDRFPWDQDSILSRDLLSASSMQLCYEKLNRSCVRSPYSPGPRLILYAVFGFGAVL
AVCGNLLVMTSILHFRQLHSPANFLVASLACADFLVGLTVMPFSMVRSVEGCWYFGDIYC
KFHSSFDGSFCYSSIFHLCFISADRYIAVSDPLIYPTRFTASVSGKCITFSWLLSIIYSF
SLFYTGVNEAGLEDLVSALTCVGGCQIAVNQSWVFINFLLFLVPALVMMTVYSKIFLIAK
QQAQNIEKMGKQTARASESYKDRVAKRERKAAKTLGIAVAAFLLSWLPYFIDSIIDAFLG
FVTPTYVYEILVWIGYYNSAMNPLIYAFFYPWFRKAIKLIVTGKILRENSSATNLFPE
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  Blast E-value cutoff:
BDBM129420
n/a
NameBDBM129420
Synonyms:US8802673, 62
TypeSmall organic molecule
Emp. Form.C16H18BrN3O
Mol. Mass.348.238
SMILESCc1cc(Nc2ccc(cc2)[C@H]2CNCCO2)ncc1Br |r|
Structure
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