Reaction Details |
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Target | Trace amine-associated receptor 1 |
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Ligand | BDBM167492 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Radioligand Binding |
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pH | 7.4±n/a |
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Ki | 2.5±n/a nM |
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Comments | extracted |
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Citation | Galley, G; Ghellamallah, C; Norcross, R; Pflieger, P Pyrazole derivatives US Patent US9073911 Publication Date 7/7/2015 |
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More Info.: | Get all data from this article, Assay Method |
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Trace amine-associated receptor 1 |
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Name: | Trace amine-associated receptor 1 |
Synonyms: | TAAR1_MOUSE | Ta1 | Taar1 | Tar1 | Trace amine receptor 1 (TARR1) | Trace amine-associated receptor 1 (TAAR1) | Trace amine-associated receptor1 | Trar1 |
Type: | Protein |
Mol. Mass.: | 37635.41 |
Organism: | Mus musculus (Mouse) |
Description: | Q923Y8 |
Residue: | 332 |
Sequence: | MHLCHAITNISHRNSDWSREVQASLYSLMSLIILATLVGNLIVIISISHFKQLHTPTNWL
LHSMAIVDFLLGCLIMPCSMVRTVERCWYFGEILCKVHTSTDIMLSSASIFHLAFISIDR
YCAVCDPLRYKAKINISTILVMILVSWSLPAVYAFGMIFLELNLKGVEELYRSQVSDLGG
CSPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRTNVQVGLEGKSQAPQ
SKETKAAKTLGIMVGVFLVCWCPFFLCTVLDPFLGYVIPPSLNDALYWFGYLNSALNPMV
YAFFYPWFRRALKMVLLGKIFQKDSSRSKLFL
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BDBM167492 |
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n/a |
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Name | BDBM167492 |
Synonyms: | US9073911, 41 |
Type | Small organic molecule |
Emp. Form. | C23H24F2N4O3 |
Mol. Mass. | 442.4585 |
SMILES | CCn1nc(cc1-c1cccc(OC(F)F)c1)C(=O)Nc1ccc(cc1)[C@H]1CNCCO1 |r| |
Structure |
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