| Reaction Details |
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 | Report a problem with these data |
| Target | Trace amine-associated receptor 1 |
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| Ligand | BDBM167458 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Radioligand Binding |
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| pH | 7.4±n/a |
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| Ki | 4.9±n/a nM |
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| Comments | extracted |
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| Citation |  Galley, G; Ghellamallah, C; Norcross, R; Pflieger, P Pyrazole derivatives US Patent US9073911 Publication Date 7/7/2015 |
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| More Info.: | Get all data from this article, Assay Method |
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| Trace amine-associated receptor 1 |
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| Name: | Trace amine-associated receptor 1 |
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| Synonyms: | TAAR1_RAT | Ta1 | Taar1 | Tar1 | Trace amine receptor 1 (TARR1) | Trace amine-associated receptor 1 | Trace amine-associated receptor 1 (TAAR1) | Trace amine-associated receptor1 | Trar1 |
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| Type: | Enzyme |
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| Mol. Mass.: | 38034.73 |
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| Organism: | Rattus norvegicus (Rat) |
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| Description: | Q923Y9 |
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| Residue: | 332 |
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| Sequence: | MHLCHNSANISHTNSNWSRDVRASLYSLISLIILTTLVGNLIVIISISHFKQLHTPTNWL
LHSMAVVDFLLGCLVMPYSMVRTVEHCWYFGELFCKLHTSTDIMLSSASILHLAFISIDR
YYAVCDPLRYKAKINLAAIFVMILISWSLPAVFAFGMIFLELNLEGVEELYHNQVFCLRG
CFPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRANLQVGLEGESRAPQ
SKETKAAKTLGIMVGVFLLCWCPFFFCMVLDPFLGYVIPPTLNDTLNWFGYLNSAFNPMV
YAFFYPWFRRALKMVLFGKIFQKDSSRSKLFL
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| BDBM167458 |
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| n/a |
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| Name | BDBM167458 |
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| Synonyms: | US9073911, 7 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H22N4O3 |
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| Mol. Mass. | 378.4244 |
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| SMILES | COc1ccc(cc1)-c1cc([nH]n1)C(=O)Nc1ccc(cc1)[C@H]1CNCCO1 |r| |
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| Structure | 
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