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TargetOpioid growth factor receptor-like protein 1
LigandBDBM172382
Substrate/Competitorn/a
Meas. Tech.Radioligand Binding Assay
pH7.4±n/a
Temperature298.15±n/a K
Ki 1.9±0.4 nM
Commentsextracted
Citation Yamawaki, KYao, JYu, JZhou, X Substituted benzimidazole-type piperidine compounds and uses thereof US Patent US9090618 Publication Date 7/28/2015
More Info.:Get all data from this article,  Assay Method
 
Opioid growth factor receptor-like protein 1
Name:Opioid growth factor receptor-like protein 1
Synonyms:OGFRL1 | OGRL1_HUMAN | Opioid Receptor-Like Receptor (ORL-1) | Opioid growth factor receptor-like protein 1 (ORL-1) | Opioid growth factor receptor-like protein 1 (ORL1) | Opioid receptor-like (ORL-1) | Opioid receptor-like (ORL1) | Opioid receptor-like protein 1 (OGL1) | Opioid receptor-like receptor (ORL1)
Type:Protein
Mol. Mass.:51247.53
Organism:Homo sapiens (Human)
Description:Q5TC84
Residue:451
Sequence:
MGNLLGGVSFREPTTVEDCDSTWQTDSEPEPEEPGPGGGSEGPGQESEQPAQPPEQAGGR
PGASPAPDEDAEAAGAEQGGDSTEATAKPKRSFYAARDLYKYRHQYPNFKDIRYQNDLSN
LRFYKNKIPFKPDGVYIEEVLSKWKGDYEKLEHNHTYIQWLFPLREQGLNFYAKELTTYE
IEEFKKTKEAIRRFLLAYKMMLEFFGIKLTDKTGNVARAVNWQERFQHLNESQHNYLRIT
RILKSLGELGYESFKSPLVKFILHEALVENTIPNIKQSALEYFVYTIRDRRERRKLLRFA
QKHYTPSENFIWGPPRKEQSEGSKAQKMSSPLASSHNSQTSMHKKAKDSKNSSSAVHLNS
KTAEDKKVAPKEPVEETDRPSPEPSNEAAKPRNTEKDSNAENMNSQPEKTVTTPTEKKES
VSPENNEEGGNDNQDNENPGNTNCHDVVLVQ
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  Blast E-value cutoff:
BDBM172382
n/a
NameBDBM172382
Synonyms:US9090618, H27b(i) | US9598411, Ref. No. H27b(i)
TypeSmall organic molecule
Emp. Form.C29H42N4
Mol. Mass.446.6706
SMILESC1CNC(C1)c1nc2ccccc2n1[C@@H]1C[C@@H]2CCC[C@H](C1)N2[C@H]1C[C@@H]2C[C@H](C1)CCCC2 |r,THB:23:22:14.15.21:17.19.18|
Structure
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