| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Opioid growth factor receptor-like protein 1 |
|---|
| Ligand | BDBM172438 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Radioligand Binding Assay |
|---|
| pH | 7.4±n/a |
|---|
| Temperature | 298.15±n/a K |
|---|
| Ki | 3.8±0.7 nM |
|---|
| Comments | extracted |
|---|
| Citation |  Yamawaki, K; Yao, J; Yu, J; Zhou, X Substituted benzimidazole-type piperidine compounds and uses thereof US Patent US9090618 Publication Date 7/28/2015 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Opioid growth factor receptor-like protein 1 |
|---|
| Name: | Opioid growth factor receptor-like protein 1 |
|---|
| Synonyms: | OGFRL1 | OGRL1_HUMAN | Opioid Receptor-Like Receptor (ORL-1) | Opioid growth factor receptor-like protein 1 (ORL-1) | Opioid growth factor receptor-like protein 1 (ORL1) | Opioid receptor-like (ORL-1) | Opioid receptor-like (ORL1) | Opioid receptor-like protein 1 (OGL1) | Opioid receptor-like receptor (ORL1) |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 51247.53 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | Q5TC84 |
|---|
| Residue: | 451 |
|---|
| Sequence: | MGNLLGGVSFREPTTVEDCDSTWQTDSEPEPEEPGPGGGSEGPGQESEQPAQPPEQAGGR
PGASPAPDEDAEAAGAEQGGDSTEATAKPKRSFYAARDLYKYRHQYPNFKDIRYQNDLSN
LRFYKNKIPFKPDGVYIEEVLSKWKGDYEKLEHNHTYIQWLFPLREQGLNFYAKELTTYE
IEEFKKTKEAIRRFLLAYKMMLEFFGIKLTDKTGNVARAVNWQERFQHLNESQHNYLRIT
RILKSLGELGYESFKSPLVKFILHEALVENTIPNIKQSALEYFVYTIRDRRERRKLLRFA
QKHYTPSENFIWGPPRKEQSEGSKAQKMSSPLASSHNSQTSMHKKAKDSKNSSSAVHLNS
KTAEDKKVAPKEPVEETDRPSPEPSNEAAKPRNTEKDSNAENMNSQPEKTVTTPTEKKES
VSPENNEEGGNDNQDNENPGNTNCHDVVLVQ
|
|
|
|---|
| BDBM172438 |
|---|
| n/a |
|---|
| Name | BDBM172438 |
|---|
| Synonyms: | US9090618, ZA61 | US9598411, Ref. No. ZA61 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C29H40N6 |
|---|
| Mol. Mass. | 472.6681 |
|---|
| SMILES | Cc1nnc(Cc2nc3ccccc3n2[C@@H]2C[C@@H]3CCC[C@H](C2)N3[C@H]2C[C@@H]3C[C@H](C2)CCCC3)[nH]1 |r,THB:24:23:15.16.22:18.20.19| |
|---|
| Structure | 
|
|---|
Search and Browse
