| Reaction Details |
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 | Report a problem with these data |
| Target | Prolactin-releasing peptide receptor |
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| Ligand | BDBM195657 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Inhibition Assay |
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| pH | 7.4±n/a |
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| Temperature | 298.15±n/a K |
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| Ki | 7±n/a nM |
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| Comments | extracted |
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| Citation |  Takahashi, A; Suzuki, M; Nakamura, Y; Sakurai, Y Heterocyclic compounds for the treatment of stress-related conditions US Patent US9206173 Publication Date 12/8/2015 |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Prolactin-releasing peptide receptor |
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| Name: | Prolactin-releasing peptide receptor |
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| Synonyms: | G-protein coupled receptor 10 (GPR10) | GPR10 | GR3 | PRLHR | PRLHR_HUMAN | Prolactin Releasing Peptide Receptor | Prolactin-releasing peptide receptor |
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| Type: | Protein |
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| Mol. Mass.: | 41138.32 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P49683 |
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| Residue: | 370 |
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| Sequence: | MASSTTRGPRVSDLFSGLPPAVTTPANQSAEASAGNGSVAGADAPAVTPFQSLQLVHQLK
GLIVLLYSVVVVVGLVGNCLLVLVIARVRRLHNVTNFLIGNLALSDVLMCTACVPLTLAY
AFEPRGWVFGGGLCHLVFFLQPVTVYVSVFTLTTIAVDRYVVLVHPLRRRISLRLSAYAV
LAIWALSAVLALPAAVHTYHVELKPHDVRLCEEFWGSQERQRQLYAWGLLLVTYLLPLLV
ILLSYVRVSVKLRNRVVPGCVTQSQADWDRARRRRTFCLLVVIVVVFAVCWLPLHVFNLL
RDLDPHAIDPYAFGLVQLLCHWLAMSSACYNPFIYAWLHDSFREELRKLLVAWPRKIAPH
GQNMTVSVVI
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| BDBM195657 |
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| n/a |
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| Name | BDBM195657 |
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| Synonyms: | US9206173, 2419 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H26F3N5O5 |
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| Mol. Mass. | 533.4996 |
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| SMILES | COc1ccc(C(=O)N2CCc3nc(NC(C)c4ccc(cc4)C(F)(F)F)n(OC)c(=O)c3C2)c(OC)n1 |
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| Structure | 
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