Compile Data Set for Download or QSAR
Found 132 with Last Name = 'zeslawska' and Initial = 'e'
TargetSerine protease 1(Bos taurus (bovine))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM16175(CHEMBL108468 | UKI-1 | ethyl 4-(3-carbamimidoyl-N-...)copy SMILEScopy InChI
Affinity DataKi:  37nM ΔG°:  -42.4kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445JRMPubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM16175(CHEMBL108468 | UKI-1 | ethyl 4-(3-carbamimidoyl-N-...)copy SMILEScopy InChI
Affinity DataKi:  410nM ΔG°:  -36.5kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445JRMPubMed
TargetSerine protease 1(Bos taurus (bovine))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM16174(3-[3-(4-beta-alanylpiperazin-1-yl)-3-oxo-2-({[2,4,...)copy SMILEScopy InChI
Affinity DataKi:  600nM ΔG°:  -35.5kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445JRMPubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM16174(3-[3-(4-beta-alanylpiperazin-1-yl)-3-oxo-2-({[2,4,...)copy SMILEScopy InChI
Affinity DataKi:  640nM ΔG°:  -35.4kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM16176(3-(1-adamantyl)-1-[(4-carbamimidamidophenyl)methyl...)copy SMILEScopy InChI
Affinity DataKi:  2.40E+3nM ΔG°:  -32.1kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM16175(CHEMBL108468 | UKI-1 | ethyl 4-(3-carbamimidoyl-N-...)copy SMILEScopy InChI
Affinity DataKi:  4.90E+3nM ΔG°:  -30.3kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445JRMPubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM16173(3,5-diamino-6-chloro-N-(diaminomethylene)pyrazinam...)copy SMILEScopy InChI
Affinity DataKi:  5.30E+3nM ΔG°:  -30.1kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM16174(3-[3-(4-beta-alanylpiperazin-1-yl)-3-oxo-2-({[2,4,...)copy SMILEScopy InChI
Affinity DataKi:  8.70E+3nM ΔG°:  -28.9kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445JRMPubMed
TargetSerine protease 1(Bos taurus (bovine))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM16173(3,5-diamino-6-chloro-N-(diaminomethylene)pyrazinam...)copy SMILEScopy InChI
Affinity DataKi:  3.20E+4nM ΔG°:  -25.7kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445JRMPubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM50223724(2-(4-guanidynephenyl)-1-phenyl-ethanone | CHEMBL23...)copy SMILEScopy InChI
Affinity DataKi:  3.40E+4nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V987T5PubMed
TargetSerine protease 1(Bos taurus (bovine))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM772(Benzamidine | CHEMBL79897 | [amino(phenyl)methylid...)copy SMILEScopy InChI
Affinity DataKi:  3.90E+4nM ΔG°:  -25.2kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM16176(3-(1-adamantyl)-1-[(4-carbamimidamidophenyl)methyl...)copy SMILEScopy InChI
Affinity DataKi:  4.60E+4nM ΔG°:  -24.8kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445JRMPubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM772(Benzamidine | CHEMBL79897 | [amino(phenyl)methylid...)copy SMILEScopy InChI
Affinity DataKi:  1.80E+5nM ΔG°:  -21.4kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM16176(3-(1-adamantyl)-1-[(4-carbamimidamidophenyl)methyl...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nM ΔG°: >-17.1kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445JRMPubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM16173(3,5-diamino-6-chloro-N-(diaminomethylene)pyrazinam...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nM ΔG°: >-17.1kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445JRMPubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM50223724(2-(4-guanidynephenyl)-1-phenyl-ethanone | CHEMBL23...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of tPAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V987T5PubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Max-Planck-Institut fuer Biochemie

LigandPNGBDBM772(Benzamidine | CHEMBL79897 | [amino(phenyl)methylid...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nM ΔG°: >-17.1kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445JRMPubMedMMDB
TargetEndothelin receptor type B(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50155245(CHEMBL3774897)copy SMILEScopy InChI
Affinity DataIC50: 0.00600nMAssay Description:Displacement of [125I]Endothelin-1 from human recombinant Endothelin-B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50208985(CHEMBL3885244)copy SMILEScopy InChI
Affinity DataIC50: 0.00600nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETB receptor expressed in CHO cells measured after 120 mins by scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM22567(3H]pyrilamine | CHEMBL511 | Dorantamin | Mepyramin...)copy SMILEScopy InChI
Affinity DataIC50: 0.0140nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMedDrugBank
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50155248(CHEMBL3774478)copy SMILEScopy InChI
Affinity DataIC50: 0.0160nMAssay Description:Displacement of [125I]apamin from rat cerebral cortex small conductance calcium-activated potassium channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50155246(CHEMBL3775234)copy SMILEScopy InChI
Affinity DataIC50: 0.0230nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETA receptor expressed in CHO cells measured after 120 mins by scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50155246(CHEMBL3775234)copy SMILEScopy InChI
Affinity DataIC50: 0.0230nMAssay Description:Displacement of [125I]Endothelin-1 from human recombinant Endothelin-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50208988(HUMAN NEUROPEPTIDE Y)copy SMILEScopy InChI
Affinity DataIC50: 0.0280nMAssay Description:Displacement of [125I]peptide YY from Y2 receptor in human KAN-TS cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50208986(CHEMBL3883526)copy SMILEScopy InChI
Affinity DataIC50: 0.0320nMAssay Description:Displacement of [125I]hCGRPa from human recombinant CGRP receptor expressed in CHO cells measured after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50250019(CHEMBL524658 | PACAP | PACAP(1-38) | PACAP-38 | PA...)copy SMILEScopy InChI
Affinity DataIC50: 0.0400nMAssay Description:Displacement of [125I]PACAP1-27 from human recombinant PAC1 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetMelatonin receptor type 1B(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)copy SMILEScopy InChI
Affinity DataIC50: 0.0740nMAssay Description:Displacement of [125I]Tyr11-somatostatin-14 from somatostatin receptor in mouse AtT20 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50208989(CHEMBL506553)copy SMILEScopy InChI
Affinity DataIC50: 0.0790nMAssay Description:Displacement of [125I]galanin from human recombinant GAL1 receptor expressed in HEK293 cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)copy SMILEScopy InChI
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125I]CGP 42112A from human recombinant AT2 receptor expressed in HEK293 cells measured after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50155247(CHEMBL385433)copy SMILEScopy InChI
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125I]CGP42112A from human recombinant AT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in CHO cells measured after 60 mins by scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMedDrugBank
TargetSubstance-P receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50335566(CHEMBL1651026 | Substance P [Sar9,Met(O2)11])copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]BH-SP from NK1 receptor in human U373MG cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50435130(CHEMBL1893324)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]VIP from human recombinant VIP1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant ML1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMedDrugBank
TargetSubstance-P receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50335566(CHEMBL1651026 | Substance P [Sar9,Met(O2)11])copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]BH-SP from NK1 receptor in human U373MG cells measured after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50208990(CHEMBL3884667)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]VIP from human recombinant VPAC1 receptor expressed in CHO cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)copy SMILEScopy InChI
Affinity DataIC50: 0.120nMAssay Description:Displacement of [125I]CCK-8s from human recombinant CCK-B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)copy SMILEScopy InChI
Affinity DataIC50: 0.120nMAssay Description:Displacement of [125I]CCK-8s from human recombinant CCK2 receptor expressed in CHO cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)copy SMILEScopy InChI
Affinity DataIC50: 0.130nMAssay Description:Displacement of [125I]CCK-8s from human recombinant CCK1 receptor expressed in CHO cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)copy SMILEScopy InChI
Affinity DataIC50: 0.130nMAssay Description:Displacement of [125I]CCK-8s from human recombinant CCK-A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 0.150nMAssay Description:Displacement of [125I]NDP-a-MSH from human recombinant MC4 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 0.150nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human recombinant MC4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50208988(HUMAN NEUROPEPTIDE Y)copy SMILEScopy InChI
Affinity DataIC50: 0.210nMAssay Description:Displacement of [125I]peptide YY from Y1 receptor in human SK-N-MC cells measured after 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataIC50: 0.25nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataIC50: 0.25nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM86180(CAS_87075-17-0 | NSC_5018 | SCH 23390 | SCH23390 |...)copy SMILEScopy InChI
Affinity DataIC50: 0.310nMAssay Description:Displacement of [3H]SCH23390 from human recombinant Dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM86180(CAS_87075-17-0 | NSC_5018 | SCH 23390 | SCH23390 |...)copy SMILEScopy InChI
Affinity DataIC50: 0.310nMAssay Description:Displacement of [3H]SCH 23390 from human recombinant dopamine D1 receptor expressed in CHO cells measured after 60 mins by scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50176065(4-DAMP | 4-Diphenylacetoxy-1,1-dimethyl-piperidini...)copy SMILEScopy InChI
Affinity DataIC50: 0.320nMAssay Description:Displacement of [3H]4-DAMP from human recombinant muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50176065(4-DAMP | 4-Diphenylacetoxy-1,1-dimethyl-piperidini...)copy SMILEScopy InChI
Affinity DataIC50: 0.320nMAssay Description:Displacement of [3H]4-DAMP from human recombinant M5 receptor expressed in CHO cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)copy SMILEScopy InChI
Affinity DataIC50: 0.350nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5-HT2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
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