TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£rzburg
Curated by ChEMBL
Julius Maximilian University of W£rzburg
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]-Diprenorphine from human mu opioid receptor expressed in HEK293-TSA cell membranes after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.09nMAssay Description:Displacement of [3H]mepyramine from human H1R expressed in Sf9 cells co-expressing RGS4 after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in human SK-N-MC cells incubated for 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.47nMAssay Description:Displacement of [3H]mepyramine from human H1R expressed in Sf9 cells co-expressing RGS4 after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Affinity DataKi: 4.90nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in HEK293T cell membranes incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]mepyramine from human H1R expressed in Sf9 cells co-expressing RGS4 after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£rzburg
Curated by ChEMBL
Julius Maximilian University of W£rzburg
Curated by ChEMBL
Affinity DataKi: 5.60nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 7.08nMAssay Description:Displacement of [3H]mepyramine from human H1R expressed in Sf9 cells co-expressing RGS4 after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Displacement of [3H]mepyramine from human histamine 1 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in human SK-N-MC cell membrane incubated for 60 minsMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in human SK-N-MC cell membrane incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 14.8nMAssay Description:Displacement of [3H]mepyramine from human H1R expressed in Sf9 cells co-expressing RGS4 after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in human SK-N-MC cell membrane incubated for 60 minsMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Affinity DataKi: 18.6nMAssay Description:Displacement of [3H]histamine from human H4R expressed in Sf9 cells co-expressing RGS19, Galphai2 and Gbeta1gamma2 after 60 mins by liquid scintillat...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£rzburg
Curated by ChEMBL
Julius Maximilian University of W£rzburg
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Binding affinity to histamine 4 receptor (unknown origin)More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£rzburg
Curated by ChEMBL
Julius Maximilian University of W£rzburg
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Affinity DataKi: 69nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in sf9 cells co-expressing mammalian Galphai2 and Gbeta1gamma2More data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Affinity DataKi: 99nMAssay Description:Displacement of [3H]UR-PI294 from human histamine H4 receptor expressed in sf9 cell membrane co-expressing mammalian Galphai2 and Gbeta1gamma2 incuba...More data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Affinity DataKi: 99nMAssay Description:Displacement of [3H]UR-PI294 from human histamine H4 receptor expressed in sf9 cell membrane co-expressing mammalian Galphai2 and Gbeta1gamma2 incuba...More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [3H]mepyramine from human H1R expressed in Sf9 cells co-expressing RGS4 after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£t Erlangen-N£rnberg
Curated by ChEMBL
Affinity DataKi: 102nMAssay Description:Displacement of [3H]histamine from human histamine 4 receptor expressed in Sf9 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
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