Compile Data Set for Download or QSAR
Found 426 with Last Name = 'celeridad' and Initial = 'm'
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50364378(CHEMBL1950289)copy SMILEScopy InChI
Affinity DataKi:  6.20nMAssay Description:Inhibition of hexa-His-tagged JNK2 expressed in baculoviral system using GST-tagged cJun as substrate preincubated for 15 mins prior ATP addition mea...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829SKPubMed
TargetSerine/threonine-protein kinase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50583973(CHEMBL5093114)copy SMILES
Affinity DataKi:  33nMAssay Description:Binding affinity to recombinant N-terminal His6-tagged human STK4 (43 to 431 residues) expressed in Escherichia coli assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52TH8PubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50364378(CHEMBL1950289)copy SMILEScopy InChI
Affinity DataKi:  44nMAssay Description:Inhibition of hexa-His-tagged JNK1 expressed in baculoviral system using GST-tagged c-Jun as substrate preincubated for 15 mins prior ATP addition me...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50059345(CHEMBL3393355 | US9156845, 83)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Binding affinity to recombinant N-terminal His6-tagged human STK4 (43 to 431 residues) expressed in Escherichia coli assessed as inhibition constantMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50059345(CHEMBL3393355 | US9156845, 83)copy SMILEScopy InChI
Affinity DataKi:  89nMAssay Description:Binding affinity to recombinant N-terminal His6-tagged human STK3 (18 to 311 residues) expressed in Escherichia coli assessed as inhibition constantMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 4(Homo sapiens (Human))TBA
LigandPNGBDBM185556(US9156845, 215)copy SMILEScopy InChI
Affinity DataKi:  96nMAssay Description:Binding affinity to recombinant N-terminal His6-tagged human STK4 (43 to 431 residues) expressed in Escherichia coli assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52TH8PubMed
TargetSerine/threonine-protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM185556(US9156845, 215)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Binding affinity to recombinant N-terminal His6-tagged human STK3 (18 to 311 residues) expressed in Escherichia coli assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52TH8PubMed
TargetSerine/threonine-protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50583973(CHEMBL5093114)copy SMILES
Affinity DataKi:  211nMAssay Description:Binding affinity to recombinant N-terminal His6-tagged human STK3 (18 to 311 residues) expressed in Escherichia coli assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52TH8PubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM251460(US9452998, 9)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573043(CHEMBL4849510)copy SMILES
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573038(CHEMBL4853353)copy SMILES
Affinity DataIC50: 1.40nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))TBA
LigandPNGBDBM251460(US9452998, 9)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of PKC-alpha (unknown origin)More data for this Ligand-Target Pair
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573042(CHEMBL4854104)copy SMILES
Affinity DataIC50: 2.20nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379404(6-((4-(cyclopropylamino)-5-(trifluoromethyl)pyrimi...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50572994(CHEMBL4854326)copy SMILES
Affinity DataIC50: 4nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573034(CHEMBL4859091)copy SMILES
Affinity DataIC50: 4nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379381(N4-cyclopropyl-N2-(quinolin-6-yl)-5-(trifluorometh...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379329(N2-(1H-benzo[d]imidazol-6-yl)-N4-cyclopropyl-5-(tr...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573033(CHEMBL4851695)copy SMILES
Affinity DataIC50: 6nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379305(N2-(1H-benzo[d][1,2,3]triazol-6-yl)-N4-cyclopropyl...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50364378(CHEMBL1950289)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of hexa-His-tagged JNK3 expressed in baculoviral system using GST-tagged cJun as substrate preincubated for 15 mins prior ATP addition mea...More data for this Ligand-Target Pair
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573029(CHEMBL4861883)copy SMILES
Affinity DataIC50: 7nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573015(CHEMBL4870774)copy SMILES
Affinity DataIC50: 7nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379307(N4-cyclopropyl-N2-(3,4-dihydro-2H-benzo[b][1,4]dio...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50364378(CHEMBL1950289)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of hexa-His-tagged JNK2 expressed in baculoviral system using GST-tagged cJun as substrate preincubated for 15 mins prior ATP addition mea...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829SKPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50364377(CHEMBL1950304)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of hexa-His-tagged JNK3 expressed in baculoviral system using GST-tagged cJun as substrate preincubated for 15 mins prior ATP addition mea...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829SKPubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573044(CHEMBL4873647)copy SMILES
Affinity DataIC50: 8nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50363465(CHEMBL1946646)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of full length Hexa-His-tagged JNK2 using GST-tagged cJun and [gamma33P]ATP as substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZP6PubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50363455(CHEMBL1946333)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of full length Hexa-His-tagged JNK2 using GST-tagged cJun and [gamma33P]ATP as substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZP6PubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50364377(CHEMBL1950304)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of hexa-His-tagged JNK2 expressed in baculoviral system using GST-tagged cJun as substrate preincubated for 15 mins prior ATP addition mea...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829SKPubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50363466(CHEMBL1946647)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of full length Hexa-His-tagged JNK2 using GST-tagged cJun and [gamma33P]ATP as substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZP6PubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573027(CHEMBL4867906)copy SMILES
Affinity DataIC50: 12nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50363455(CHEMBL1946333)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of full length Hexa-His-tagged JNK3 using GST-tagged cJun and [gamma33P]ATP as substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZP6PubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379414(N-(4-((4-(cyclopropylamino)-5-(trifluoromethyl)pyr...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379408(N4-cyclopropyl-N2-(quinoxalin-6-yl)-5-(trifluorome...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379450(US10266549, Example 349 | US10774092, Example 349)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50363465(CHEMBL1946646)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of full length Hexa-His-tagged JNK3 using GST-tagged cJun and [gamma33P]ATP as substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZP6PubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379352(N4-cyclopropyl-N2-(5-methoxypyridin-3-yl)-5-(trifl...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50363462(CHEMBL1946340)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of full length Hexa-His-tagged JNK2 using GST-tagged cJun and [gamma33P]ATP as substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZP6PubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379259(US10266549, Example 158a | US10774092, Example 158...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379311(N4-cyclopropyl-N2-(1H-indazol-5-yl)-5-(trifluorome...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50363466(CHEMBL1946647)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of full length Hexa-His-tagged JNK3 using GST-tagged cJun and [gamma33P]ATP as substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZP6PubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379387(N4-cyclopropyl-N2-(quinolin-3-yl)-5-(trifluorometh...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379264(US10266549, Example 161a | US10774092, Example 161...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50363462(CHEMBL1946340)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of full length Hexa-His-tagged JNK3 using GST-tagged cJun and [gamma33P]ATP as substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZP6PubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379325(US10266549, Example 208a | US10774092, Example 208...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573014(CHEMBL4858914)copy SMILES
Affinity DataIC50: 20nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573028(CHEMBL4856779)copy SMILES
Affinity DataIC50: 20nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379406(US10266549, Example 304a | US10774092, Example 304...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))TBA
LigandPNGBDBM379332(N2-(benzo[d][1,3]dioxol-5-yl)-N4-cyclopropyl-5-(tr...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K0JPubMed
Displayed 1 to 50 (of 426 total ) | Next | Last >>
Jump to: