Compile Data Set for Download or QSAR
Found 26 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50001136
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269944(CHEMBL4081970)copy SMILEScopy InChI
Affinity DataEC50:  13nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269967(CHEMBL4096184)copy SMILEScopy InChI
Affinity DataEC50:  4.30nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269946(CHEMBL4071437)copy SMILEScopy InChI
Affinity DataEC50:  6.30nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269947(CHEMBL4062799)copy SMILEScopy InChI
Affinity DataEC50:  10nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269949(CHEMBL4074175)copy SMILEScopy InChI
Affinity DataEC50:  14nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269950(CHEMBL4100932)copy SMILEScopy InChI
Affinity DataEC50:  9.30nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269970(CHEMBL4065552)copy SMILEScopy InChI
Affinity DataEC50:  6.30nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269953(CHEMBL4103468)copy SMILEScopy InChI
Affinity DataEC50:  5nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269954(CHEMBL4077689)copy SMILEScopy InChI
Affinity DataEC50:  10nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269980(CHEMBL4095707)copy SMILEScopy InChI
Affinity DataEC50:  11nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269955(CHEMBL4066696)copy SMILEScopy InChI
Affinity DataEC50:  10nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269957(CHEMBL4068478)copy SMILEScopy InChI
Affinity DataEC50:  3.70nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269981(CHEMBL4090653)copy SMILEScopy InChI
Affinity DataEC50:  4.90nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269958(CHEMBL4076985)copy SMILEScopy InChI
Affinity DataEC50:  3.70nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269960(CHEMBL4076150)copy SMILEScopy InChI
Affinity DataEC50:  4nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269983(CHEMBL4070119)copy SMILEScopy InChI
Affinity DataEC50:  5.80nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269964(CHEMBL4077479)copy SMILEScopy InChI
Affinity DataEC50:  5.20nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269968(CHEMBL4087877)copy SMILEScopy InChI
Affinity DataEC50:  6.60nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269969(CHEMBL4060368)copy SMILEScopy InChI
Affinity DataEC50:  3.5nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269951(CHEMBL4069649)copy SMILEScopy InChI
Affinity DataEC50:  7.80nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269988(CHEMBL4099974)copy SMILEScopy InChI
Affinity DataEC50:  10nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269989(CHEMBL4084476)copy SMILEScopy InChI
Affinity DataEC50:  20nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269956(CHEMBL4087993)copy SMILEScopy InChI
Affinity DataEC50:  20nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269952(CHEMBL4085539)copy SMILEScopy InChI
Affinity DataEC50:  4nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269959(CHEMBL4064003)copy SMILEScopy InChI
Affinity DataEC50:  15nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269945(CHEMBL4092221)copy SMILEScopy InChI
Affinity DataEC50:  8.5nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed