Compile Data Set for Download or QSAR
Found 6 Enz. Inhib. hit(s) with Target = 'Urotensin-2 receptor' and Ligand = 'BDBM50269950'
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269950(CHEMBL4100932)copy SMILEScopy InChI
Affinity DataEC50:  17nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(RAT)
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269950(CHEMBL4100932)copy SMILEScopy InChI
Affinity DataEC50:  9.30nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269950(CHEMBL4100932)copy SMILEScopy InChI
Affinity DataEC50:  2.19E+3nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in human urotensin-2-induced G12 activation by measu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269950(CHEMBL4100932)copy SMILEScopy InChI
Affinity DataEC50:  14nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in human urotensin-2-induced Gq activation by measur...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269950(CHEMBL4100932)copy SMILEScopy InChI
Affinity DataEC50:  4.20nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in URP-induced Gq activation by measuring URP pEC50 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Universit£ de Montr£al

Curated by ChEMBL
LigandPNGBDBM50269950(CHEMBL4100932)copy SMILEScopy InChI
Affinity DataEC50:  117nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in URP-induced G12 activation by measuring URP pEC50...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V1279DPubMed