Compile Data Set for Download or QSAR
Found 63 of ic50 data for polymerid = 49001048,49001049
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50013027(CHEMBL262655 | Sodium; 3-[4-(4-chloro-benzenesulfo...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70FQG
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075089(CHEMBL133420 | Sodium; [2-(4-chloro-benzenesulfony...)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075088(CHEMBL336846 | Sodium; {2-[(4-chloro-benzenesulfon...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353639(CHEMBL1829806)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353632(CHEMBL1829812)copy SMILEScopy InChI
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353635(CHEMBL1829801)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353643(CHEMBL1829808)copy SMILEScopy InChI
Affinity DataIC50: 9.40nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075086(CHEMBL341221 | Sodium; [2-(benzenesulfonylamino-me...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075091(CHEMBL131894 | Sodium; 3-{2-[(4-chloro-benzenesulf...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353645(CHEMBL1829810)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075077(CHEMBL131497 | Sodium; {2-[(naphthalene-2-sulfonyl...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075082(CHEMBL264516 | Sodium; 2-[(4-chloro-benzenesulfony...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353640(CHEMBL65121)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075094(CHEMBL132659 | Sodium; {2-[2-(4-chloro-benzenesulf...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075093(CHEMBL130377 | Sodium; 5-{2-[(4-chloro-benzenesulf...)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50002805((daltroban){4-[2-(4-Chloro-benzenesulfonylamino)-e...)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075079(CHEMBL334501 | Sodium; 4-{2-[(4-chloro-benzenesulf...)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353638(CHEMBL1829805)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075096(CHEMBL336352 | Sodium; 2-[2-(4-chloro-benzenesulfo...)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075092(CHEMBL339994 | Sodium; 2-[3-(4-chloro-benzenesulfo...)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075076(CHEMBL335043 | Sodium; {2-[(thiophene-2-sulfonylam...)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353636(CHEMBL1829802)copy SMILEScopy InChI
Affinity DataIC50: 91nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075085(CHEMBL131036 | Sodium; {2-[(4-chloro-benzenesulfon...)copy SMILEScopy InChI
Affinity DataIC50: 141nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282138(CHEMBL298462 | Sodium; 3-[4-(4-chloro-phenylsulfam...)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70FQG
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353646(CHEMBL1829811)copy SMILEScopy InChI
Affinity DataIC50: 259nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075090(CHEMBL422441 | Sodium; {2-[(naphthalene-1-sulfonyl...)copy SMILEScopy InChI
Affinity DataIC50: 295nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353644(CHEMBL1829809)copy SMILEScopy InChI
Affinity DataIC50: 463nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075081(CHEMBL130045 | Sodium; 2-[4-(4-chloro-benzenesulfo...)copy SMILEScopy InChI
Affinity DataIC50: 479nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075084(CHEMBL130170 | Sodium; {2-[3-(4-chloro-benzenesulf...)copy SMILEScopy InChI
Affinity DataIC50: 513nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282141(CHEMBL46338 | Sodium; 3-[5-(4-chloro-phenylsulfamo...)copy SMILEScopy InChI
Affinity DataIC50: 860nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70FQG
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282135(CHEMBL430569 | Sodium; 3-[3-(4-chloro-phenylsulfam...)copy SMILEScopy InChI
Affinity DataIC50: 860nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70FQG
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075095(CHEMBL131336 | Sodium; {2-[4-(4-chloro-benzenesulf...)copy SMILEScopy InChI
Affinity DataIC50: 977nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075080(CHEMBL130460 | Sodium; [2-(cyclohexanesulfonylamin...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353641(CHEMBL1829804)copy SMILEScopy InChI
Affinity DataIC50: 1.23E+3nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075083(CHEMBL340073 | Sodium; {2-[(pentane-1-sulfonylamin...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282152(CHEMBL47605 | Sodium; 6-isopropyl-3-(5-phenylsulfa...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70FQG
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282146(CHEMBL48013 | Sodium; 6-isopropyl-3-(4-phenylsulfa...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70FQG
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282136(6-Isopropyl-3-(5-phenylsulfamoyl-pentyl)-azulene-1...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70FQG
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50002765(BM 13177 | BM-13177 | CHEMBL8273 | Sulotroban | [4...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70FQG
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353634(CHEMBL1828642)copy SMILEScopy InChI
Affinity DataIC50: 1.63E+3nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282156(3-[5-(4-Chloro-phenylsulfamoyl)-pentyl]-6-isopropy...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70FQG
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353642(CHEMBL1829807)copy SMILEScopy InChI
Affinity DataIC50: 1.79E+3nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075087(CHEMBL134128 | Sodium; {2-[(pyridine-3-sulfonylami...)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353633(CHEMBL1829813)copy SMILEScopy InChI
Affinity DataIC50: 2.52E+3nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282139(3-[4-(4-Chloro-phenylsulfamoyl)-butyl]-6-isopropyl...)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70FQG
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50075078(CHEMBL132573 | Sodium; [2-(phenylmethanesulfonylam...)copy SMILEScopy InChI
Affinity DataIC50: 5.90E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB2363PubMed
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282133(CHEMBL47510 | Sodium; 6-isopropyl-3-(3-phenylsulfa...)copy SMILEScopy InChI
Affinity DataIC50: 8.70E+3nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70FQG
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282154(6-Isopropyl-3-(4-phenylsulfamoyl-butyl)-azulene-1-...)copy SMILEScopy InChI
Affinity DataIC50: 8.70E+3nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70FQG
TargetThromboxane A2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282147(3-[3-(4-Chloro-phenylsulfamoyl)-propyl]-6-isopropy...)copy SMILEScopy InChI
Affinity DataIC50: 9.10E+3nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70FQG
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353637(CHEMBL1829803)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
Displayed 1 to 50 (of 63 total ) | Next | Last >>
Jump to: