Compile Data Set for Download or QSAR
Found 225 of ic50 data for polymerid = 5183
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420761(CHEMBL2087507)copy SMILEScopy InChI
Affinity DataIC50: 0.640nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420769(CHEMBL2087515)copy SMILEScopy InChI
Affinity DataIC50: 0.830nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420767(CHEMBL2087513)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420746(CHEMBL2087524)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420763(CHEMBL2087509)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420756(CHEMBL2087501)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420758(CHEMBL2087503)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420747(CHEMBL2087526)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50296636(4-chloro-N-cyclopropyl-3-(1-(4-fluorophenyl)-7-met...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of p38deltaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7NT0PubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM563647(N-(4-{4-[3-(5-tert-Butyl-2- methyl-2H-pyrazol-3-yl...)copy SMILES
Affinity DataIC50: 6nMAssay Description:ach of these analogs were checked for physical chemical characteristics based on molecular weight, Lipinski's Rule of 5, partition coefficient (l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FN19DPUS Patent
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420740(CHEMBL2087742)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420766(CHEMBL2087512)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420749(CHEMBL2087743)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420773(CHEMBL2087505)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM563618(N-[4-[2-[2-[[5-tert-butyl-2-(p- tolyl)pyrazol-3- y...)copy SMILES
Affinity DataIC50: 8nMAssay Description:ach of these analogs were checked for physical chemical characteristics based on molecular weight, Lipinski's Rule of 5, partition coefficient (l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FN19DPUS Patent
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM563619(N-[4-[2-[2-[[5-tert-butyl-2-(p- tolyl)pyrazol-3- y...)copy SMILES
Affinity DataIC50: 9nMAssay Description:ach of these analogs were checked for physical chemical characteristics based on molecular weight, Lipinski's Rule of 5, partition coefficient (l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FN19DPUS Patent
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM563649(N-(4-{4-[3-(5-tert-Butyl-isoxazol- 3-yl)-ureido]-3...)copy SMILES
Affinity DataIC50: 9nMAssay Description:ach of these analogs were checked for physical chemical characteristics based on molecular weight, Lipinski's Rule of 5, partition coefficient (l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FN19DPUS Patent
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420744(CHEMBL2087522)copy SMILEScopy InChI
Affinity DataIC50: 9.40nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420750(CHEMBL2087744)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM563612(Cyclopropanecarboxylic acid [4- (2-{2-[3-(5-tert-b...)copy SMILES
Affinity DataIC50: 11nMAssay Description:ach of these analogs were checked for physical chemical characteristics based on molecular weight, Lipinski's Rule of 5, partition coefficient (l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FN19DPUS Patent
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50396845(CHEMBL2170294)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of human MAPK p38alpha by Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN67XZPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM563650(N-(4-{4-[3-(3-tert-Butyl-isoxazol- 5-yl)-ureido]-3...)copy SMILES
Affinity DataIC50: 11nMAssay Description:ach of these analogs were checked for physical chemical characteristics based on molecular weight, Lipinski's Rule of 5, partition coefficient (l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FN19DPUS Patent
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420752(CHEMBL2087746)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420760(CHEMBL2087506)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420754(CHEMBL2087499)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420753(CHEMBL2087747)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420743(CHEMBL2087521)copy SMILEScopy InChI
Affinity DataIC50: 15.4nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420739(CHEMBL2087500)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420774(CHEMBL2087525)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM563615(Cyclobutanecarboxylic acid [4-(2- {2-[3-(5-tert-bu...)copy SMILES
Affinity DataIC50: 18nMAssay Description:ach of these analogs were checked for physical chemical characteristics based on molecular weight, Lipinski's Rule of 5, partition coefficient (l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FN19DPUS Patent
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420771(CHEMBL2087517)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420762(CHEMBL2087508)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420751(CHEMBL2087745)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420759(CHEMBL2087504)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420757(CHEMBL2087502)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM192498(US9187470, 89)copy SMILEScopy InChI
Affinity DataIC50: 27.5nMT: 2°CAssay Description:The MAPK13 blocking activity of test compounds was determined using an immobilized metal affinity polarization (IMAP) assay containing activated MAPK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N878M9US Patent
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420765(CHEMBL2087511)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420768(CHEMBL2087514)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50536679(CHEMBL4568087)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of full-length recombinant human His-tagged MAPK13 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP27X5PubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420770(CHEMBL2087516)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420748(CHEMBL2087741)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420764(CHEMBL2087510)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50305692(3-tert-butyl-6-(2,4-difluorophenylthio)-[1,2,4]tri...)copy SMILEScopy InChI
Affinity DataIC50: 62nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 81nMAssay Description:Inhibition of human p38delta using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5KB8PubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50249406(1-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-3-(4-(py...)copy SMILEScopy InChI
Affinity DataIC50: 82.7nMT: 2°CAssay Description:The MAPK13 blocking activity of test compounds was determined using an immobilized metal affinity polarization (IMAP) assay containing activated MAPK...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420741(CHEMBL2087519)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50420742(CHEMBL2087520)copy SMILEScopy InChI
Affinity DataIC50: 102nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MNXPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50536681(CHEMBL4552628)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of full-length recombinant human His-tagged MAPK13 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP27X5PubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of human p38delta using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W380MTPubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50563891(CHEMBL4793380)copy SMILES
Affinity DataIC50: 214nMAssay Description:Inhibition of recombinant human full length SAPK4 using myelin basic protein as substrate incubated for 40 mins in presence of [gamma33P]ATP by scint...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q270854PPubMed
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