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20 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27810597 12 Structure-activity relationship studies on 1-(2-oxopropyl)indole-5-carboxylic acids acting as inhibitors of cytosolic phospholipase AEBI University of M£Nster
25102418 36 Design, synthesis, and biological evaluation of 3-(1-Aryl-1H-indol-5-yl)propanoic acids as new indole-based cytosolic phospholipase A2a inhibitors.EBI Asubio Pharma
25152071 2 Inhibition of group IVA cytosolic phospholipase A2 by thiazolyl ketones in vitro, ex vivo, and in vivo.EBI University of Athens
19327988 9 1-(5-Carboxyindol-1-yl)propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha: synthesis and properties of bioisosteric benzimidazole, benzotriazole and indazole analogues.EBI University of M£Nster
18321717 17 1-(2-Carboxyindol-5-yloxy)propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha: synthesis, biological activity, metabolic stability, and solubility.EBI University of M£Nster
20005725 61 1-Indol-1-yl-propan-2-ones and related heterocyclic compounds as dual inhibitors of cytosolic phospholipase A(2)alpha and fatty acid amide hydrolase.EBI University of M£Nster
19178292 64 Reactions of functionalized sulfonamides: application to lowering the lipophilicity of cytosolic phospholipase A2alpha inhibitors.EBI Wyeth Research
 8 Dicarboxylic acid inhibitors of phospholipase A2EBI TBA
17826099 24 Inhibitory effect of synthetic C-C biflavones on various phospholipase A(2)s activity.EBI Yeungnam University
17320401 13 1-(5-Carboxy- and 5-carbamoylindol-1-yl)propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha: bioisosteric replacement of the carboxylic acid and carboxamide moiety.EBI University of MüNster
17305324 38 Discovery of Ecopladib, an indole inhibitor of cytosolic phospholipase A2alpha.EBI Wyeth Research
16610804 39 Design and synthesis of 1-indol-1-yl-propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha.EBI University of MüNster
16545564 20 1,2,4-Oxadiazolidin-3,5-diones and 1,3,5-triazin-2,4,6-triones as cytosolic phospholipase A2alpha inhibitors.EBI Wyeth Research
16392799 46 Inhibition of cytosolic phospholipase A2alpha: hit to lead optimization.EBI Wyeth Research
14643356 32 Structure-activity relationships of indole cytosolic phospholipase A(2)alpha inhibitors: substrate mimetics.EBI Wyeth Research
10737736 19 Pyrrolidine inhibitors of human cytosolic phospholipase A(2).EBI Shionogi
30615445 64 Substrate-Specific Inhibition Constants for Phospholipase AEBI University of California
30798607 3 ?-Lactones: A Novel Class of CaEBI National and Kapodistrian University of Athens
16610787 112 Synthesis and characterization of 3-arylquinazolinone and 3-arylquinazolinethione derivatives as selective estrogen receptor beta modulators.BDB Bristol-Myers Squibb
12941314 17 Discovery and evaluation of 3-(5-thien-3-ylpyridin-3-yl)-1H-indoles as a novel class of KDR kinase inhibitors.BDB Merck Research Laboratories