The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
27810597 |
12 |
Structure-activity relationship studies on 1-(2-oxopropyl)indole-5-carboxylic acids acting as inhibitors of cytosolic phospholipase A |
University of M£Nster |
25102418 |
36 |
Design, synthesis, and biological evaluation of 3-(1-Aryl-1H-indol-5-yl)propanoic acids as new indole-based cytosolic phospholipase A2a inhibitors. |
Asubio Pharma |
25152071 |
2 |
Inhibition of group IVA cytosolic phospholipase A2 by thiazolyl ketones in vitro, ex vivo, and in vivo. |
University of Athens |
19327988 |
9 |
1-(5-Carboxyindol-1-yl)propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha: synthesis and properties of bioisosteric benzimidazole, benzotriazole and indazole analogues. |
University of M£Nster |
18321717 |
17 |
1-(2-Carboxyindol-5-yloxy)propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha: synthesis, biological activity, metabolic stability, and solubility. |
University of M£Nster |
20005725 |
61 |
1-Indol-1-yl-propan-2-ones and related heterocyclic compounds as dual inhibitors of cytosolic phospholipase A(2)alpha and fatty acid amide hydrolase. |
University of M£Nster |
19178292 |
64 |
Reactions of functionalized sulfonamides: application to lowering the lipophilicity of cytosolic phospholipase A2alpha inhibitors. |
Wyeth Research |
| 8 |
Dicarboxylic acid inhibitors of phospholipase A2 |
TBA |
17826099 |
24 |
Inhibitory effect of synthetic C-C biflavones on various phospholipase A(2)s activity. |
Yeungnam University |
17320401 |
13 |
1-(5-Carboxy- and 5-carbamoylindol-1-yl)propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha: bioisosteric replacement of the carboxylic acid and carboxamide moiety. |
University of MüNster |
17305324 |
38 |
Discovery of Ecopladib, an indole inhibitor of cytosolic phospholipase A2alpha. |
Wyeth Research |
16610804 |
39 |
Design and synthesis of 1-indol-1-yl-propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha. |
University of MüNster |
16545564 |
20 |
1,2,4-Oxadiazolidin-3,5-diones and 1,3,5-triazin-2,4,6-triones as cytosolic phospholipase A2alpha inhibitors. |
Wyeth Research |
16392799 |
46 |
Inhibition of cytosolic phospholipase A2alpha: hit to lead optimization. |
Wyeth Research |
14643356 |
32 |
Structure-activity relationships of indole cytosolic phospholipase A(2)alpha inhibitors: substrate mimetics. |
Wyeth Research |
10737736 |
19 |
Pyrrolidine inhibitors of human cytosolic phospholipase A(2). |
Shionogi |
30615445 |
64 |
Substrate-Specific Inhibition Constants for Phospholipase A |
University of California |
30798607 |
3 |
?-Lactones: A Novel Class of Ca |
National and Kapodistrian University of Athens |
16610787 |
112 |
Synthesis and characterization of 3-arylquinazolinone and 3-arylquinazolinethione derivatives as selective estrogen receptor beta modulators. |
Bristol-Myers Squibb |
12941314 |
17 |
Discovery and evaluation of 3-(5-thien-3-ylpyridin-3-yl)-1H-indoles as a novel class of KDR kinase inhibitors. |
Merck Research Laboratories |