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16 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
25127101 26 Discovery of furan-2-carbohydrazides as orally active glucagon receptor antagonists.EBI Dainippon Sumitomo Pharma
22708876 106 Discovery of a novel glucagon receptor antagonist N-[(4-{(1S)-1-[3-(3, 5-dichlorophenyl)-5-(6-methoxynaphthalen-2-yl)-1H-pyrazol-1-yl]ethyl}phenyl)carbonyl]-ß-alanine (MK-0893) for the treatment of type II diabetes.EBI Merck Research Laboratories
11543679 15 A new approach to search for the bioactive conformation of glucagon: positional cyclization scanning.EBI University of Arizona
10794689 10 Design and synthesis of conformationally constrained glucagon analogues.EBI University of Arizona
9258362 30 The role of phenylalanine at position 6 in glucagon's mechanism of biological action: multiple replacement analogues of glucagon.EBI University of Arizona
8691441 19 Topographical amino acid substitution in position 10 of glucagon leads to antagonists/partial agonists with greater binding differences.EBI University of Arizona
21147532 82 Discovery of novel, potent, selective, and orally active human glucagon receptor antagonists containing a pyrazole core.EBI Merck Research Laboratories
 2 [des His1, des Phe6, Glu9]glucagon amide: A newly designed “pure” glucagon antagonistEBI TBA
 1 CP-99,711: a non-peptide glucagon receptor antagonistEBI TBA
18707090 68 Novel glucagon receptor antagonists with improved selectivity over the glucose-dependent insulinotropic polypeptide receptor.EBI Novo Nordisk
17201415 47 New beta-alanine derivatives are orally available glucagon receptor antagonists.EBI Novo Nordisk
12477359 78 Optimization of alkylidene hydrazide based human glucagon receptor antagonists. Discovery of the highly potent and orally available 3-cyano-4-hydroxybenzoic acid [1-(2,3,5,6-tetramethylbenzyl)-1H-indol-4-ylmethylene]hydrazide.EBI Novo Nordisk
11844695 35 Human glucagon receptor antagonists based on alkylidene hydrazides.EBI Pfizer
11543683 42 Identification of alkylidene hydrazides as glucagon receptor antagonists.EBI Pfizer
11311060 12 Development of potent truncated glucagon antagonists.EBI University of Arizona