The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
24972724 |
16 |
Influence of azide incorporation on binding affinity by small papain inhibitors. |
Radboud University Nijmegen |
24077527 |
11 |
Squaric acid/4-aminoquinoline conjugates: novel potent antiplasmodial agents. |
University Of Lisbon. Av. Prof. Gama Pinto |
23834438 |
10 |
Design, synthesis, and optimization of novel epoxide incorporating peptidomimetics as selective calpain inhibitors. |
University Of Illinois College Of Pharmacy |
23611656 |
9 |
Inhibition of rhodesain as a novel therapeutic modality for human African trypanosomiasis. |
Universit£ |
9804696 |
2 |
Use of papain as a model for the structure-based design of cathepsin K inhibitors: crystal structures of two papain-inhibitor complexes demonstrate binding to S'-subsites. |
Smithkline Beecham Pharmaceuticals |
22884354 |
36 |
Tanshinones as selective and slow-binding inhibitors for SARS-CoV cysteine proteases. |
Korea Research Institute Of Bioscience And Biotechnology |
19715320 |
87 |
Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
University Of Florida |
18995931 |
16 |
Natural polyprenylated benzophenones inhibiting cysteine and serine proteases. |
Federal University Of Alfenas |
10669559 |
180 |
Protease inhibitors: current status and future prospects. |
University Of Queensland |
9873373 |
20 |
Peptidyl beta-homo-aspartals: specific inhibitors of interleukin-1 beta converting enzyme and its homologues (caspases). |
Institute For Drug Research |
22019466 |
13 |
Design, synthesis and biological evaluation of peptidyl-vinylaminophosphonates as novel cysteine protease inhibitors. |
National Chemical Laboratory (Csir-Ncl) |
22071522 |
6 |
Aza vinyl sulfones: synthesis and evaluation as antiplasmodial agents. |
University Of Lisbon |
21923104 |
12 |
HLE-inhibitory alkaloids with a polyketide skeleton from the marine-derived fungus Coniothyrium cereale. |
University Of Bonn |
19913414 |
7 |
Antimalarial activity of azadipeptide nitriles. |
University Of Queensland |
19908842 |
84 |
Identification and optimization of inhibitors of Trypanosomal cysteine proteases: cruzain, rhodesain, and TbCatB. |
National Human Genome Research Institute |
| 4 |
Design of a new selective cysteine protease inactivator and its mechanistic implications |
TBA |
18789705 |
6 |
Peptidyl epoxides extended in the P' direction as cysteine protease inhibitors: effect on affinity and mechanism of inhibition. |
Bar-Ilan University |
16759084 |
12 |
Isatin compounds as noncovalent SARS coronavirus 3C-like protease inhibitors. |
Peking University |
12213061 |
23 |
Azapeptides structurally based upon inhibitory sites of cystatins as potent and selective inhibitors of cysteine proteases. |
University Of Gda£?Sk |
11720861 |
24 |
Discovery, total synthesis, HRV 3C-protease inhibitory activity, and structure-activity relationships of 2-methoxystypandrone and its analogues. |
Merck Research Laboratories |
11141092 |
85 |
Novel, nonpeptidic cyanamides as potent and reversible inhibitors of human cathepsins K and L. |
Merck Frosst Centre For Therapeutic Research |
11128643 |
4 |
(S)-Thiirancarboxylic acid as a reactive building block for a new class of cysteine protease inhibitors. |
University Of WüRzburg |
27396732 |
14 |
Discovery of New Anti-Schistosomal Hits by Integration of QSAR-Based Virtual Screening and High Content Screening. |
Universidade Federal De Goi£S |
10508448 |
11 |
Combinatorial library of serine and cysteine protease inhibitors that interact with both the S and S' binding sites. |
Brown University |
30830783 |
13 |
Potential Anticancer Agents Characterized from Selected Tropical Plants. |
The Ohio State University |
8765519 |
6 |
Mechanistic studies on the inactivation of papain by epoxysuccinyl inhibitors. |
University Of Wisconsin |
8230139 |
165 |
Peptide alpha-keto ester, alpha-keto amide, and alpha-keto acid inhibitors of calpains and other cysteine proteases. |
Georgia Institute Of Technology |
7932558 |
30 |
Nonpeptidic inhibitors of human leukocyte elastase. 2. Design, synthesis, and in vitro activity of a series of 3-amino-6-arylopyridin-2-one trifluoromethyl ketones. |
Zeneca Pharmaceuticals Group |
7562931 |
41 |
Peptidyl alpha-ketoheterocyclic inhibitors of human neutrophil elastase. 3. In vitro and in vivo potency of a series of peptidyl alpha-ketobenzoxazoles. |
Zeneca Pharmaceuticals |
9599275 |
1 |
Isolation of 1-carboxymethylnicotinic acid from the marine sponge anthosigmella cf. raromicrosclera As a cysteine protease inhibitor1 |
The University Of Tokyo |
6547487 |
3 |
Vinylogous amino acid esters: a new class of inactivators for thiol proteases. |
TBA |
11170666 |
6 |
Isolation and structure determination of nostocyclopeptides A1 and A2 from the terrestrial cyanobacterium Nostoc sp. ATCC53789. |
University Of Hawaii At Manoa |
3941405 |
15 |
Carboxyl-modified amino acids and peptides as protease inhibitors. |
TBA |
2724298 |
11 |
Acid-sensitive latent inhibitors for proteolytic enzymes: synthesis and characterization. |
Amherst College |
22468751 |
2 |
Inhibition of cysteine proteases by a natural biflavone: behavioral evaluation of fukugetin as papain and cruzain inhibitor. |
Federal University Of Sao Paulo |
26132413 |
2 |
Identification and Co-complex Structure of a New S. pyogenes SpeB Small Molecule Inhibitor. |
The Scripps Research Institute |
19912058 |
11 |
Dipeptide-derived nitriles containing additional electrophilic sites: potentially irreversible inhibitors of cysteine proteases. |
Rheinische Friedrich-Wilhelms-Universitat Bonn |
16302809 |
196 |
Interaction of papain-like cysteine proteases with dipeptide-derived nitriles. |
Rheinische Friedrich-Wilhelms-Universitat Bonn |