The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
26638045 |
58 |
Synthesis, experimental evaluation and molecular modelling of hydroxamate derivatives as zinc metalloproteinase inhibitors. |
Uit The Arctic University of Norway |
25559080 |
38 |
Additivity or cooperativity: which model can predict the influence of simultaneous incorporation of two or more functionalities in a ligand molecule? |
The State University of New York |
23988485 |
5 |
Synthesis and enzymatic evaluation of phosphoramidon and itsß anomer: Anomerization ofa-l-rhamnose triacetate upon phosphitylation. |
Jiangxi Science and Technology Normal University |
22894131 |
4 |
Water mediated ligand functional group cooperativity: the contribution of a methyl group to binding affinity is enhanced by a COO(-) group through changes in the structure and thermodynamics of the hydration waters of ligand-thermolysin complexes. |
The State University of New York |
7783143 |
66 |
Hydroxamic acids as potent inhibitors of endothelin-converting enzyme from human bronchiolar smooth muscle. |
Berlex Laboratories |
8021926 |
41 |
New thiol inhibitors of neutral endopeptidase EC 3.4.24.11: synthesis and enzyme active-site recognition. |
University of Paris |
8340909 |
14 |
Excursions in drug discovery. |
Merck Research Laboratories |
1588550 |
10 |
Definition and display of steric, hydrophobic, and hydrogen-bonding properties of ligand binding sites in proteins using Lee and Richards accessible surface: validation of a high-resolution graphical tool for drug design. |
Ciba-Geigy |
12443790 |
3 |
Silanediol-based inhibitor of thermolysin. |
State University of New York |
| 11 |
Thiol and hydroxamic acid containing inhibitors of endothelin converting enzyme |
TBA |
20494587 |
24 |
Identification of novel quinazolin-4(3H)-ones as inhibitors of thermolysin, the prototype of the M4 family of proteinases. |
University of Troms£ |
| 2 |
Inhibitory stereochemistry of N-chloroacetyl-N-hydroxyleucine methyl ester for thermolysin |
TBA |
19072688 |
22 |
Discovery of potent thermolysin inhibitors using structure based virtual screening and binding assays. |
University of Tromsø |
12951085 |
10 |
Reversed hydroxamate-bearing thermolysin inhibitors mimic a high-energy intermediate along the enzyme-catalyzed proteolytic reaction pathway. |
Pohang University of Science and Technology |
9934463 |
6 |
Inhibition stereochemistry of hydroxamate inhibitors for thermolysin. |
Pohang University of Science and Technology |
9871678 |
8 |
Inhibition of thermolysin with nitrone-bearing substrate analogs: a new type of thermolysin inhibitors. |
Pohang University of Science and Technology |
9046341 |
44 |
Meta-substituted benzofused macrocyclic lactams as zinc metalloprotease inhibitors. |
Ciba-Geigy |
9046340 |
23 |
Ortho-substituted benzofused macrocyclic lactams as zinc metalloprotease inhibitors. |
Novartis Pharmaceuticals |
14519960 |
9 |
Biological activity of tropolone. |
Osaka Organic Chemical Industry |
11931613 |
76 |
Development of new hydrogen-bond descriptors and their application to comparative molecular field analyses. |
University of Marburg |
12061879 |
44 |
SMall Molecule Growth 2001 (SMoG2001): an improved knowledge-based scoring function for protein-ligand interactions. |
Harvard University |