Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50249644 (CHEMBL4073895) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | MMDB PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from human ERG | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50249651 (CHEMBL4098533) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from human ERG | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50249650 (CHEMBL4088372) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from human ERG | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 2A (Homo sapiens (Human)) | BDBM50249723 (CHEMBL4070546) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 650 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Inhibition of 5-HT2A receptor (unknown origin) | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50249645 (CHEMBL4078859) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from human ERG | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50249731 (CHEMBL4080513) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 900 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from human ERG | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50249699 (CHEMBL4094458) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from human ERG | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50249624 (CHEMBL4095178) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from human ERG | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50249728 (CHEMBL4072841) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from human ERG | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50249647 (CHEMBL4099725) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from human ERG | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50249623 (CHEMBL4074704) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from human ERG | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 2A (Homo sapiens (Human)) | BDBM50249664 (CHEMBL4065786) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Inhibition of 5-HT2A receptor (unknown origin) | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50249646 (CHEMBL4103135) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from human ERG | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 2A (Homo sapiens (Human)) | BDBM50249699 (CHEMBL4094458) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Inhibition of 5-HT2A receptor (unknown origin) | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 2C19 (Homo sapiens (Human)) | BDBM50249652 (CHEMBL4103847) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Inhibition of CYP2C19 in human liver microsomes after 10 mins by LC/MS analysis | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 1A2 (Homo sapiens (Human)) | BDBM50249652 (CHEMBL4103847) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Inhibition of CYP1A2 in human liver microsomes after 10 mins by LC/MS analysis | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 2C8 (Homo sapiens (Human)) | BDBM50249652 (CHEMBL4103847) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Inhibition of CYP2C8 in human liver microsomes after 10 mins by LC/MS analysis | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 2D6 (Homo sapiens (Human)) | BDBM50249652 (CHEMBL4103847) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Inhibition of CYP2D6 in human liver microsomes after 10 mins by LC/MS analysis | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 2C9 (Homo sapiens (Human)) | BDBM50249652 (CHEMBL4103847) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Inhibition of CYP2C9 in human liver microsomes after 10 mins by LC/MS analysis | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50249744 (CHEMBL4096097) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.47E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from human ERG | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50249654 (CHEMBL4068797) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from human ERG | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50249652 (CHEMBL4103847) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from human ERG | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50249653 (CHEMBL4079597) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from human ERG | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249623 (CHEMBL4074704) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 6 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249624 (CHEMBL4095178) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249700 (CHEMBL4075866) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 60 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249701 (CHEMBL4085732) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 60 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249702 (CHEMBL4077873) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 220 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249703 (CHEMBL4079841) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 30 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249707 (CHEMBL4066900) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 130 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249708 (CHEMBL4096964) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 60 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249709 (CHEMBL4075398) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 260 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249710 (CHEMBL4091156) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 750 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249714 (CHEMBL4063409) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 280 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249715 (CHEMBL4080468) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 140 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249716 (CHEMBL4101498) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249717 (CHEMBL4075504) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 500 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249718 (CHEMBL4071587) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 500 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249719 (CHEMBL4082112) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 70 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249720 (CHEMBL4100122) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 40 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249721 (CHEMBL4061921) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 90 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249722 (CHEMBL4097707) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 130 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249723 (CHEMBL4070546) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249724 (CHEMBL4103525) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 560 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249725 (CHEMBL4086717) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 9 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249726 (CHEMBL4065280) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 420 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249644 (CHEMBL4073895) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | MMDB PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 8 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249727 (CHEMBL4067994) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 20 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249645 (CHEMBL4078859) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50249646 (CHEMBL4103135) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 1 | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica , N. V. Turnhoutseweg 30, 2340 Beerse, Belgium. Curated by ChEMBL | Assay Description Agonist activity at TLR7 in human PBMC assessed as induction of IFNalpha-mediated inhibition of HCV genotype 1b RNA replication in human HuH luc/neo ... | J Med Chem 60: 6137-6151 (2017) Article DOI: 10.1021/acs.jmedchem.7b00365 BindingDB Entry DOI: 10.7270/Q2XP77CC | |||||||||||
More data for this Ligand-Target Pair |
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