Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cholecystokinin receptor type A (RAT) | BDBM50060321 (1H-Indole-2-carboxylic acid ((R)-1-methyl-2-oxo-5-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreas | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.520 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreas | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50060322 (CHEMBL332261 | [(S)-1-((4aS,5S)-2-Benzyl-1,3-dioxo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.620 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreas | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | 2.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]- pCCK-8 binding to Cholecystokinin type B receptor of rat cerebral cortex membranes | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50060323 (CHEMBL431858 | [(S)-1-((4aR,5R)-2-Benzyl-1,3-dioxo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 10.6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreas | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50060326 (CHEMBL116001 | [(R)-1-((4aS,5S)-2-Benzyl-1,3-dioxo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 298 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreas | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50060321 (1H-Indole-2-carboxylic acid ((R)-1-methyl-2-oxo-5-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 342 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]- pCCK-8 binding to Cholecystokinin type B receptor of rat cerebral cortex membranes | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50060327 (CHEMBL116127 | [(S)-1-((4aR,5S)-2-Benzyl-1,3-dioxo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 572 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreas | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50060320 (CHEMBL326064 | [(R)-1-((4aR,5R)-2-Benzyl-1,3-dioxo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 813 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreas | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50060325 ((2S,8S,8aR)-2-Benzyl-8-[(S)-2-tert-butoxycarbonyla...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.03E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreas | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50060328 ((2R,8S,8aR)-2-Benzyl-8-[(R)-2-tert-butoxycarbonyla...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.56E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]- pCCK-8 binding to Cholecystokinin type B receptor of rat cerebral cortex membranes | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50060318 (CHEMBL324294 | [(R)-1-((4aS,5R)-2-Benzyl-1,3-dioxo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.89E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]- pCCK-8 binding to Cholecystokinin type B receptor of rat cerebral cortex membranes | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50060323 (CHEMBL431858 | [(S)-1-((4aR,5R)-2-Benzyl-1,3-dioxo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.73E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]- pCCK-8 binding to Cholecystokinin type B receptor of rat cerebral cortex membranes | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50060319 (CHEMBL113718 | [(S)-1-((4aS,5R)-2-Benzyl-1,3-dioxo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.89E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreas | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50060319 (CHEMBL113718 | [(S)-1-((4aS,5R)-2-Benzyl-1,3-dioxo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.91E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]- pCCK-8 binding to Cholecystokinin type B receptor of rat cerebral cortex membranes | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50060325 ((2S,8S,8aR)-2-Benzyl-8-[(S)-2-tert-butoxycarbonyla...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]- pCCK-8 binding to Cholecystokinin type B receptor of rat cerebral cortex membranes | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50060324 (CHEMBL114517 | [(R)-1-((4aR,5S)-2-Benzyl-1,3-dioxo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]- pCCK-8 binding to Cholecystokinin type B receptor of rat cerebral cortex membranes | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50060324 (CHEMBL114517 | [(R)-1-((4aR,5S)-2-Benzyl-1,3-dioxo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreas | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50060318 (CHEMBL324294 | [(R)-1-((4aS,5R)-2-Benzyl-1,3-dioxo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreas | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50060322 (CHEMBL332261 | [(S)-1-((4aS,5S)-2-Benzyl-1,3-dioxo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]- pCCK-8 binding to Cholecystokinin type B receptor of rat cerebral cortex membranes | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50060326 (CHEMBL116001 | [(R)-1-((4aS,5S)-2-Benzyl-1,3-dioxo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]- pCCK-8 binding to Cholecystokinin type B receptor of rat cerebral cortex membranes | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50060320 (CHEMBL326064 | [(R)-1-((4aR,5R)-2-Benzyl-1,3-dioxo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]- pCCK-8 binding to Cholecystokinin type B receptor of rat cerebral cortex membranes | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50060327 (CHEMBL116127 | [(S)-1-((4aR,5S)-2-Benzyl-1,3-dioxo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]- pCCK-8 binding to Cholecystokinin type B receptor of rat cerebral cortex membranes | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50060328 ((2R,8S,8aR)-2-Benzyl-8-[(R)-2-tert-butoxycarbonyla...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Química Médica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreas | J Med Chem 40: 3402-7 (1997) Article DOI: 10.1021/jm9703247 BindingDB Entry DOI: 10.7270/Q2B56HV4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50106593 (CHEMBL135602 | [1-(2-Benzyl-3-oxo-1-thioxo-octahyd...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.0900 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Qu£mica M£dica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 binding to cholecystokinin type A receptor of rat pancreas | J Med Chem 44: 4196-206 (2001) BindingDB Entry DOI: 10.7270/Q2TD9Z23 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50005463 ((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 0.710 | n/a | n/a | n/a | n/a | n/a | n/a |
Insituto de Qu�mica M�dica (CSIC), Juan de la Cierva 3, E-28006 Madrid, Spain. Curated by ChEMBL | Assay Description Binding affinity by competitive inhibition of the radioligand [3H]pCCK-8 at Cholecystokinin type A receptor from rat pancreas | J Med Chem 42: 4659-68 (1999) BindingDB Entry DOI: 10.7270/Q24T6K2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Insituto de Qu�mica M�dica (CSIC), Juan de la Cierva 3, E-28006 Madrid, Spain. Curated by ChEMBL | Assay Description Binding affinity by competitive inhibition of the radioligand [3H]pCCK-8 at Cholecystokinin type A receptor from rat pancreas | J Med Chem 42: 4659-68 (1999) BindingDB Entry DOI: 10.7270/Q24T6K2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.04 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Qu£mica M£dica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 binding to cholecystokinin type A receptor of rat pancreas | J Med Chem 44: 4196-206 (2001) BindingDB Entry DOI: 10.7270/Q2TD9Z23 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.04 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Qu£mica M£dica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 specific binding to cholecystokinin type A receptor in rat pancreas | J Med Chem 44: 2219-28 (2001) BindingDB Entry DOI: 10.7270/Q2M32WG1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50106588 (CHEMBL133446 | [1-(2-Benzyl-1,3-dithioxo-octahydro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.34 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Qu£mica M£dica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 binding to cholecystokinin type A receptor of rat pancreas | J Med Chem 44: 4196-206 (2001) BindingDB Entry DOI: 10.7270/Q2TD9Z23 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50106591 (CHEMBL337620 | [1-(2-Benzyl-1,3-dioxo-4a(S)-octahy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.59 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Qu£mica M£dica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 binding to cholecystokinin type A receptor of rat pancreas | J Med Chem 44: 4196-206 (2001) BindingDB Entry DOI: 10.7270/Q2TD9Z23 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50106597 (CHEMBL133983 | [1-(2-Benzyl-1-oxo-3-thioxo-octahyd...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.83 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Qu£mica M£dica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 binding to cholecystokinin type A receptor of rat pancreas | J Med Chem 44: 4196-206 (2001) BindingDB Entry DOI: 10.7270/Q2TD9Z23 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Insituto de Qu�mica M�dica (CSIC), Juan de la Cierva 3, E-28006 Madrid, Spain. Curated by ChEMBL | Assay Description Binding affinity by competitive inhibition of the radioligand [3H]pCCK-8 at Cholecystokinin type B receptor from rat cerebral cortex membrane | J Med Chem 42: 4659-68 (1999) BindingDB Entry DOI: 10.7270/Q24T6K2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Qu£mica M£dica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 specific binding cholecystokinin type B receptor in rat cerebral cortex membranes | J Med Chem 44: 2219-28 (2001) BindingDB Entry DOI: 10.7270/Q2M32WG1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Qu£mica M£dica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 binding to cholecystokinin type B receptor of rat cerebral cortex | J Med Chem 44: 4196-206 (2001) BindingDB Entry DOI: 10.7270/Q2TD9Z23 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50106589 (CHEMBL132467 | [1-(2-Benzyl-1-oxo-3-thioxo-octahyd...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 13.8 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Qu£mica M£dica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 binding to cholecystokinin type A receptor of rat pancreas | J Med Chem 44: 4196-206 (2001) BindingDB Entry DOI: 10.7270/Q2TD9Z23 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50100686 (CHEMBL71996 | {2-(1H-Indol-3-yl)-1-[2-(4-methoxy-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 15.9 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Qu£mica M£dica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 specific binding to cholecystokinin type A receptor in rat pancreas | J Med Chem 44: 2219-28 (2001) BindingDB Entry DOI: 10.7270/Q2M32WG1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50106596 (CHEMBL132938 | [1-(2-Benzyl-1,3-dioxo-4a(R)-octahy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 22.7 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Qu£mica M£dica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 binding to cholecystokinin type A receptor of rat pancreas | J Med Chem 44: 4196-206 (2001) BindingDB Entry DOI: 10.7270/Q2TD9Z23 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50082644 (CHEMBL356765 | [1-((4aS,5S)-2-Benzyl-1,3-dioxo-oct...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
Insituto de Qu�mica M�dica (CSIC), Juan de la Cierva 3, E-28006 Madrid, Spain. Curated by ChEMBL | Assay Description Binding affinity by competitive inhibition of the radioligand [3H]pCCK-8 at Cholecystokinin type A receptor from rat pancreas | J Med Chem 42: 4659-68 (1999) BindingDB Entry DOI: 10.7270/Q24T6K2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50082647 (CHEMBL142349 | [1-((4aR,5R)-2-Benzyl-1,3-dioxo-oct...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 66 | n/a | n/a | n/a | n/a | n/a | n/a |
Insituto de Qu�mica M�dica (CSIC), Juan de la Cierva 3, E-28006 Madrid, Spain. Curated by ChEMBL | Assay Description Binding affinity by competitive inhibition of the radioligand [3H]pCCK-8 at Cholecystokinin type A receptor from rat pancreas | J Med Chem 42: 4659-68 (1999) BindingDB Entry DOI: 10.7270/Q24T6K2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50082642 (3-((4aR,5R)-2-Benzyl-1,3-dioxo-octahydro-pyrido[1,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 226 | n/a | n/a | n/a | n/a | n/a | n/a |
Insituto de Qu�mica M�dica (CSIC), Juan de la Cierva 3, E-28006 Madrid, Spain. Curated by ChEMBL | Assay Description Binding affinity by competitive inhibition of the radioligand [3H]pCCK-8 at Cholecystokinin type A receptor from rat pancreas | J Med Chem 42: 4659-68 (1999) BindingDB Entry DOI: 10.7270/Q24T6K2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50106599 (CHEMBL337639 | [1-(2-Benzyl-3-methoxy-1-oxo-octahy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 370 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Qu£mica M£dica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 binding to cholecystokinin type A receptor of rat pancreas | J Med Chem 44: 4196-206 (2001) BindingDB Entry DOI: 10.7270/Q2TD9Z23 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50082655 (Adamantane-1-carboxylic acid [(S)-1-((4aS,5S)-2-be...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 486 | n/a | n/a | n/a | n/a | n/a | n/a |
Insituto de Qu�mica M�dica (CSIC), Juan de la Cierva 3, E-28006 Madrid, Spain. Curated by ChEMBL | Assay Description Binding affinity by competitive inhibition of the radioligand [3H]pCCK-8 at Cholecystokinin type A receptor from rat pancreas | J Med Chem 42: 4659-68 (1999) BindingDB Entry DOI: 10.7270/Q24T6K2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50005463 ((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 696 | n/a | n/a | n/a | n/a | n/a | n/a |
Insituto de Qu�mica M�dica (CSIC), Juan de la Cierva 3, E-28006 Madrid, Spain. Curated by ChEMBL | Assay Description Binding affinity by competitive inhibition of the radioligand [3H]pCCK-8 at Cholecystokinin type B receptor from rat cerebral cortex membrane | J Med Chem 42: 4659-68 (1999) BindingDB Entry DOI: 10.7270/Q24T6K2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50106598 (CHEMBL335274 | [1-(2-Benzyl-3-oxo-1-thioxo-octahyd...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 825 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Qu£mica M£dica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 binding to cholecystokinin type A receptor of rat pancreas | J Med Chem 44: 4196-206 (2001) BindingDB Entry DOI: 10.7270/Q2TD9Z23 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50106594 (CHEMBL334358 | [1-(2-Benzyl-1,3-dithioxo-octahydro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 900 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Qu£mica M£dica (CSIC) Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 binding to cholecystokinin type A receptor of rat pancreas | J Med Chem 44: 4196-206 (2001) BindingDB Entry DOI: 10.7270/Q2TD9Z23 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50082637 ((S)-2-Amino-N-((4aR,5R)-2-benzyl-1,3-dioxo-octahyd...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Insituto de Qu�mica M�dica (CSIC), Juan de la Cierva 3, E-28006 Madrid, Spain. Curated by ChEMBL | Assay Description Binding affinity by competitive inhibition of the radioligand [3H]pCCK-8 at Cholecystokinin type A receptor from rat pancreas | J Med Chem 42: 4659-68 (1999) BindingDB Entry DOI: 10.7270/Q24T6K2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50082638 (CHEMBL343560 | [(S)-1-[((4aR,5R)-2-Benzyl-1,3-diox...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Insituto de Qu�mica M�dica (CSIC), Juan de la Cierva 3, E-28006 Madrid, Spain. Curated by ChEMBL | Assay Description Binding affinity by competitive inhibition of the radioligand [3H]pCCK-8 at Cholecystokinin type A receptor from rat pancreas | J Med Chem 42: 4659-68 (1999) BindingDB Entry DOI: 10.7270/Q24T6K2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50082645 (CHEMBL140098 | [(1S,2S)-2-((4aR,5R)-2-Benzyl-1,3-d...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Insituto de Qu�mica M�dica (CSIC), Juan de la Cierva 3, E-28006 Madrid, Spain. Curated by ChEMBL | Assay Description Binding affinity by competitive inhibition of the radioligand [3H]pCCK-8 at Cholecystokinin type A receptor from rat pancreas | J Med Chem 42: 4659-68 (1999) BindingDB Entry DOI: 10.7270/Q24T6K2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (RAT) | BDBM50369471 (CHEMBL1794878) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Insituto de Qu�mica M�dica (CSIC), Juan de la Cierva 3, E-28006 Madrid, Spain. Curated by ChEMBL | Assay Description Binding affinity by competitive inhibition of the radioligand [3H]pCCK-8 at Cholecystokinin type A receptor from rat pancreas | J Med Chem 42: 4659-68 (1999) BindingDB Entry DOI: 10.7270/Q24T6K2B | |||||||||||
More data for this Ligand-Target Pair |
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