Compile Data Set for Download or QSAR

Found 22 hits with Last Name = 'sakasai' and Initial = 'm'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Transient receptor potential cation channel subfamily A member 1 (Homo sapiens (Human))	BDBM50269659 (CHEMBL4069984) Show SMILES CCOC(C(C)Oc1c(OC)cc(CC=C)cc1OC)c1ccc(O)c(OC)c1 Show InChI InChI=1S/C23H30O6/c1-7-9-16-12-20(26-5)23(21(13-16)27-6)29-15(3)22(28-8-2)17-10-11-18(24)19(14-17)25-4/h7,10-15,22,24H,1,8-9H2,2-6H3	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	1.91E+4	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at recombinant human TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for 5 mins by Fl...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269684 (CHEMBL4062360) Show SMILES COC(C(C)Oc1c(OC)cc(CC=C)cc1OC)c1ccc(O)c(OC)c1 Show InChI InChI=1S/C22H28O6/c1-7-8-15-11-19(25-4)22(20(12-15)26-5)28-14(2)21(27-6)16-9-10-17(23)18(13-16)24-3/h7,9-14,21,23H,1,8H2,2-6H3	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	3.45E+3	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269663 (CHEMBL4076583) Show SMILES COc1cc(ccc1O)C(O[C@@H]1C[C@H](C)CC[C@H]1C(C)C)C(C)Oc1c(OC)cc(CC=C)cc1OC |r| Show InChI InChI=1S/C31H44O6/c1-9-10-22-16-28(34-7)31(29(17-22)35-8)36-21(5)30(23-12-14-25(32)27(18-23)33-6)37-26-15-20(4)11-13-24(26)19(2)3/h9,12,14,16-21,24,26,30,32H,1,10-11,13,15H2,2-8H3/t20-,21?,24+,26-,30?/m1/s1	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	28	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269664 (CHEMBL4076657) Show SMILES COc1cc(ccc1O)C(OC1CCCCC1)C(C)Oc1c(OC)cc(CC=C)cc1OC Show InChI InChI=1S/C27H36O6/c1-6-10-19-15-24(30-4)27(25(16-19)31-5)32-18(2)26(33-21-11-8-7-9-12-21)20-13-14-22(28)23(17-20)29-3/h6,13-18,21,26,28H,1,7-12H2,2-5H3	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	54	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269668 (CHEMBL4073357) Show SMILES COc1cc(ccc1O)C(OCC(C)C)C(C)Oc1c(OC)cc(CC=C)cc1OC Show InChI InChI=1S/C25H34O6/c1-8-9-18-12-22(28-6)25(23(13-18)29-7)31-17(4)24(30-15-16(2)3)19-10-11-20(26)21(14-19)27-5/h8,10-14,16-17,24,26H,1,9,15H2,2-7H3	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	138	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269669 (CHEMBL4065256) Show SMILES COc1cc(ccc1O)C(OC(C)C)C(C)Oc1c(OC)cc(CC=C)cc1OC Show InChI InChI=1S/C24H32O6/c1-8-9-17-12-21(27-6)24(22(13-17)28-7)30-16(4)23(29-15(2)3)18-10-11-19(25)20(14-18)26-5/h8,10-16,23,25H,1,9H2,2-7H3	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	82	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269670 (CHEMBL4072058) Show SMILES CCCCOCCOC(C(C)Oc1c(OC)cc(CC=C)cc1OC)c1ccc(O)c(OC)c1 Show InChI InChI=1S/C27H38O7/c1-7-9-13-32-14-15-33-26(21-11-12-22(28)23(18-21)29-4)19(3)34-27-24(30-5)16-20(10-8-2)17-25(27)31-6/h8,11-12,16-19,26,28H,2,7,9-10,13-15H2,1,3-6H3	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	153	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (Homo sapiens (Human))	BDBM50318482 ((-)-menthol | CHEMBL470670 | MENTHOL | US11406649,...) Show SMILES CC(C)[C@@H]1CC[C@@H](C)C[C@H]1O |r| Show InChI InChI=1S/C10H20O/c1-7(2)9-5-4-8(3)6-10(9)11/h7-11H,4-6H2,1-3H3/t8-,9+,10-/m1/s1	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars	DrugBank Article PubMed	n/a	n/a	n/a	n/a	9.60E+4	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at recombinant human TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for 5 mins by Fl...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269671 (CHEMBL4084423) Show SMILES CCO[C@@H]([C@H](C)Oc1c(OC)cc(CC=C)cc1OC)c1ccc(O)c(OC)c1 |r| Show InChI InChI=1S/C23H30O6/c1-7-9-16-12-20(26-5)23(21(13-16)27-6)29-15(3)22(28-8-2)17-10-11-18(24)19(14-17)25-4/h7,10-15,22,24H,1,8-9H2,2-6H3/t15-,22-/m0/s1	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.13E+3	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50318482 ((-)-menthol | CHEMBL470670 | MENTHOL | US11406649,...) Show SMILES CC(C)[C@@H]1CC[C@@H](C)C[C@H]1O |r| Show InChI InChI=1S/C10H20O/c1-7(2)9-5-4-8(3)6-10(9)11/h7-11H,4-6H2,1-3H3/t8-,9+,10-/m1/s1	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars	DrugBank Article PubMed	n/a	n/a	n/a	n/a	1.01E+4	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269659 (CHEMBL4069984) Show SMILES CCOC(C(C)Oc1c(OC)cc(CC=C)cc1OC)c1ccc(O)c(OC)c1 Show InChI InChI=1S/C23H30O6/c1-7-9-16-12-20(26-5)23(21(13-16)27-6)29-15(3)22(28-8-2)17-10-11-18(24)19(14-17)25-4/h7,10-15,22,24H,1,8-9H2,2-6H3	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	332	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269672 (CHEMBL463097) Show SMILES COc1ccc(cc1OC)[C@H](O)[C@@H](C)Oc1c(OC)cc(CC=C)cc1OC |r| Show InChI InChI=1S/C22H28O6/c1-7-8-15-11-19(26-5)22(20(12-15)27-6)28-14(2)21(23)16-9-10-17(24-3)18(13-16)25-4/h7,9-14,21,23H,1,8H2,2-6H3/t14-,21-/m1/s1	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269673 (CHEMBL1909927) Show SMILES COc1ccc(cc1OC)[C@H](OC(C)=O)[C@@H](C)Oc1c(OC)cc(CC=C)cc1OC |r| Show InChI InChI=1S/C24H30O7/c1-8-9-17-12-21(28-6)24(22(13-17)29-7)30-15(2)23(31-16(3)25)18-10-11-19(26-4)20(14-18)27-5/h8,10-15,23H,1,9H2,2-7H3/t15-,23-/m1/s1	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269674 (CHEMBL4065676) Show SMILES COc1cc(ccc1O)[C@H](OC(C)=O)[C@@H](C)Oc1c(OC)cc(CC=C)cc1OC |r| Show InChI InChI=1S/C23H28O7/c1-7-8-16-11-20(27-5)23(21(12-16)28-6)29-14(2)22(30-15(3)24)17-9-10-18(25)19(13-17)26-4/h7,9-14,22,25H,1,8H2,2-6H3/t14-,22-/m1/s1	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269675 (CHEMBL4087839) Show SMILES COc1cc(ccc1O)C(O)C(C)Oc1c(OC)cc(CC=C)cc1OC Show InChI InChI=1S/C21H26O6/c1-6-7-14-10-18(25-4)21(19(11-14)26-5)27-13(2)20(23)15-8-9-16(22)17(12-15)24-3/h6,8-13,20,22-23H,1,7H2,2-5H3	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269676 (CHEMBL4074380) Show SMILES CCO[C@H]([C@H](C)Oc1c(OC)cc(CC=C)cc1OC)c1ccc(O)c(OC)c1 |r| Show InChI InChI=1S/C23H30O6/c1-7-9-16-12-20(26-5)23(21(13-16)27-6)29-15(3)22(28-8-2)17-10-11-18(24)19(14-17)25-4/h7,10-15,22,24H,1,8-9H2,2-6H3/t15-,22+/m0/s1	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	87	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269678 (CHEMBL4092140) Show SMILES CCO[C@@H]([C@@H](C)Oc1c(OC)cc(CC=C)cc1OC)c1ccc(O)c(OC)c1 |r| Show InChI InChI=1S/C23H30O6/c1-7-9-16-12-20(26-5)23(21(13-16)27-6)29-15(3)22(28-8-2)17-10-11-18(24)19(14-17)25-4/h7,10-15,22,24H,1,8-9H2,2-6H3/t15-,22+/m1/s1	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	583	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269680 (CHEMBL4073694) Show SMILES CCO[C@H]([C@@H](C)Oc1c(OC)cc(CC=C)cc1OC)c1ccc(O)c(OC)c1 |r| Show InChI InChI=1S/C23H30O6/c1-7-9-16-12-20(26-5)23(21(13-16)27-6)29-15(3)22(28-8-2)17-10-11-18(24)19(14-17)25-4/h7,10-15,22,24H,1,8-9H2,2-6H3/t15-,22-/m1/s1	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.15E+3	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269681 (CHEMBL4077565) Show SMILES CCCCCCCCCCOC(C(C)Oc1c(OC)cc(CC=C)cc1OC)c1ccc(O)c(OC)c1 Show InChI InChI=1S/C31H46O6/c1-7-9-10-11-12-13-14-15-19-36-30(25-17-18-26(32)27(22-25)33-4)23(3)37-31-28(34-5)20-24(16-8-2)21-29(31)35-6/h8,17-18,20-23,30,32H,2,7,9-16,19H2,1,3-6H3	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	66	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269682 (CHEMBL4076994) Show SMILES CCCCCCCCOC(C(C)Oc1c(OC)cc(CC=C)cc1OC)c1ccc(O)c(OC)c1 Show InChI InChI=1S/C29H42O6/c1-7-9-10-11-12-13-17-34-28(23-15-16-24(30)25(20-23)31-4)21(3)35-29-26(32-5)18-22(14-8-2)19-27(29)33-6/h8,15-16,18-21,28,30H,2,7,9-14,17H2,1,3-6H3	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	86	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269683 (CHEMBL4084074) Show SMILES CCCCCCOC(C(C)Oc1c(OC)cc(CC=C)cc1OC)c1ccc(O)c(OC)c1 Show InChI InChI=1S/C27H38O6/c1-7-9-10-11-15-32-26(21-13-14-22(28)23(18-21)29-4)19(3)33-27-24(30-5)16-20(12-8-2)17-25(27)31-6/h8,13-14,16-19,26,28H,2,7,9-12,15H2,1,3-6H3	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	329	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM50269660 (CHEMBL4067554) Show SMILES COc1cc(ccc1O)C(O[C@H]1C[C@@H](C)CC[C@@H]1C(C)C)C(C)Oc1c(OC)cc(CC=C)cc1OC |r| Show InChI InChI=1S/C31H44O6/c1-9-10-22-16-28(34-7)31(29(17-22)35-8)36-21(5)30(23-12-14-25(32)27(18-23)33-6)37-26-15-20(4)11-13-24(26)19(2)3/h9,12,14,16-21,24,26,30,32H,1,10-11,13,15H2,2-8H3/t20-,21?,24+,26-,30?/m0/s1	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	11	n/a	n/a	n/a	n/a
Kansei Science Research and Biological Science Research, Kao Corporation, 2606 Akabane, Ichikai-Machi, Haga-Gun, Tochigi 321-3497, Japan. Curated by ChEMBL					Assay Description Agonist activity at full length recombinant human TRPM8 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for ...				ACS Med Chem Lett 8: 715-719 (2017) Article DOI: 10.1021/acsmedchemlett.7b00104 BindingDB Entry DOI: 10.7270/Q2CZ39N2
					More data for this Ligand-Target Pair