Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Dihydroorotate dehydrogenase (quinone), mitochondrial (Plasmodium falciparum (isolate 3D7)) | BDBM24400 (5-methyl-N-(naphthalen-2-yl)-[1,2,4]triazolo[1,5-a...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 65 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Turin Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ... | Eur J Med Chem 163: 266-280 (2019) Article DOI: 10.1016/j.ejmech.2018.11.044 BindingDB Entry DOI: 10.7270/Q2VT1WCQ | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50339906 (((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50339906 (((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50339906 (((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50339906 (((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50530866 (CHEMBL4529844) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50530866 (CHEMBL4529844) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50530864 (CHEMBL4467050) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 380 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50530864 (CHEMBL4467050) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 380 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50530866 (CHEMBL4529844) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 450 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50530866 (CHEMBL4529844) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 450 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50530862 (CHEMBL4446951) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.24E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50530862 (CHEMBL4446951) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.24E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50530864 (CHEMBL4467050) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.36E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50530864 (CHEMBL4467050) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.36E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50530862 (CHEMBL4446951) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.44E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50530862 (CHEMBL4446951) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.44E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase, cytoplasmic (Homo sapiens) | BDBM50339906 (((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 2.17E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of human N-terminal polyHis-tagged SerRS expressed in Escherichia coli BL21 (DE3) using Ap4A as substrate in presence of serine by leucono... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Serine--tRNA ligase, cytoplasmic (Homo sapiens) | BDBM50339906 (((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 2.17E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of human N-terminal polyHis-tagged SerRS expressed in Escherichia coli BL21 (DE3) using Ap4A as substrate in presence of serine by leucono... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Dihydroorotate dehydrogenase (quinone), mitochondrial (Plasmodium falciparum (isolate 3D7)) | BDBM50507739 (CHEMBL4458056) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | 2.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Turin Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ... | Eur J Med Chem 163: 266-280 (2019) Article DOI: 10.1016/j.ejmech.2018.11.044 BindingDB Entry DOI: 10.7270/Q2VT1WCQ | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50530861 (CHEMBL4452350) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.46E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50530861 (CHEMBL4452350) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.46E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dihydroorotate dehydrogenase (quinone), mitochondrial (Plasmodium falciparum (isolate 3D7)) | BDBM50507740 (CHEMBL4539458) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Turin Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ... | Eur J Med Chem 163: 266-280 (2019) Article DOI: 10.1016/j.ejmech.2018.11.044 BindingDB Entry DOI: 10.7270/Q2VT1WCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-lactamase TEM (Escherichia coli) | BDBM50247467 (CHEMBL4083640) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Leeds Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged bacterial Escherichia coli TEM-1 (24 to 286 residues) expressed in Escherichia coli BL21 (DE3) cells ... | J Med Chem 61: 1255-1260 (2018) Article DOI: 10.1021/acs.jmedchem.7b01728 BindingDB Entry DOI: 10.7270/Q2GQ716Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50530859 (CHEMBL4561900) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 6.34E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50530859 (CHEMBL4561900) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 6.34E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50530859 (CHEMBL4561900) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | 6.65E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50530859 (CHEMBL4561900) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | 6.65E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50530861 (CHEMBL4452350) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.38E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50530861 (CHEMBL4452350) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.38E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dihydroorotate dehydrogenase (quinone), mitochondrial (Plasmodium falciparum (isolate 3D7)) | BDBM50507745 (CHEMBL4517934) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Turin Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ... | Eur J Med Chem 163: 266-280 (2019) Article DOI: 10.1016/j.ejmech.2018.11.044 BindingDB Entry DOI: 10.7270/Q2VT1WCQ | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Dihydroorotate dehydrogenase (quinone), mitochondrial (Plasmodium falciparum (isolate 3D7)) | BDBM50507737 (CHEMBL4514989) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Turin Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ... | Eur J Med Chem 163: 266-280 (2019) Article DOI: 10.1016/j.ejmech.2018.11.044 BindingDB Entry DOI: 10.7270/Q2VT1WCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50530860 (CHEMBL4461782) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.77E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50530860 (CHEMBL4461782) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.77E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dihydroorotate dehydrogenase (quinone), mitochondrial (Plasmodium falciparum (isolate 3D7)) | BDBM50507736 (CHEMBL4457827) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Turin Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ... | Eur J Med Chem 163: 266-280 (2019) Article DOI: 10.1016/j.ejmech.2018.11.044 BindingDB Entry DOI: 10.7270/Q2VT1WCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dihydroorotate dehydrogenase (quinone), mitochondrial (Plasmodium falciparum (isolate 3D7)) | BDBM50507738 (CHEMBL4451149) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Turin Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ... | Eur J Med Chem 163: 266-280 (2019) Article DOI: 10.1016/j.ejmech.2018.11.044 BindingDB Entry DOI: 10.7270/Q2VT1WCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase, cytoplasmic (Homo sapiens) | BDBM50530864 (CHEMBL4467050) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of human N-terminal polyHis-tagged SerRS expressed in Escherichia coli BL21 (DE3) using Ap4A as substrate in presence of serine by leucono... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase, cytoplasmic (Homo sapiens) | BDBM50530864 (CHEMBL4467050) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of human N-terminal polyHis-tagged SerRS expressed in Escherichia coli BL21 (DE3) using Ap4A as substrate in presence of serine by leucono... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dihydroorotate dehydrogenase (quinone), mitochondrial (Plasmodium falciparum (isolate 3D7)) | BDBM50507734 (CHEMBL4514633) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Turin Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ... | Eur J Med Chem 163: 266-280 (2019) Article DOI: 10.1016/j.ejmech.2018.11.044 BindingDB Entry DOI: 10.7270/Q2VT1WCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50530863 (CHEMBL4449289) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.24E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50530863 (CHEMBL4449289) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.24E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-lactamase TEM (Escherichia coli) | BDBM50247459 (CHEMBL4065946) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.28E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Leeds Curated by ChEMBL | Assay Description Inhibition of recombinant N-terminal His-tagged bacterial Escherichia coli TEM-1 (24 to 286 residues) expressed in Escherichia coli BL21 (DE3) cells ... | J Med Chem 61: 1255-1260 (2018) Article DOI: 10.1021/acs.jmedchem.7b01728 BindingDB Entry DOI: 10.7270/Q2GQ716Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dihydroorotate dehydrogenase (quinone), mitochondrial (Plasmodium falciparum (isolate 3D7)) | BDBM50507732 (CHEMBL4436588) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Turin Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ... | Eur J Med Chem 163: 266-280 (2019) Article DOI: 10.1016/j.ejmech.2018.11.044 BindingDB Entry DOI: 10.7270/Q2VT1WCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50530863 (CHEMBL4449289) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.62E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50530863 (CHEMBL4449289) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.62E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-lactamase OXA-10 (Pseudomonas aeruginosa) | BDBM50247467 (CHEMBL4083640) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.73E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Leeds Curated by ChEMBL | Assay Description Inhibition of recombinant Pseudomonas aeruginosa OXA-10 expressed in Escherichia coli BL21 (DE3) cells using FC5 as substrate preincubated up to 360 ... | J Med Chem 61: 1255-1260 (2018) Article DOI: 10.1021/acs.jmedchem.7b01728 BindingDB Entry DOI: 10.7270/Q2GQ716Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acyl-[acyl-carrier-protein]--UDP-N-acetylglucosamine O-acyltransferase (Escherichia coli (Enterobacteria)) | BDBM50577526 (CHEMBL4871671) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant Escherichia coli LpxA using UDP-GlcNAc as substrate incubated for 30 mins by spectrophotometric method | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00888 BindingDB Entry DOI: 10.7270/Q2N301RT | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50530860 (CHEMBL4461782) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.27E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Staphylococcus aureus (strain NCTC 8325 / PS 47)) | BDBM50530860 (CHEMBL4461782) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.27E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase, cytoplasmic (Homo sapiens) | BDBM50530866 (CHEMBL4529844) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.73E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warwick Curated by ChEMBL | Assay Description Inhibition of human N-terminal polyHis-tagged SerRS expressed in Escherichia coli BL21 (DE3) using Ap4A as substrate in presence of serine by leucono... | J Med Chem 62: 9703-9717 (2019) Article DOI: 10.1021/acs.jmedchem.9b01131 BindingDB Entry DOI: 10.7270/Q2GX4G11 | |||||||||||
More data for this Ligand-Target Pair |
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