Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Prothrombin (Homo sapiens (Human)) | BDBM50010247 (CHEMBL3247184) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | PubMed | 3.98E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human thrombin assessed as decrease in p-nitrophenol production using Nalpha-Z-L-Lys-ONp as substrate ... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM50010252 (CHEMBL3247187) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human plasmin assessed as assessed as decrease in p-nitrophenol production using N-Z-L-Tyr-ONp as subs... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50010249 (CHEMBL3247185) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 6.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human thrombin assessed as decrease in p-nitrophenol production using Nalpha-Z-L-Lys-ONp as substrate ... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM50010258 (CHEMBL3247193) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM50010258 (CHEMBL3247193) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM8527 (n,n-dimethyl, m-aminobenzamidine) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | PubMed | 1.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human plasmin assessed as assessed as decrease in p-nitrophenol production using N-Z-L-Tyr-ONp as subs... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50010258 (CHEMBL3247193) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.58E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50010253 (CHEMBL3247189) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | PubMed | 1.58E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human plasmin assessed as assessed as decrease in p-nitrophenol production using N-Z-L-Tyr-ONp as subs... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM8527 (n,n-dimethyl, m-aminobenzamidine) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | PubMed | 1.99E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human plasmin assessed as assessed as decrease in p-nitrophenol production using N-Z-L-Tyr-ONp as subs... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM50010258 (CHEMBL3247193) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50010287 (CHEMBL3138844) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | PubMed | 3.16E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50010244 (CHEMBL3247181) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | PubMed | 3.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human thrombin assessed as decrease in p-nitrophenol production using Nalpha-Z-L-Lys-ONp as substrate ... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50010245 (CHEMBL3247182) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | 3.98E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human thrombin assessed as decrease in p-nitrophenol production using Nalpha-Z-L-Lys-ONp as substrate ... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM93094 (2-Guanidino-4-methylguinazoline) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | 7.65E+4 | -23.5 | n/a | n/a | n/a | n/a | n/a | 8.05 | 25.5 |
Michigan State University | Assay Description All readings were made in a Hitachi-Coleman ultraviolet-visible 101 spectrophotometer. | Biochemistry 8: 4503-10 (1969) Article DOI: 10.1021/bi00839a042 BindingDB Entry DOI: 10.7270/Q22R3Q87 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM50010256 (CHEMBL3247192) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | 7.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM50010304 (CHEMBL3247195) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 7.94E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human thrombin assessed as decrease in p-nitrophenol production using Nalpha-Z-L-Tyr-ONp as substrate ... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM50010257 (CHEMBL1231012) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL DrugBank KEGG PC cid PC sid UniChem Similars | PubMed | 7.94E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50010249 (CHEMBL3247185) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 9.99E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human thrombin assessed as decrease in p-nitrophenol production using Nalpha-Z-L-Lys-ONp as substrate ... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM50010257 (CHEMBL1231012) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL DrugBank KEGG PC cid PC sid UniChem Similars | PubMed | 9.99E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM50010279 (CHEMBL3138975) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid UniChem Patents Similars | PubMed | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM50010287 (CHEMBL3138844) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | PubMed | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM50010250 (CHEMBL3247186) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | PubMed | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human plasmin assessed as assessed as decrease in p-nitrophenol production using N-Z-L-Tyr-ONp as subs... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50010257 (CHEMBL1231012) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL DrugBank KEGG PC cid PC sid UniChem Similars | PubMed | 1.25E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM50010250 (CHEMBL3247186) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | PubMed | 1.25E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human plasmin assessed as assessed as decrease in p-nitrophenol production using N-Z-L-Tyr-ONp as subs... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50010243 (CHEMBL3247180) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | 1.30E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human thrombin assessed as decrease in p-nitrophenol production using Nalpha-Z-L-Lys-ONp as substrate ... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM50010257 (CHEMBL1231012) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL DrugBank KEGG PC cid PC sid UniChem Similars | PubMed | 1.58E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50010247 (CHEMBL3247184) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | PubMed | 1.58E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human thrombin assessed as decrease in p-nitrophenol production using Nalpha-Z-L-Lys-ONp as substrate ... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50153443 (4-(HYDROXYMETHYL)BENZAMIDINE | 4-Hydroxymethyl-ben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MMDB PC cid PC sid PDB UniChem Patents | PubMed | 1.58E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human thrombin assessed as decrease in p-nitrophenol production using Nalpha-Z-L-Tyr-ONp as substrate ... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM50010253 (CHEMBL3247189) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | PubMed | 1.60E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM50010245 (CHEMBL3247182) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | 1.99E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human thrombin assessed as decrease in p-nitrophenol production using Nalpha-Z-L-Lys-ONp as substrate ... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM50010256 (CHEMBL3247192) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | 2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM8527 (n,n-dimethyl, m-aminobenzamidine) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | PubMed | 2.51E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human plasmin assessed as assessed as decrease in p-nitrophenol production using N-Z-L-Tyr-ONp as subs... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM50010303 (CHEMBL3247194) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 2.51E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM50010250 (CHEMBL3247186) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | PubMed | 3.16E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human plasmin assessed as assessed as decrease in p-nitrophenol production using N-Z-L-Tyr-ONp as subs... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50010252 (CHEMBL3247187) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 3.16E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human plasmin assessed as assessed as decrease in p-nitrophenol production using N-Z-L-Tyr-ONp as subs... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50038002 (Benzamidine (Protonated) | CHEMBL20936 | CHEMBL537...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid UniChem Patents Similars | PubMed | 3.16E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human plasmin assessed as assessed as decrease in p-nitrophenol production using N-Z-L-Tyr-ONp as subs... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM93100 (N-z-L-Tyr) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | 3.70E+5 | -19.6 | n/a | n/a | n/a | n/a | n/a | 8.05 | 25.5 |
Michigan State University | Assay Description All readings were made in a Hitachi-Coleman ultraviolet-visible 101 spectrophotometer. | Biochemistry 8: 4503-10 (1969) Article DOI: 10.1021/bi00839a042 BindingDB Entry DOI: 10.7270/Q22R3Q87 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM50038002 (Benzamidine (Protonated) | CHEMBL20936 | CHEMBL537...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid UniChem Patents Similars | PubMed | 3.98E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human plasmin assessed as assessed as decrease in p-nitrophenol production using N-Z-L-Tyr-ONp as subs... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM50010244 (CHEMBL3247181) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | PubMed | 3.98E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human thrombin assessed as decrease in p-nitrophenol production using Nalpha-Z-L-Lys-ONp as substrate ... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM50038002 (Benzamidine (Protonated) | CHEMBL20936 | CHEMBL537...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid UniChem Patents Similars | PubMed | 5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human plasmin assessed as assessed as decrease in p-nitrophenol production using N-Z-L-Tyr-ONp as subs... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50010250 (CHEMBL3247186) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | PubMed | 5.01E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human plasmin assessed as assessed as decrease in p-nitrophenol production using N-Z-L-Tyr-ONp as subs... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM93095 (Alpha-Phenylguanidine) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Similars | Article PubMed | 5.48E+5 | -18.6 | n/a | n/a | n/a | n/a | n/a | 8.05 | 25.5 |
Michigan State University | Assay Description All readings were made in a Hitachi-Coleman ultraviolet-visible 101 spectrophotometer. | Biochemistry 8: 4503-10 (1969) Article DOI: 10.1021/bi00839a042 BindingDB Entry DOI: 10.7270/Q22R3Q87 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM772 (Benzamidine | CHEMBL79897 | [amino(phenyl)methylid...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 6.03E+5 | -18.4 | n/a | n/a | n/a | n/a | n/a | 8.05 | 25.5 |
Michigan State University | Assay Description All readings were made in a Hitachi-Coleman ultraviolet-visible 101 spectrophotometer. | Biochemistry 8: 4503-10 (1969) Article DOI: 10.1021/bi00839a042 BindingDB Entry DOI: 10.7270/Q22R3Q87 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50010255 (CHEMBL3247191) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | PubMed | 6.30E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM50010255 (CHEMBL3247191) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | PubMed | 6.30E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM50010256 (CHEMBL3247192) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | 6.30E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human activated C1s subunit of first complement component assessed as decrease in p-nitrophenol produc... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM50010253 (CHEMBL3247189) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | PubMed | 6.30E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human plasmin assessed as assessed as decrease in p-nitrophenol production using N-Z-L-Tyr-ONp as subs... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Complement C1s subcomponent (Homo sapiens (Human)) | BDBM50010249 (CHEMBL3247185) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 6.30E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human plasmin assessed as assessed as decrease in p-nitrophenol production using N-Z-L-Tyr-ONp as subs... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50010246 (CHEMBL3247183) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | PubMed | 7.94E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human thrombin assessed as decrease in p-nitrophenol production using Nalpha-Z-L-Lys-ONp as substrate ... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Homo sapiens (Human)) | BDBM50153443 (4-(HYDROXYMETHYL)BENZAMIDINE | 4-Hydroxymethyl-ben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MMDB PC cid PC sid PDB UniChem Patents | PubMed | 9.99E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Competitive inhibition of esterase activity of human thrombin assessed as decrease in p-nitrophenol production using Nalpha-Z-L-Tyr-ONp as substrate ... | J Med Chem 21: 1202-7 (1979) BindingDB Entry DOI: 10.7270/Q2ST7RCQ | |||||||||||
More data for this Ligand-Target Pair |
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