Compile Data Set for Download or QSAR

Found 80 hits with Last Name = 'bolinger' and Initial = 'jd'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325104 (CHEMBL1223159 | N-(4-(N-cyclohexylsulfamoyl)phenyl...) Show SMILES O=C(Nc1ccc(cc1)S(=O)(=O)NC1CCCCC1)c1ccccn1 Show InChI InChI=1S/C18H21N3O3S/c22-18(17-8-4-5-13-19-17)20-14-9-11-16(12-10-14)25(23,24)21-15-6-2-1-3-7-15/h4-5,8-13,15,21H,1-3,6-7H2,(H,20,22)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	1.03E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325105 (CHEMBL1223385 | N-(4-((2-chlorophenylsulfonyl)meth...) Show SMILES Clc1ccccc1S(=O)(=O)Cc1ccc(NC(=O)c2ccccn2)cc1 Show InChI InChI=1S/C19H15ClN2O3S/c20-16-5-1-2-7-18(16)26(24,25)13-14-8-10-15(11-9-14)22-19(23)17-6-3-4-12-21-17/h1-12H,13H2,(H,22,23)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	2.17E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325106 (CHEMBL1223384 | N-(4-(2-chlorobenzylsulfonyl)pheny...) Show SMILES Clc1ccccc1CS(=O)(=O)c1ccc(NC(=O)c2ccccn2)cc1 Show InChI InChI=1S/C19H15ClN2O3S/c20-17-6-2-1-5-14(17)13-26(24,25)16-10-8-15(9-11-16)22-19(23)18-7-3-4-12-21-18/h1-12H,13H2,(H,22,23)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	237	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325107 (CHEMBL1223383 | N-(4-chloro-3-(N-(2-chlorophenyl)s...) Show SMILES Clc1ccccc1NS(=O)(=O)c1cc(NC(=O)c2ccccn2)ccc1Cl Show InChI InChI=1S/C18H13Cl2N3O3S/c19-13-5-1-2-6-15(13)23-27(25,26)17-11-12(8-9-14(17)20)22-18(24)16-7-3-4-10-21-16/h1-11,23H,(H,22,24)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	731	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325108 (CHEMBL1223381 | N-(3-chloro-4-(N-(2-chlorophenyl)s...) Show SMILES Clc1ccccc1NS(=O)(=O)c1ccc(NC(=O)c2ccccn2)cc1Cl Show InChI InChI=1S/C18H13Cl2N3O3S/c19-13-5-1-2-6-15(13)23-27(25,26)17-9-8-12(11-14(17)20)22-18(24)16-7-3-4-10-21-16/h1-11,23H,(H,22,24)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	19.8	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325109 (CHEMBL1223316 | N-(3-methoxy-4-(N-(2-methoxyphenyl...) Show SMILES COc1ccccc1NS(=O)(=O)c1ccc(NC(=O)c2ccccn2)cc1OC Show InChI InChI=1S/C20H19N3O5S/c1-27-17-9-4-3-7-15(17)23-29(25,26)19-11-10-14(13-18(19)28-2)22-20(24)16-8-5-6-12-21-16/h3-13,23H,1-2H3,(H,22,24)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	132	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325110 (CHEMBL1223315 | N-(4-(N-(2-chlorophenyl)-N-methyls...) Show SMILES CN(c1ccccc1Cl)S(=O)(=O)c1ccc(NC(=O)c2nccs2)cc1 Show InChI InChI=1S/C17H14ClN3O3S2/c1-21(15-5-3-2-4-14(15)18)26(23,24)13-8-6-12(7-9-13)20-16(22)17-19-10-11-25-17/h2-11H,1H3,(H,20,22)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	686	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325111 (CHEMBL1223314 | N-(4-(N-(2-chlorophenyl)-N-methyls...) Show SMILES CN(c1ccccc1Cl)S(=O)(=O)c1ccc(NC(=O)c2ccncn2)cc1 Show InChI InChI=1S/C18H15ClN4O3S/c1-23(17-5-3-2-4-15(17)19)27(25,26)14-8-6-13(7-9-14)22-18(24)16-10-11-20-12-21-16/h2-12H,1H3,(H,22,24)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	990	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325112 (CHEMBL1223313 | N-(4-(N-(2-chlorophenyl)sulfamoyl)...) Show SMILES Clc1ccccc1NS(=O)(=O)c1ccc(NC(=O)c2ccsc2)cc1 Show InChI InChI=1S/C17H13ClN2O3S2/c18-15-3-1-2-4-16(15)20-25(22,23)14-7-5-13(6-8-14)19-17(21)12-9-10-24-11-12/h1-11,20H,(H,19,21)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	269	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325113 (CHEMBL1223312 | N-(4-(N-(2-chlorophenyl)sulfamoyl)...) Show SMILES Clc1ccccc1NS(=O)(=O)c1ccc(NC(=O)c2nccs2)cc1 Show InChI InChI=1S/C16H12ClN3O3S2/c17-13-3-1-2-4-14(13)20-25(22,23)12-7-5-11(6-8-12)19-15(21)16-18-9-10-24-16/h1-10,20H,(H,19,21)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	77.4	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325114 (CHEMBL1223243 | N-(4-(N-(2-chlorophenyl)sulfamoyl)...) Show SMILES Clc1ccccc1NS(=O)(=O)c1ccc(NC(=O)c2ccncn2)cc1 Show InChI InChI=1S/C17H13ClN4O3S/c18-14-3-1-2-4-15(14)22-26(24,25)13-7-5-12(6-8-13)21-17(23)16-9-10-19-11-20-16/h1-11,22H,(H,21,23)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	478	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325115 (CHEMBL1223241 | N-(4-(N-(2-chlorophenyl)sulfamoyl)...) Show SMILES Fc1cccc(n1)C(=O)Nc1ccc(cc1)S(=O)(=O)Nc1ccccc1Cl Show InChI InChI=1S/C18H13ClFN3O3S/c19-14-4-1-2-5-15(14)23-27(25,26)13-10-8-12(9-11-13)21-18(24)16-6-3-7-17(20)22-16/h1-11,23H,(H,21,24)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	122	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325116 (CHEMBL1223164 | N-(4-(4-methylpiperidin-1-ylsulfon...) Show SMILES CC1CCN(CC1)S(=O)(=O)c1ccc(NC(=O)c2ccccn2)cc1 Show InChI InChI=1S/C18H21N3O3S/c1-14-9-12-21(13-10-14)25(23,24)16-7-5-15(6-8-16)20-18(22)17-4-2-3-11-19-17/h2-8,11,14H,9-10,12-13H2,1H3,(H,20,22)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	372	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325117 (CHEMBL1223163 | N-(4-(N-(2-methoxyethyl)sulfamoyl)...) Show SMILES COCCNS(=O)(=O)c1ccc(NC(=O)c2ccccn2)cc1 Show InChI InChI=1S/C15H17N3O4S/c1-22-11-10-17-23(20,21)13-7-5-12(6-8-13)18-15(19)14-4-2-3-9-16-14/h2-9,17H,10-11H2,1H3,(H,18,19)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325118 (CHEMBL1223162 | N-(4-(N-(cyclopropylmethyl)sulfamo...) Show SMILES O=C(Nc1ccc(cc1)S(=O)(=O)NCC1CC1)c1ccccn1 Show InChI InChI=1S/C16H17N3O3S/c20-16(15-3-1-2-10-17-15)19-13-6-8-14(9-7-13)23(21,22)18-11-12-4-5-12/h1-3,6-10,12,18H,4-5,11H2,(H,19,20)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	>5.00E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325119 (CHEMBL1223161 | N-(4-(N-cyclobutylsulfamoyl)phenyl...) Show SMILES O=C(Nc1ccc(cc1)S(=O)(=O)NC1CCC1)c1ccccn1 Show InChI InChI=1S/C16H17N3O3S/c20-16(15-6-1-2-11-17-15)18-12-7-9-14(10-8-12)23(21,22)19-13-4-3-5-13/h1-2,6-11,13,19H,3-5H2,(H,18,20)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	>5.00E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325120 (CHEMBL1223160 | N-(4-(N-cyclopropylsulfamoyl)pheny...) Show SMILES O=C(Nc1ccc(cc1)S(=O)(=O)NC1CC1)c1ccccn1 Show InChI InChI=1S/C15H15N3O3S/c19-15(14-3-1-2-10-16-14)17-11-6-8-13(9-7-11)22(20,21)18-12-4-5-12/h1-3,6-10,12,18H,4-5H2,(H,17,19)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325121 (CHEMBL1223085 | N-(4-(N-(2,5-difluorophenyl)sulfam...) Show SMILES Fc1ccc(F)c(NS(=O)(=O)c2ccc(NC(=O)c3ccccn3)cc2)c1 Show InChI InChI=1S/C18H13F2N3O3S/c19-12-4-9-15(20)17(11-12)23-27(25,26)14-7-5-13(6-8-14)22-18(24)16-3-1-2-10-21-16/h1-11,23H,(H,22,24)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	325	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325122 (CHEMBL1223084 | N-(4-(N-(2-fluorophenyl)sulfamoyl)...) Show SMILES Fc1ccccc1NS(=O)(=O)c1ccc(NC(=O)c2ccccn2)cc1 Show InChI InChI=1S/C18H14FN3O3S/c19-15-5-1-2-6-16(15)22-26(24,25)14-10-8-13(9-11-14)21-18(23)17-7-3-4-12-20-17/h1-12,22H,(H,21,23)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	206	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325123 (CHEMBL1223083 | N-(4-(N-(2-chlorophenyl)sulfamoyl)...) Show SMILES Clc1ccccc1NS(=O)(=O)c1ccc(NC(=O)c2ccccn2)cc1 Show InChI InChI=1S/C18H14ClN3O3S/c19-15-5-1-2-6-16(15)22-26(24,25)14-10-8-13(9-11-14)21-18(23)17-7-3-4-12-20-17/h1-12,22H,(H,21,23)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	27	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325124 (CHEMBL1223015 | N-(4-(N-phenylsulfamoyl)phenyl)pic...) Show SMILES O=C(Nc1ccc(cc1)S(=O)(=O)Nc1ccccc1)c1ccccn1 Show InChI InChI=1S/C18H15N3O3S/c22-18(17-8-4-5-13-19-17)20-14-9-11-16(12-10-14)25(23,24)21-15-6-2-1-3-7-15/h1-13,21H,(H,20,22)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	177	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325125 (CHEMBL1223014 | N-(4-(N-mesitylsulfamoyl)phenyl)pi...) Show SMILES Cc1cc(C)c(NS(=O)(=O)c2ccc(NC(=O)c3ccccn3)cc2)c(C)c1 Show InChI InChI=1S/C21H21N3O3S/c1-14-12-15(2)20(16(3)13-14)24-28(26,27)18-9-7-17(8-10-18)23-21(25)19-6-4-5-11-22-19/h4-13,24H,1-3H3,(H,23,25)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	159	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50325126 (CHEMBL1223013 | N-(4-(N-mesitylsulfamoyl)phenyl)fu...) Show SMILES Cc1cc(C)c(NS(=O)(=O)c2ccc(NC(=O)c3ccco3)cc2)c(C)c1 Show InChI InChI=1S/C20H20N2O4S/c1-13-11-14(2)19(15(3)12-13)22-27(24,25)17-8-6-16(7-9-17)21-20(23)18-5-4-10-26-18/h4-12,22H,1-3H3,(H,21,23)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	5.96E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells assessed as potentiation of glutamate-induced calcium mobilization				Bioorg Med Chem Lett 20: 5175-8 (2010) Article DOI: 10.1016/j.bmcl.2010.07.007 BindingDB Entry DOI: 10.7270/Q2PZ591J
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50336625 (5-bromo-N-(4-(2-chlorobenzamido)-3-methoxyphenyl)f...) Show SMILES COc1cc(NC(=O)c2ccc(Br)o2)ccc1NC(=O)c1ccccc1Cl Show InChI InChI=1S/C19H14BrClN2O4/c1-26-16-10-11(22-19(25)15-8-9-17(20)27-15)6-7-14(16)23-18(24)12-4-2-3-5-13(12)21/h2-10H,1H3,(H,22,25)(H,23,24)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.44E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50336626 (CHEMBL1385271 | N-(4-(2-chlorobenzamido)-3-methoxy...) Show SMILES COc1cc(NC(=O)c2ccco2)ccc1NC(=O)c1ccccc1Cl Show InChI InChI=1S/C19H15ClN2O4/c1-25-17-11-12(21-19(24)16-7-4-10-26-16)8-9-15(17)22-18(23)13-5-2-3-6-14(13)20/h2-11H,1H3,(H,21,24)(H,22,23)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	977	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM77724 (MLS000592149 | N-[(5-nitro-2-thienyl)methyleneamin...) Show SMILES [O-][N+](=O)c1ccc(\C=N\NC(=O)c2cccnc2)s1 Show InChI InChI=1S/C11H8N4O3S/c16-11(8-2-1-5-12-6-8)14-13-7-9-3-4-10(19-9)15(17)18/h1-7H,(H,14,16)/b13-7+	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.17E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50336628 (CHEMBL1672232 | N-(4-(2-chlorobenzamido)-3-methoxy...) Show SMILES COc1cc(NC(=O)c2nccs2)ccc1NC(=O)c1ccccc1Cl Show InChI InChI=1S/C18H14ClN3O3S/c1-25-15-10-11(21-17(24)18-20-8-9-26-18)6-7-14(15)22-16(23)12-4-2-3-5-13(12)19/h2-10H,1H3,(H,21,24)(H,22,23)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	627	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50336629 (CHEMBL1672233 | N-(4-(2-chlorobenzamido)-3-methoxy...) Show SMILES COc1cc(NC(=O)c2cscn2)ccc1NC(=O)c1ccccc1Cl Show InChI InChI=1S/C18H14ClN3O3S/c1-25-16-8-11(21-18(24)15-9-26-10-20-15)6-7-14(16)22-17(23)12-4-2-3-5-13(12)19/h2-10H,1H3,(H,21,24)(H,22,23)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	845	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM55082 (N-[4-[(2-chlorobenzoyl)amino]-3-methoxy-phenyl]pic...) Show SMILES COc1cc(NC(=O)c2ccccn2)ccc1NC(=O)c1ccccc1Cl Show InChI InChI=1S/C20H16ClN3O3/c1-27-18-12-13(23-20(26)17-8-4-5-11-22-17)9-10-16(18)24-19(25)14-6-2-3-7-15(14)21/h2-12H,1H3,(H,23,26)(H,24,25)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	99.5	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50336630 (CHEMBL1672235 | N-(4-(2-chlorobenzamido)-3-methoxy...) Show SMILES COc1cc(NC(=O)c2cnccn2)ccc1NC(=O)c1ccccc1Cl Show InChI InChI=1S/C19H15ClN4O3/c1-27-17-10-12(23-19(26)16-11-21-8-9-22-16)6-7-15(17)24-18(25)13-4-2-3-5-14(13)20/h2-11H,1H3,(H,23,26)(H,24,25)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.78E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50336631 (CHEMBL1672236 | N-(4-(2-chlorobenzamido)-3-methoxy...) Show SMILES COc1cc(NC(=O)c2ccncn2)ccc1NC(=O)c1ccccc1Cl Show InChI InChI=1S/C19H15ClN4O3/c1-27-17-10-12(23-19(26)16-8-9-21-11-22-16)6-7-15(17)24-18(25)13-4-2-3-5-14(13)20/h2-11H,1H3,(H,23,26)(H,24,25)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.33E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50336632 (2-chloro-N-(4-(cyclohexanecarboxamido)-2-methoxyph...) Show SMILES COc1cc(NC(=O)C2CCCCC2)ccc1NC(=O)c1ccccc1Cl Show InChI InChI=1S/C21H23ClN2O3/c1-27-19-13-15(23-20(25)14-7-3-2-4-8-14)11-12-18(19)24-21(26)16-9-5-6-10-17(16)22/h5-6,9-14H,2-4,7-8H2,1H3,(H,23,25)(H,24,26)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	1.12E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50263669 ((1aS,7aS)-7-(hydroxyimino)-N-phenyl-1,1a,7,7a-tetr...) Show SMILES O=NC1[C@@H]2C[C@@]2(Oc2ccccc12)C(=O)Nc1ccccc1 |r| Show InChI InChI=1S/C17H14N2O3/c20-16(18-11-6-2-1-3-7-11)17-10-13(17)15(19-21)12-8-4-5-9-14(12)22-17/h1-9,13,15H,10H2,(H,18,20)/t13-,15?,17-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	4.74E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM55083 (N-[3-chloranyl-4-[(2-chlorophenyl)carbonylamino]ph...) Show SMILES Clc1ccccc1C(=O)Nc1ccc(NC(=O)c2ccccn2)cc1Cl Show InChI InChI=1S/C19H13Cl2N3O2/c20-14-6-2-1-5-13(14)18(25)24-16-9-8-12(11-15(16)21)23-19(26)17-7-3-4-10-22-17/h1-11H,(H,23,26)(H,24,25)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	517	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50336633 (CHEMBL1672239 | N-(4-(2-chlorobenzamido)-3-(triflu...) Show SMILES FC(F)(F)c1cc(NC(=O)c2ccccn2)ccc1NC(=O)c1ccccc1Cl Show InChI InChI=1S/C20H13ClF3N3O2/c21-15-6-2-1-5-13(15)18(28)27-16-9-8-12(11-14(16)20(22,23)24)26-19(29)17-7-3-4-10-25-17/h1-11H,(H,26,29)(H,27,28)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	2.09E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50336634 (CHEMBL1672240 | N-(4-(2-chlorobenzamido)phenyl)pic...) Show SMILES Clc1ccccc1C(=O)Nc1ccc(NC(=O)c2ccccn2)cc1 Show InChI InChI=1S/C19H14ClN3O2/c20-16-6-2-1-5-15(16)18(24)22-13-8-10-14(11-9-13)23-19(25)17-7-3-4-12-21-17/h1-12H,(H,22,24)(H,23,25)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.61E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM55084 (N-[4-[(2-chlorobenzoyl)amino]-3-fluoro-phenyl]pico...) Show SMILES Fc1cc(NC(=O)c2ccccn2)ccc1NC(=O)c1ccccc1Cl Show InChI InChI=1S/C19H13ClFN3O2/c20-14-6-2-1-5-13(14)18(25)24-16-9-8-12(11-15(16)21)23-19(26)17-7-3-4-10-22-17/h1-11H,(H,23,26)(H,24,25)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	556	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50336635 (CHEMBL1672242 | N-(3-chloro-4-(2-methylbenzamido)p...) Show SMILES Cc1ccccc1C(=O)Nc1ccc(NC(=O)c2ccccn2)cc1Cl Show InChI InChI=1S/C20H16ClN3O2/c1-13-6-2-3-7-15(13)19(25)24-17-10-9-14(12-16(17)21)23-20(26)18-8-4-5-11-22-18/h2-12H,1H3,(H,23,26)(H,24,25)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	958	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50336636 (CHEMBL1672243 | N-(3-chloro-4-(cyclohexanecarboxam...) Show SMILES Clc1cc(NC(=O)c2ccccn2)ccc1NC(=O)C1CCCCC1 Show InChI InChI=1S/C19H20ClN3O2/c20-15-12-14(22-19(25)17-8-4-5-11-21-17)9-10-16(15)23-18(24)13-6-2-1-3-7-13/h4-5,8-13H,1-3,6-7H2,(H,22,25)(H,23,24)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	426	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50336614 (CHEMBL1672244 | N-(4-benzamido-3-chlorophenyl)pico...) Show SMILES Clc1cc(NC(=O)c2ccccn2)ccc1NC(=O)c1ccccc1 Show InChI InChI=1S/C19H14ClN3O2/c20-15-12-14(22-19(25)17-8-4-5-11-21-17)9-10-16(15)23-18(24)13-6-2-1-3-7-13/h1-12H,(H,22,25)(H,23,24)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	361	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50336615 (CHEMBL1672245 | N-(3-chloro-4-(2-chloro-4-fluorobe...) Show SMILES Fc1ccc(C(=O)Nc2ccc(NC(=O)c3ccccn3)cc2Cl)c(Cl)c1 Show InChI InChI=1S/C19H12Cl2FN3O2/c20-14-9-11(22)4-6-13(14)18(26)25-16-7-5-12(10-15(16)21)24-19(27)17-3-1-2-8-23-17/h1-10H,(H,24,27)(H,25,26)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	114	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat))	BDBM50378891 (CHEMBL1909430) Show SMILES Fc1ccc(C(=O)Nc2ccc(NC(=O)c3ccccn3)cc2Cl)c(F)c1 Show InChI InChI=1S/C19H12ClF2N3O2/c20-14-10-12(24-19(27)17-3-1-2-8-23-17)5-7-16(14)25-18(26)13-6-4-11(21)9-15(13)22/h1-10H,(H,24,27)(H,25,26)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	2.10E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of rat mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat))	BDBM50378892 (CHEMBL1909431) Show SMILES Clc1cc(Cl)cc(c1)C(=O)Nc1ccc(NC(=O)c2ccccn2)cc1Cl Show InChI InChI=1S/C19H12Cl3N3O2/c20-12-7-11(8-13(21)9-12)18(26)25-16-5-4-14(10-15(16)22)24-19(27)17-3-1-2-6-23-17/h1-10H,(H,24,27)(H,25,26)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	2.34E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of rat mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat))	BDBM50378893 (CHEMBL1909433) Show SMILES Clc1cc(NC(=O)c2ccccn2)ccc1NC(=O)c1cncs1 Show InChI InChI=1S/C16H11ClN4O2S/c17-11-7-10(20-15(22)13-3-1-2-6-19-13)4-5-12(11)21-16(23)14-8-18-9-24-14/h1-9H,(H,20,22)(H,21,23)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.73E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of rat mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat))	BDBM50378894 (CHEMBL1909434) Show SMILES Clc1cc(NC(=O)c2ccccn2)ccc1NC(=O)c1nccs1 Show InChI InChI=1S/C16H11ClN4O2S/c17-11-9-10(20-14(22)13-3-1-2-6-18-13)4-5-12(11)21-15(23)16-19-7-8-24-16/h1-9H,(H,20,22)(H,21,23)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	533	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of rat mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat))	BDBM50378895 (CHEMBL1909435) Show SMILES Clc1cc(NC(=O)c2ccccn2)ccc1NC(=O)c1cccs1 Show InChI InChI=1S/C17H12ClN3O2S/c18-12-10-11(20-16(22)14-4-1-2-8-19-14)6-7-13(12)21-17(23)15-5-3-9-24-15/h1-10H,(H,20,22)(H,21,23)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.13E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of rat mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat))	BDBM50378896 (CHEMBL1909436) Show SMILES Cn1c(cc2ccccc12)C(=O)Nc1ccc(NC(=O)c2ccccn2)cc1Cl Show InChI InChI=1S/C22H17ClN4O2/c1-27-19-8-3-2-6-14(19)12-20(27)22(29)26-17-10-9-15(13-16(17)23)25-21(28)18-7-4-5-11-24-18/h2-13H,1H3,(H,25,28)(H,26,29)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	2.97E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of rat mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat))	BDBM50378897 (CHEMBL1909437) Show SMILES Clc1cc(NC(=O)c2ccccn2)ccc1NC(=O)c1ccc(o1)-c1ccccc1 Show InChI InChI=1S/C23H16ClN3O3/c24-17-14-16(26-22(28)19-8-4-5-13-25-19)9-10-18(17)27-23(29)21-12-11-20(30-21)15-6-2-1-3-7-15/h1-14H,(H,26,28)(H,27,29)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	3.35E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of rat mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat))	BDBM50336623 (CHEMBL1672256 | N-(1-(2-chloro-4-fluorobenzoyl)-1H...) Show SMILES Fc1ccc(C(=O)n2ccc3cc(NC(=O)c4ccccn4)ccc23)c(Cl)c1 Show InChI InChI=1S/C21H13ClFN3O2/c22-17-12-14(23)4-6-16(17)21(28)26-10-8-13-11-15(5-7-19(13)26)25-20(27)18-3-1-2-9-24-18/h1-12H,(H,25,27)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	1.66E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of rat mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat))	BDBM50336624 (CHEMBL1672257 | N-(1-(2-methoxybenzoyl)-1H-indol-5...) Show SMILES COc1ccccc1C(=O)n1ccc2cc(NC(=O)c3ccccn3)ccc12 Show InChI InChI=1S/C22H17N3O3/c1-28-20-8-3-2-6-17(20)22(27)25-13-11-15-14-16(9-10-19(15)25)24-21(26)18-7-4-5-12-23-18/h2-14H,1H3,(H,24,26)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	1.34E+3	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Positive allosteric modulation of rat mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization				J Med Chem 54: 1106-10 (2011) Article DOI: 10.1021/jm101271s BindingDB Entry DOI: 10.7270/Q27P90C1
					More data for this Ligand-Target Pair

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