BindingDB PrimarySearch

Found 37 hits with Last Name = 'brunschwig' and Initial = 'c'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50030836 (CHEMBL3355639) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	400	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of human ERG potassium channel by ionworks patch-clamp electrophysiology assay				J Med Chem 58: 8713-22 (2015) Article DOI: 10.1021/acs.jmedchem.5b01605 BindingDB Entry DOI: 10.7270/Q24F1SJD
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50554417 (CHEMBL4758157) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	400	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG by patch clamp method				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01411 BindingDB Entry DOI: 10.7270/Q2TB1BKN
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50554407 (CHEMBL4746185) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	400	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG by patch clamp method				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01411 BindingDB Entry DOI: 10.7270/Q2TB1BKN
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50503392 (CHEMBL4545990) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	500	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of human ERG by patch clamp electrophysiology				J Med Chem 61: 9371-9385 (2018) Article DOI: 10.1021/acs.jmedchem.8b01333 BindingDB Entry DOI: 10.7270/Q2222Z1Q
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50129589 (CHEMBL3628223) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	500	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of human ERG potassium channel by ionworks patch-clamp electrophysiology assay				J Med Chem 58: 8713-22 (2015) Article DOI: 10.1021/acs.jmedchem.5b01605 BindingDB Entry DOI: 10.7270/Q24F1SJD
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50129559 (CHEMBL3234071) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	900	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of human ERG potassium channel by ionworks patch-clamp electrophysiology assay				J Med Chem 58: 8713-22 (2015) Article DOI: 10.1021/acs.jmedchem.5b01605 BindingDB Entry DOI: 10.7270/Q24F1SJD
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50250844 (CHEMBL4070191) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	900	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of full length human ERG expressed in CHO cells at -70 mV holding potential by patch clamp assay				J Med Chem 60: 10118-10134 (2017) Article DOI: 10.1021/acs.jmedchem.7b01347 BindingDB Entry DOI: 10.7270/Q2RR21P5
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50276209 (CHEMBL4127800) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of full length human ERG expressed in HEK293 cells assessed as reduction in tail current at holding potential of -70 mV after 6 to 7 mins ...				J Med Chem 61: 5692-5703 (2018) Article DOI: 10.1021/acs.jmedchem.8b00648 BindingDB Entry DOI: 10.7270/Q2B85BMK
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50129562 (CHEMBL3628220) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of human ERG potassium channel by ionworks patch-clamp electrophysiology assay				J Med Chem 58: 8713-22 (2015) Article DOI: 10.1021/acs.jmedchem.5b01605 BindingDB Entry DOI: 10.7270/Q24F1SJD
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50563339 (CHEMBL4756352) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.60E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG incubated for 4 hrs by fluorescene microplate reader assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00034 BindingDB Entry DOI: 10.7270/Q21N84VC
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50563340 (CHEMBL4743418) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG incubated for 4 hrs by fluorescene microplate reader assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00034 BindingDB Entry DOI: 10.7270/Q21N84VC
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50554415 (CHEMBL4757759) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG by patch clamp method				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01411 BindingDB Entry DOI: 10.7270/Q2TB1BKN
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50250842 (CHEMBL4088721) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of full length human ERG expressed in CHO cells at -70 mV holding potential by patch clamp assay				J Med Chem 60: 10118-10134 (2017) Article DOI: 10.1021/acs.jmedchem.7b01347 BindingDB Entry DOI: 10.7270/Q2RR21P5
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50554412 (CHEMBL4743530) Show SMILES Fc1ccc(cc1F)-c1nc2c(nccc2[nH]1)N1CCNCC1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG by patch clamp method				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01411 BindingDB Entry DOI: 10.7270/Q2TB1BKN
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50554416 (CHEMBL4778630) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	4.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG by patch clamp method				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01411 BindingDB Entry DOI: 10.7270/Q2TB1BKN
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50250847 (CHEMBL4088719) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.10E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of full length human ERG expressed in CHO cells at -70 mV holding potential by patch clamp assay				J Med Chem 60: 10118-10134 (2017) Article DOI: 10.1021/acs.jmedchem.7b01347 BindingDB Entry DOI: 10.7270/Q2RR21P5
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50250845 (CHEMBL4101551) Show SMILES CN(Cc1ccc(F)cc1)c1cc(ncn1)C(=O)Nc1nncs1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of full length human ERG expressed in CHO cells at -70 mV holding potential by patch clamp assay				J Med Chem 60: 10118-10134 (2017) Article DOI: 10.1021/acs.jmedchem.7b01347 BindingDB Entry DOI: 10.7270/Q2RR21P5
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50129560 (CHEMBL3628216) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	4.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of human ERG potassium channel by ionworks patch-clamp electrophysiology assay				J Med Chem 58: 8713-22 (2015) Article DOI: 10.1021/acs.jmedchem.5b01605 BindingDB Entry DOI: 10.7270/Q24F1SJD
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50554410 (CHEMBL4789774) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	5.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG by patch clamp method				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01411 BindingDB Entry DOI: 10.7270/Q2TB1BKN
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50503394 (CHEMBL4447741) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	5.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of human ERG by patch clamp electrophysiology				J Med Chem 61: 9371-9385 (2018) Article DOI: 10.1021/acs.jmedchem.8b01333 BindingDB Entry DOI: 10.7270/Q2222Z1Q
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50250843 (CHEMBL4075071) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	5.60E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of full length human ERG expressed in CHO cells at -70 mV holding potential by patch clamp assay				J Med Chem 60: 10118-10134 (2017) Article DOI: 10.1021/acs.jmedchem.7b01347 BindingDB Entry DOI: 10.7270/Q2RR21P5
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50276210 (CHEMBL4127879) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of full length human ERG expressed in HEK293 cells assessed as reduction in tail current at holding potential of -70 mV after 6 to 7 mins ...				J Med Chem 61: 5692-5703 (2018) Article DOI: 10.1021/acs.jmedchem.8b00648 BindingDB Entry DOI: 10.7270/Q2B85BMK
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50276211 (CHEMBL4128198) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of full length human ERG expressed in HEK293 cells assessed as reduction in tail current at holding potential of -70 mV after 6 to 7 mins ...				J Med Chem 61: 5692-5703 (2018) Article DOI: 10.1021/acs.jmedchem.8b00648 BindingDB Entry DOI: 10.7270/Q2B85BMK
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50276212 (CHEMBL4129258) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of full length human ERG expressed in HEK293 cells assessed as reduction in tail current at holding potential of -70 mV after 6 to 7 mins ...				J Med Chem 61: 5692-5703 (2018) Article DOI: 10.1021/acs.jmedchem.8b00648 BindingDB Entry DOI: 10.7270/Q2B85BMK
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50554413 (CHEMBL4776200) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.20E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG by patch clamp method				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01411 BindingDB Entry DOI: 10.7270/Q2TB1BKN
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50503393 (CHEMBL4575250) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of human ERG by patch clamp electrophysiology				J Med Chem 61: 9371-9385 (2018) Article DOI: 10.1021/acs.jmedchem.8b01333 BindingDB Entry DOI: 10.7270/Q2222Z1Q
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50250846 (CHEMBL4083549) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.40E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of full length human ERG expressed in CHO cells at -70 mV holding potential by patch clamp assay				J Med Chem 60: 10118-10134 (2017) Article DOI: 10.1021/acs.jmedchem.7b01347 BindingDB Entry DOI: 10.7270/Q2RR21P5
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50554414 (CHEMBL4782651) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	>3.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG by patch clamp method				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01411 BindingDB Entry DOI: 10.7270/Q2TB1BKN
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50554411 (CHEMBL4760907) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	>3.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG by patch clamp method				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01411 BindingDB Entry DOI: 10.7270/Q2TB1BKN
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50554409 (CHEMBL4758653) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	>3.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG by patch clamp method				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01411 BindingDB Entry DOI: 10.7270/Q2TB1BKN
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50554408 (CHEMBL4793720) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	>3.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG by patch clamp method				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01411 BindingDB Entry DOI: 10.7270/Q2TB1BKN
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50557136 (CHEMBL4759520) Show SMILES Cc1cc(C)n(n1)-c1nc(cc(=O)[nH]1)C(F)(F)F Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	>3.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01727 BindingDB Entry DOI: 10.7270/Q2X92FZS
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50557135 (CHEMBL2098048 \| SB-615575 \| TCMDC-142445) Show SMILES Cc1cc(C)n(n1)-c1nc(O)cc(n1)-c1ccccc1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	>3.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01727 BindingDB Entry DOI: 10.7270/Q2X92FZS
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50563338 (CHEMBL4764956) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	>3.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG incubated for 4 hrs by fluorescene microplate reader assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00034 BindingDB Entry DOI: 10.7270/Q21N84VC
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50503391 (CHEMBL4471705) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of human ERG by patch clamp electrophysiology				J Med Chem 61: 9371-9385 (2018) Article DOI: 10.1021/acs.jmedchem.8b01333 BindingDB Entry DOI: 10.7270/Q2222Z1Q
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50581159 (CHEMBL5082703) Show SMILES CN(C)C(=O)O\N=C(/C#N)c1nc2ccccc2o1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	>3.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human ERG by Ionworks electrophysiology assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00707 BindingDB Entry DOI: 10.7270/Q2P2730D
TBA					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM50129561 (CHEMBL3628219) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cape Town Curated by ChEMBL					Assay Description Inhibition of human ERG potassium channel by ionworks patch-clamp electrophysiology assay				J Med Chem 58: 8713-22 (2015) Article DOI: 10.1021/acs.jmedchem.5b01605 BindingDB Entry DOI: 10.7270/Q24F1SJD
University of Cape Town Curated by ChEMBL					More data for this Ligand-Target Pair