Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human)) | BDBM205483 (US9260417, 6) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 52 | n/a | n/a | n/a | n/a | n/a |
AMITECH THERAPEUTIC SOLUTIONS, INC. US Patent | Assay Description For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc... | US Patent US9260417 (2016) BindingDB Entry DOI: 10.7270/Q270807Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mast/stem cell growth factor receptor Kit (Homo sapiens (Human)) | BDBM205483 (US9260417, 6) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a |
AMITECH THERAPEUTIC SOLUTIONS, INC. US Patent | Assay Description For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc... | US Patent US9260417 (2016) BindingDB Entry DOI: 10.7270/Q270807Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-derived growth factor receptor alpha (Homo sapiens (Human)) | BDBM205483 (US9260417, 6) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a |
AMITECH THERAPEUTIC SOLUTIONS, INC. US Patent | Assay Description For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc... | US Patent US9260417 (2016) BindingDB Entry DOI: 10.7270/Q270807Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-derived growth factor receptor beta (Homo sapiens (Human)) | BDBM205483 (US9260417, 6) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 520 | n/a | n/a | n/a | n/a | n/a |
AMITECH THERAPEUTIC SOLUTIONS, INC. US Patent | Assay Description For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc... | US Patent US9260417 (2016) BindingDB Entry DOI: 10.7270/Q270807Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase-like 2 (Homo sapiens (Human)) | BDBM205483 (US9260417, 6) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 5.10E+3 | n/a | n/a | n/a | n/a | n/a |
AMITECH THERAPEUTIC SOLUTIONS, INC. US Patent | Assay Description For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc... | US Patent US9260417 (2016) BindingDB Entry DOI: 10.7270/Q270807Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 11B (Homo sapiens (Human)) | BDBM205483 (US9260417, 6) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 7.50E+3 | n/a | n/a | n/a | n/a | n/a |
AMITECH THERAPEUTIC SOLUTIONS, INC. US Patent | Assay Description For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc... | US Patent US9260417 (2016) BindingDB Entry DOI: 10.7270/Q270807Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human)) | BDBM205483 (US9260417, 6) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
AMITECH THERAPEUTIC SOLUTIONS, INC. US Patent | Assay Description For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc... | US Patent US9260417 (2016) BindingDB Entry DOI: 10.7270/Q270807Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase B-raf (Homo sapiens (Human)) | BDBM205483 (US9260417, 6) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
AMITECH THERAPEUTIC SOLUTIONS, INC. US Patent | Assay Description For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc... | US Patent US9260417 (2016) BindingDB Entry DOI: 10.7270/Q270807Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Macrophage colony-stimulating factor 1 receptor (Homo sapiens (Human)) | BDBM205483 (US9260417, 6) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
AMITECH THERAPEUTIC SOLUTIONS, INC. US Patent | Assay Description For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc... | US Patent US9260417 (2016) BindingDB Entry DOI: 10.7270/Q270807Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor receptor 2 (Homo sapiens (Human)) | BDBM205483 (US9260417, 6) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
AMITECH THERAPEUTIC SOLUTIONS, INC. US Patent | Assay Description For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc... | US Patent US9260417 (2016) BindingDB Entry DOI: 10.7270/Q270807Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mitogen-activated protein kinase 14 (Homo sapiens (Human)) | BDBM205483 (US9260417, 6) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
AMITECH THERAPEUTIC SOLUTIONS, INC. US Patent | Assay Description For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc... | US Patent US9260417 (2016) BindingDB Entry DOI: 10.7270/Q270807Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase PAK 1 (Homo sapiens (Human)) | BDBM205483 (US9260417, 6) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
AMITECH THERAPEUTIC SOLUTIONS, INC. US Patent | Assay Description For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc... | US Patent US9260417 (2016) BindingDB Entry DOI: 10.7270/Q270807Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proto-oncogene tyrosine-protein kinase receptor Ret (Homo sapiens (Human)) | BDBM205483 (US9260417, 6) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
AMITECH THERAPEUTIC SOLUTIONS, INC. US Patent | Assay Description For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc... | US Patent US9260417 (2016) BindingDB Entry DOI: 10.7270/Q270807Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase ABL1 (Homo sapiens (Human)) | BDBM205483 (US9260417, 6) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
AMITECH THERAPEUTIC SOLUTIONS, INC. US Patent | Assay Description For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc... | US Patent US9260417 (2016) BindingDB Entry DOI: 10.7270/Q270807Z | |||||||||||
More data for this Ligand-Target Pair |