Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Translocator protein (Rattus norvegicus (rat)) | BDBM50243005 (2-(6-Chloro-2-(4-(2-fluoroethoxy)phenyl)imidazo[1,...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Radiopharmaceuticals Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]Ro 5-4864 from peripheral benzodiazepine receptor in rat kidney membrane | J Med Chem 51: 3700-12 (2008) Article DOI: 10.1021/jm7014556 BindingDB Entry DOI: 10.7270/Q2Z037ZW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50243006 (2-(6-Chloro-2-(4-(3-fluoropropoxy)phenyl)imidazo[1...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Radiopharmaceuticals Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]PK11195 from peripheral benzodiazepine receptor in rat kidney membrane | J Med Chem 51: 3700-12 (2008) Article DOI: 10.1021/jm7014556 BindingDB Entry DOI: 10.7270/Q2Z037ZW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50243008 (CHEMBL469682 | N,N-Diethyl-2-(2-(4-(3-fluoropropox...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 4.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Radiopharmaceuticals Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]PK11195 from peripheral benzodiazepine receptor in rat kidney membrane | J Med Chem 51: 3700-12 (2008) Article DOI: 10.1021/jm7014556 BindingDB Entry DOI: 10.7270/Q2Z037ZW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50243006 (2-(6-Chloro-2-(4-(3-fluoropropoxy)phenyl)imidazo[1...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Radiopharmaceuticals Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]Ro 5-4864 from peripheral benzodiazepine receptor in rat kidney membrane | J Med Chem 51: 3700-12 (2008) Article DOI: 10.1021/jm7014556 BindingDB Entry DOI: 10.7270/Q2Z037ZW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50243007 (2-(2-(4-(2-Fluoroethoxy)phenyl)-5,7-dimethylpyrazo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Radiopharmaceuticals Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]PK11195 from peripheral benzodiazepine receptor in rat kidney membrane | J Med Chem 51: 3700-12 (2008) Article DOI: 10.1021/jm7014556 BindingDB Entry DOI: 10.7270/Q2Z037ZW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50243007 (2-(2-(4-(2-Fluoroethoxy)phenyl)-5,7-dimethylpyrazo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 5.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Radiopharmaceuticals Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]Ro 5-4864 from peripheral benzodiazepine receptor in rat kidney membrane | J Med Chem 51: 3700-12 (2008) Article DOI: 10.1021/jm7014556 BindingDB Entry DOI: 10.7270/Q2Z037ZW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50243008 (CHEMBL469682 | N,N-Diethyl-2-(2-(4-(3-fluoropropox...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 5.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Radiopharmaceuticals Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]Ro 5-4864 from peripheral benzodiazepine receptor in rat kidney membrane | J Med Chem 51: 3700-12 (2008) Article DOI: 10.1021/jm7014556 BindingDB Entry DOI: 10.7270/Q2Z037ZW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50243005 (2-(6-Chloro-2-(4-(2-fluoroethoxy)phenyl)imidazo[1,...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 5.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Radiopharmaceuticals Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]PK11195 from peripheral benzodiazepine receptor in rat kidney membrane | J Med Chem 51: 3700-12 (2008) Article DOI: 10.1021/jm7014556 BindingDB Entry DOI: 10.7270/Q2Z037ZW | |||||||||||
More data for this Ligand-Target Pair |