BindingDB PrimarySearch

Found 203 hits with Last Name = 'hollick' and Initial = 'jj'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM181015 (US9133199, 254) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	<10	n/a	n/a	n/a	n/a	n/a	n/a	7.5	n/a
Cyclacel Limited US Patent					Assay Description CDC25C (2 ug/well) with PLKl (1 ug/well) in 20 mM Tris/HCl buffer pH 7.5, supplemented with 25 mM beta-glycerophosphate, 5 mM EGTA, 1 mM DTT and 1 mM...				US Patent US9133199 (2015) BindingDB Entry DOI: 10.7270/Q21C1VNZ
Cyclacel Limited US Patent					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM181016 (US9133199, I-253) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	<10	n/a	n/a	n/a	n/a	n/a	n/a	7.5	n/a
Cyclacel Limited US Patent					Assay Description CDC25C (2 ug/well) with PLKl (1 ug/well) in 20 mM Tris/HCl buffer pH 7.5, supplemented with 25 mM beta-glycerophosphate, 5 mM EGTA, 1 mM DTT and 1 mM...				US Patent US9133199 (2015) BindingDB Entry DOI: 10.7270/Q21C1VNZ
Cyclacel Limited US Patent					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM12915 (2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one \|...) Show SMILES O=c1cc(oc2c(cccc12)-c1ccccc1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	PubMed	6.00E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description Affinity for DNA-dependent protein kinase(DNA-PK) from HeLa cell extract				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
Serine-protein kinase ATM (Homo sapiens (Human))	BDBM50208517 (2-morpholin-4-yl-6-thianthren-1-yl-pyran-4-one \| C...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents	PDB Article PubMed	n/a	n/a	13	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of ATM kinase				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132371 (2-Morpholin-4-yl-6-(4-naphthalen-1-yl-phenyl)-thio...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	160	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132373 (2-(4-(benzo[b]thiophen-3-yl)phenyl)-6-morpholino-4...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	160	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132355 (2-(4-Chloro-phenyl)-6-morpholin-4-yl-pyran-4-one \|...) Show SMILES Clc1ccc(cc1)-c1cc(=O)cc(o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	180	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132355 (2-(4-Chloro-phenyl)-6-morpholin-4-yl-pyran-4-one \|...) Show SMILES Clc1ccc(cc1)-c1cc(=O)cc(o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	180	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132371 (2-Morpholin-4-yl-6-(4-naphthalen-1-yl-phenyl)-thio...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	190	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132361 (2-(4-Methoxy-phenyl)-6-morpholin-4-yl-pyran-4-one ...) Show SMILES COc1ccc(cc1)-c1cc(=O)cc(o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	220	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132361 (2-(4-Methoxy-phenyl)-6-morpholin-4-yl-pyran-4-one ...) Show SMILES COc1ccc(cc1)-c1cc(=O)cc(o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	220	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50098126 (2-(morpholin-4-yl)-benzo[h]chromen-4-one \| 2-Morph...) Show SMILES O=c1cc(oc2c3ccccc3ccc12)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	230	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132368 (2-[4-(4-Methyl-naphthalen-1-yl)-phenyl]-6-morpholi...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	260	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132368 (2-[4-(4-Methyl-naphthalen-1-yl)-phenyl]-6-morpholi...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	260	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132365 (2-(4-Methoxy-phenyl)-6-morpholin-4-yl-thiopyran-4-...) Show SMILES COc1ccc(cc1)-c1cc(=O)cc(s1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	280	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132365 (2-(4-Methoxy-phenyl)-6-morpholin-4-yl-thiopyran-4-...) Show SMILES COc1ccc(cc1)-c1cc(=O)cc(s1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	280	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132363 (2-(2-Methoxy-phenyl)-6-morpholin-4-yl-pyran-4-one ...) Show SMILES COc1ccccc1-c1cc(=O)cc(o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	310	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132373 (2-(4-(benzo[b]thiophen-3-yl)phenyl)-6-morpholino-4...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	330	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132370 (2-(4-Fluoro-phenyl)-6-morpholin-4-yl-pyran-4-one \|...) Show SMILES Fc1ccc(cc1)-c1cc(=O)cc(o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	350	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132366 (2-(4'-Hydroxy-biphenyl-3-yl)-6-morpholin-4-yl-thio...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	350	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132370 (2-(4-Fluoro-phenyl)-6-morpholin-4-yl-pyran-4-one \|...) Show SMILES Fc1ccc(cc1)-c1cc(=O)cc(o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	350	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132363 (2-(2-Methoxy-phenyl)-6-morpholin-4-yl-pyran-4-one ...) Show SMILES COc1ccccc1-c1cc(=O)cc(o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	380	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50208499 (6-(2-fluorophenyl)-2-(4-morpholin-4-yl)pyran-4-one...) Show SMILES Fc1ccccc1-c1cc(=O)cc(o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	390	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50208505 (2-(1H-indol-5-yl)-6-morpholino-4H-pyran-4-one \| CH...) Show SMILES O=c1cc(oc(c1)-c1ccc2[nH]ccc2c1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	400	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50208552 (6-(4-chlorophenyl)-4-morpholino-2H-pyran-2-one \| C...) Show SMILES Clc1ccc(cc1)-c1cc(cc(=O)o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	470	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132358 (2-(4-tert-Butyl-phenyl)-6-morpholin-4-yl-pyran-4-o...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	480	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132358 (2-(4-tert-Butyl-phenyl)-6-morpholin-4-yl-pyran-4-o...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	480	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50208494 (2-(4-(6-morpholino-4-oxo-4H-pyran-2-yl)benzyl)isoi...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	500	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50208558 (6-(4-methoxyphenyl)-4-morpholino-2H-pyran-2-one \| ...) Show SMILES COc1ccc(cc1)-c1cc(cc(=O)o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	530	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132369 (2-(4-Chloro-phenyl)-6-morpholin-4-yl-thiopyran-4-o...) Show SMILES Clc1ccc(cc1)-c1cc(=O)cc(s1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	530	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132369 (2-(4-Chloro-phenyl)-6-morpholin-4-yl-thiopyran-4-o...) Show SMILES Clc1ccc(cc1)-c1cc(=O)cc(s1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	530	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132360 (2-(3-Fluoro-phenyl)-6-morpholin-4-yl-pyran-4-one \|...) Show SMILES Fc1cccc(c1)-c1cc(=O)cc(o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	530	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132356 (2-(3-Methoxy-phenyl)-6-morpholin-4-yl-pyran-4-one ...) Show SMILES COc1cccc(c1)-c1cc(=O)cc(o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	540	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132356 (2-(3-Methoxy-phenyl)-6-morpholin-4-yl-pyran-4-one ...) Show SMILES COc1cccc(c1)-c1cc(=O)cc(o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	540	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50208507 (2-(benzo[b]thiophen-2-yl)-6-morpholino-4H-pyran-4-...) Show SMILES O=c1cc(oc(c1)-c1cc2ccccc2s1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	600	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132364 (2-Morpholin-4-yl-6-phenyl-thiopyran-4-one \| 2-morp...) Show SMILES O=c1cc(sc(c1)-c1ccccc1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	650	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132367 (2-(4-Bromo-phenyl)-6-morpholin-4-yl-thiopyran-4-on...) Show SMILES Brc1ccc(cc1)-c1cc(=O)cc(s1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	680	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132367 (2-(4-Bromo-phenyl)-6-morpholin-4-yl-thiopyran-4-on...) Show SMILES Brc1ccc(cc1)-c1cc(=O)cc(s1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	680	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50208557 (CHEMBL222820 \| N-[3'-(6-morpholin-4-yl-4-oxo-4H-th...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	680	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132360 (2-(3-Fluoro-phenyl)-6-morpholin-4-yl-pyran-4-one \|...) Show SMILES Fc1cccc(c1)-c1cc(=O)cc(o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	690	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132354 (2-(3-Bromo-phenyl)-6-morpholin-4-yl-thiopyran-4-on...) Show SMILES Brc1cccc(c1)-c1cc(=O)cc(s1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	700	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132364 (2-Morpholin-4-yl-6-phenyl-thiopyran-4-one \| 2-morp...) Show SMILES O=c1cc(sc(c1)-c1ccccc1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	720	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50208500 (2-biphenyl-4-yl-6-morpholin-4-yl-pyran-4-one \| CHE...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	800	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132354 (2-(3-Bromo-phenyl)-6-morpholin-4-yl-thiopyran-4-on...) Show SMILES Brc1cccc(c1)-c1cc(=O)cc(s1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	800	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50208493 (2-(benzofuran-2-yl)-6-morpholino-4H-pyran-4-one \| ...) Show SMILES O=c1cc(oc(c1)-c1cc2ccccc2o1)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	800	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132357 ((E)-3-[3'-(6-Morpholin-4-yl-4-oxo-4H-thiopyran-2-y...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	PubMed	n/a	n/a	840	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132357 ((E)-3-[3'-(6-Morpholin-4-yl-4-oxo-4H-thiopyran-2-y...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	840	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50208495 (2-morpholino-6-(quinolin-8-yl)-4H-pyran-4-one \| CH...) Show SMILES O=c1cc(oc(c1)-c1cccc2cccnc12)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	900	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50208533 (2-(4-(benzyloxy)phenyl)-6-morpholino-4H-pyran-4-on...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	910	n/a	n/a	n/a	n/a	n/a	n/a
Newcastle University Curated by ChEMBL					Assay Description Inhibition of DNA-PK in HeLa cell nuclear extracts				J Med Chem 50: 1958-72 (2007) Article DOI: 10.1021/jm061121y BindingDB Entry DOI: 10.7270/Q2FB52MW
Newcastle University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50132362 (2-(3'-hydroxy-biphenyl-3-yl)-6-morpholin-4-yl-thio...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	920	n/a	n/a	n/a	n/a	n/a	n/a
University of Newcastle Curated by ChEMBL					Assay Description In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.				Bioorg Med Chem Lett 13: 3083-6 (2003) BindingDB Entry DOI: 10.7270/Q2WS8SP4
University of Newcastle Curated by ChEMBL					More data for this Ligand-Target Pair

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