Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melanocortin receptor 4 (Mus musculus) | BDBM50144869 (CHEMBL411775 | Tyr-c[Asp-His-DPhe-Arg-Trp-Asn-Ala-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.260 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132) | J Med Chem 47: 2194-207 (2004) Article DOI: 10.1021/jm0303608 BindingDB Entry DOI: 10.7270/Q2474BM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50144869 (CHEMBL411775 | Tyr-c[Asp-His-DPhe-Arg-Trp-Asn-Ala-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.960 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSH | J Med Chem 47: 2194-207 (2004) Article DOI: 10.1021/jm0303608 BindingDB Entry DOI: 10.7270/Q2474BM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50144877 (CHEMBL269274) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.46 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSH | J Med Chem 47: 2194-207 (2004) Article DOI: 10.1021/jm0303608 BindingDB Entry DOI: 10.7270/Q2474BM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273103 (3-[(3-methylbenzene)sulfonyl]-1-({4-[({[(3-methylb...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273103 (3-[(3-methylbenzene)sulfonyl]-1-({4-[({[(3-methylb...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50272993 (1-[(3-chlorobenzene)sulfonyl]-3-[7-({[(3-chloroben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273102 (3-[(3-chlorobenzene)sulfonyl]-1-({4-[({[(3-chlorob...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50121900 (Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.22 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-NDP-MSH; ND = not determined | J Med Chem 47: 2194-207 (2004) Article DOI: 10.1021/jm0303608 BindingDB Entry DOI: 10.7270/Q2474BM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50144877 (CHEMBL269274) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.45 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132) | J Med Chem 47: 2194-207 (2004) Article DOI: 10.1021/jm0303608 BindingDB Entry DOI: 10.7270/Q2474BM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50144871 (CHEMBL428134) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.74 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132) | J Med Chem 47: 2194-207 (2004) Article DOI: 10.1021/jm0303608 BindingDB Entry DOI: 10.7270/Q2474BM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50272994 (1-[(3-methylbenzene)sulfonyl]-3-[7-({[(3-methylben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50144882 (CHEMBL266288) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.48 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132) | J Med Chem 47: 2194-207 (2004) Article DOI: 10.1021/jm0303608 BindingDB Entry DOI: 10.7270/Q2474BM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273104 (3-[(3-methylbenzene)sulfonyl]-1-({3-[({[(3-methylb...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273102 (3-[(3-chlorobenzene)sulfonyl]-1-({4-[({[(3-chlorob...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50272991 (1-[(3-chlorobenzene)sulfonyl]-3-[6-({[(3-chloroben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273035 (3-[(3-methylbenzene)sulfonyl]-1-[8-({[(3-methylben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50272993 (1-[(3-chlorobenzene)sulfonyl]-3-[7-({[(3-chloroben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273193 (1-[(3-chlorobenzene)sulfonyl]-3-(2-{[2-({[(3-chlor...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50272994 (1-[(3-methylbenzene)sulfonyl]-3-[7-({[(3-methylben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273104 (3-[(3-methylbenzene)sulfonyl]-1-({3-[({[(3-methylb...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273070 (3-[(3-methylbenzene)sulfonyl]-1-[6-({[(3-methylben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273194 (1-[(3-methylbenzene)sulfonyl]-3-(2-{[2-({[(3-methy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50272992 (1-[(3-methylbenzene)sulfonyl]-3-[6-({[(3-methylben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273036 (1-[(3-chlorobenzene)sulfonyl]-3-[(3E)-6-({[(3-chlo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273071 (3-[(3-chlorobenzene)sulfonyl]-1-({4-[({[(3-chlorob...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50272991 (1-[(3-chlorobenzene)sulfonyl]-3-[6-({[(3-chloroben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273034 (3-[(3-chlorobenzene)sulfonyl]-1-[8-({[(3-chloroben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273139 (1-[(3-methylbenzene)sulfonyl]-3-(2-{[2-({[(3-methy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50272913 (1-[(3-chlorobenzene)sulfonyl]-3-[5-({[(3-chloroben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50272914 (1-[(3-methylbenzene)sulfonyl]-3-[5-({[(3-methylben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50272992 (1-[(3-methylbenzene)sulfonyl]-3-[6-({[(3-methylben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273071 (3-[(3-chlorobenzene)sulfonyl]-1-({4-[({[(3-chlorob...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273037 (1-[(3-methylbenzene)sulfonyl]-3-[(3E)-6-({[(3-meth...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273194 (1-[(3-methylbenzene)sulfonyl]-3-(2-{[2-({[(3-methy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 29 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50144871 (CHEMBL428134) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 29.8 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Florida Curated by ChEMBL | Assay Description Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSH | J Med Chem 47: 2194-207 (2004) Article DOI: 10.1021/jm0303608 BindingDB Entry DOI: 10.7270/Q2474BM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50305572 (CHEMBL590111 | N-(5-bromothiazol-2-ylcarbamoyl)-5-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of FBPase in human liver using fructose-2,6phosphate as a substrate | Bioorg Med Chem Lett 20: 594-9 (2010) Article DOI: 10.1016/j.bmcl.2009.11.093 BindingDB Entry DOI: 10.7270/Q27H1JPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50305562 (CHEMBL590359 | N-(5-bromothiazol-2-ylcarbamoyl)-5-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of FBPase in human liver using fructose-2,6phosphate as a substrate | Bioorg Med Chem Lett 20: 594-9 (2010) Article DOI: 10.1016/j.bmcl.2009.11.093 BindingDB Entry DOI: 10.7270/Q27H1JPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273035 (3-[(3-methylbenzene)sulfonyl]-1-[8-({[(3-methylben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50305595 (CHEMBL591317 | N-(7-chloro-4-methoxybenzo[d]thiazo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of FBPase in human liver | Bioorg Med Chem Lett 20: 594-9 (2010) Article DOI: 10.1016/j.bmcl.2009.11.093 BindingDB Entry DOI: 10.7270/Q27H1JPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273036 (1-[(3-chlorobenzene)sulfonyl]-3-[(3E)-6-({[(3-chlo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50305569 (CHEMBL590597 | N-(5-bromothiazol-2-ylcarbamoyl)-5-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of FBPase in human liver using fructose-2,6phosphate as a substrate | Bioorg Med Chem Lett 20: 594-9 (2010) Article DOI: 10.1016/j.bmcl.2009.11.093 BindingDB Entry DOI: 10.7270/Q27H1JPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50305562 (CHEMBL590359 | N-(5-bromothiazol-2-ylcarbamoyl)-5-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of FBPase in human liver | Bioorg Med Chem Lett 20: 594-9 (2010) Article DOI: 10.1016/j.bmcl.2009.11.093 BindingDB Entry DOI: 10.7270/Q27H1JPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50305567 (CHEMBL589863 | N-(5-bromothiazol-2-ylcarbamoyl)-5-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of FBPase in human liver using fructose-2,6phosphate as a substrate | Bioorg Med Chem Lett 20: 594-9 (2010) Article DOI: 10.1016/j.bmcl.2009.11.093 BindingDB Entry DOI: 10.7270/Q27H1JPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273034 (3-[(3-chlorobenzene)sulfonyl]-1-[8-({[(3-chloroben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 45 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50305573 (CHEMBL590839 | N-(5-bromothiazol-2-ylcarbamoyl)-5-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of FBPase in human liver using fructose-2,6phosphate as a substrate | Bioorg Med Chem Lett 20: 594-9 (2010) Article DOI: 10.1016/j.bmcl.2009.11.093 BindingDB Entry DOI: 10.7270/Q27H1JPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50272913 (1-[(3-chlorobenzene)sulfonyl]-3-[5-({[(3-chloroben...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50305571 (CHEMBL601691 | N-(5-bromothiazol-2-ylcarbamoyl)-5-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of FBPase in human liver using fructose-2,6phosphate as a substrate | Bioorg Med Chem Lett 20: 594-9 (2010) Article DOI: 10.1016/j.bmcl.2009.11.093 BindingDB Entry DOI: 10.7270/Q27H1JPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273193 (1-[(3-chlorobenzene)sulfonyl]-3-(2-{[2-({[(3-chlor...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 55 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50273235 (1-[(3-chlorobenzene)sulfonyl]-3-{3-[3-({[(3-chloro...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 57 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphate | Bioorg Med Chem Lett 18: 4708-12 (2008) Article DOI: 10.1016/j.bmcl.2008.06.103 BindingDB Entry DOI: 10.7270/Q26W99W7 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Fructose-1,6-bisphosphatase 1 (Homo sapiens (Human)) | BDBM50305565 (CHEMBL590361 | N-(5-bromothiazol-2-ylcarbamoyl)-5-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd Curated by ChEMBL | Assay Description Inhibition of FBPase in human liver using fructose-2,6phosphate as a substrate | Bioorg Med Chem Lett 20: 594-9 (2010) Article DOI: 10.1016/j.bmcl.2009.11.093 BindingDB Entry DOI: 10.7270/Q27H1JPX | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |
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