Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207195 ((S)-N-((S)-5-acetamido-5-(1H-benzo[d]imidazol-2-yl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.210 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207188 ((S)-N-((S)-5-acetamido-6-(benzylamino)-6-oxohexyl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.210 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207196 ((S)-N-((S)-5-acetamido-6-oxo-6-(phenylamino)hexyl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.220 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM50181392 ((R)-N-(3-(3H-spiro[isobenzofuran-1,4'-piperidine]-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | 0.240 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cells | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207190 (CHEMBL396423 | benzyl (S)-6-((S)-2-((S)-2-amino-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.470 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207194 (CHEMBL232812 | benzyl (S)-6-((S)-2-((S)-2-amino-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.530 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50000788 ((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | DrugBank Article PubMed | 0.562 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]DPN from human recombinant mu-type opioid receptor expressed in CHO cell membranes | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207192 ((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO 2 from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM50418594 (CHEMBL1783826) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | 0.724 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cells | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207189 (CHEMBL438681 | benzyl (S)-5-((S)-2-((S)-2-amino-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.860 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207193 ((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.890 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO 2 from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207195 ((S)-N-((S)-5-acetamido-5-(1H-benzo[d]imidazol-2-yl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.990 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO 2 from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207192 ((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207191 ((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.02 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO 2 from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207193 ((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.02 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207196 ((S)-N-((S)-5-acetamido-6-oxo-6-(phenylamino)hexyl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.57 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO 2 from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207191 ((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.64 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207190 (CHEMBL396423 | benzyl (S)-6-((S)-2-((S)-2-amino-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.67 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO 2 from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207189 (CHEMBL438681 | benzyl (S)-5-((S)-2-((S)-2-amino-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.78 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO 2 from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207194 (CHEMBL232812 | benzyl (S)-6-((S)-2-((S)-2-amino-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO 2 from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50207188 ((S)-N-((S)-5-acetamido-6-(benzylamino)-6-oxohexyl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.43 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO 2 from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50000788 ((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | DrugBank Article PubMed | 4.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]DPN from human recombinant kappa-type opioid receptor expressed in CHO cell membranes | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50000788 ((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | DrugBank Article PubMed | 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]DPN from human recombinant delta-type opioid receptor expressed in CHO cell membranes | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prokineticin receptor 1 (Homo sapiens (Human)) | BDBM26335 (3-[2-({5-[(4-ethylphenyl)methyl]-1-[(4-methoxyphen...) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 22 | -45.5 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
University of Ferrara | Assay Description Nonspecific binding was determined in the presence of 1 uM Bv8. Displacement curves were determined in triplicate. The inhibition constant (Ki) of th... | J Med Chem 51: 7635-9 (2008) Article DOI: 10.1021/jm800854e BindingDB Entry DOI: 10.7270/Q23J3B9C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM50418589 (CHEMBL1783821) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 49 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cells | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM50418587 (CHEMBL1783817) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 59 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cells | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM50418598 (CHEMBL1783818) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 59 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cells | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM50418588 (CHEMBL1783819) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cells | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM50418595 (CHEMBL1783827) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 83 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cells | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM50418590 (CHEMBL1783822) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 107 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cells | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM50418591 (CHEMBL1783823) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 158 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cells | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50418594 (CHEMBL1783826) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | 191 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]DPN from human recombinant mu-type opioid receptor expressed in CHO cell membranes | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50418594 (CHEMBL1783826) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | 316 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]DPN from human recombinant kappa-type opioid receptor expressed in CHO cell membranes | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prokineticin receptor 1 (Homo sapiens (Human)) | BDBM26336 (6-[(2-aminoethyl)amino]-3-[(4-ethylphenyl)methyl]-...) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 440 | -37.7 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
University of Ferrara | Assay Description Nonspecific binding was determined in the presence of 1 uM Bv8. Displacement curves were determined in triplicate. The inhibition constant (Ki) of th... | J Med Chem 51: 7635-9 (2008) Article DOI: 10.1021/jm800854e BindingDB Entry DOI: 10.7270/Q23J3B9C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50418594 (CHEMBL1783826) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]DPN from human recombinant delta-type opioid receptor expressed in CHO cell membranes | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM50418597 (CHEMBL1783820) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.15E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cells | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prokineticin receptor 2 (Homo sapiens (Human)) | BDBM26335 (3-[2-({5-[(4-ethylphenyl)methyl]-1-[(4-methoxyphen...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 1.61E+3 | -34.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
University of Ferrara | Assay Description Nonspecific binding was determined in the presence of 1 uM Bv8. Displacement curves were determined in triplicate. The inhibition constant (Ki) of th... | J Med Chem 51: 7635-9 (2008) Article DOI: 10.1021/jm800854e BindingDB Entry DOI: 10.7270/Q23J3B9C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prokineticin receptor 1 (Homo sapiens (Human)) | BDBM26337 (6-{[2-(4,5-dihydro-1H-imidazol-2-ylamino)ethyl]ami...) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 4.72E+3 | -31.6 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
University of Ferrara | Assay Description Nonspecific binding was determined in the presence of 1 uM Bv8. Displacement curves were determined in triplicate. The inhibition constant (Ki) of th... | J Med Chem 51: 7635-9 (2008) Article DOI: 10.1021/jm800854e BindingDB Entry DOI: 10.7270/Q23J3B9C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM50418592 (CHEMBL1783824) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cells | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM50418596 (CHEMBL1783828) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cells | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM50418593 (CHEMBL1783825) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]N/OFQ from human recombinant NOP receptor expressed in CHO cells | Bioorg Med Chem 17: 5080-95 (2009) Article DOI: 10.1016/j.bmc.2009.05.068 BindingDB Entry DOI: 10.7270/Q2P270C3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prokineticin receptor 2 (Homo sapiens (Human)) | BDBM26336 (6-[(2-aminoethyl)amino]-3-[(4-ethylphenyl)methyl]-...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 2.34E+4 | -27.5 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
University of Ferrara | Assay Description Nonspecific binding was determined in the presence of 1 uM Bv8. Displacement curves were determined in triplicate. The inhibition constant (Ki) of th... | J Med Chem 51: 7635-9 (2008) Article DOI: 10.1021/jm800854e BindingDB Entry DOI: 10.7270/Q23J3B9C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prokineticin receptor 2 (Homo sapiens (Human)) | BDBM26337 (6-{[2-(4,5-dihydro-1H-imidazol-2-ylamino)ethyl]ami...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 7.12E+4 | -24.6 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
University of Ferrara | Assay Description Nonspecific binding was determined in the presence of 1 uM Bv8. Displacement curves were determined in triplicate. The inhibition constant (Ki) of th... | J Med Chem 51: 7635-9 (2008) Article DOI: 10.1021/jm800854e BindingDB Entry DOI: 10.7270/Q23J3B9C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50207191 ((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 434 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated contraction | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50207196 ((S)-N-((S)-5-acetamido-6-oxo-6-(phenylamino)hexyl)...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 486 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated contraction | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50207193 ((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 515 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated contraction | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50207192 ((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 553 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated contraction | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50207195 ((S)-N-((S)-5-acetamido-5-(1H-benzo[d]imidazol-2-yl...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 610 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated contraction | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50207189 (CHEMBL438681 | benzyl (S)-5-((S)-2-((S)-2-amino-3-...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 618 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated contraction | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50207190 (CHEMBL396423 | benzyl (S)-6-((S)-2-((S)-2-amino-3-...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 711 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated contraction | Bioorg Med Chem 15: 3143-51 (2007) Article DOI: 10.1016/j.bmc.2007.02.039 BindingDB Entry DOI: 10.7270/Q2ST7PHP | |||||||||||
More data for this Ligand-Target Pair |
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