Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sphingosine 1-phosphate receptor 5 (Homo sapiens (Human)) | BDBM50250631 (CHEMBL4093489) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | 0.574 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ono Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Displacement of [33P]-S1P from human S1P5 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting method | J Med Chem 60: 9508-9530 (2017) Article DOI: 10.1021/acs.jmedchem.7b00785 BindingDB Entry DOI: 10.7270/Q2J968SK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sphingosine 1-phosphate receptor 1 (Homo sapiens (Human)) | BDBM50250631 (CHEMBL4093489) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | 0.626 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ono Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Displacement of [33P]-S1P from human S1P1 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting method | J Med Chem 60: 9508-9530 (2017) Article DOI: 10.1021/acs.jmedchem.7b00785 BindingDB Entry DOI: 10.7270/Q2J968SK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sphingosine 1-phosphate receptor 1 (Rattus norvegicus) | BDBM50250631 (CHEMBL4093489) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | 0.772 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ono Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Displacement of [33P]-S1P from rat S1P1 receptor after 60 mins by scintillation counting method | J Med Chem 60: 9508-9530 (2017) Article DOI: 10.1021/acs.jmedchem.7b00785 BindingDB Entry DOI: 10.7270/Q2J968SK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sphingosine 1-phosphate receptor 4 (Homo sapiens (Human)) | BDBM50250631 (CHEMBL4093489) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | 29 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ono Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Displacement of [33P]-S1P from human S1P4 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting method | J Med Chem 60: 9508-9530 (2017) Article DOI: 10.1021/acs.jmedchem.7b00785 BindingDB Entry DOI: 10.7270/Q2J968SK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sphingosine 1-phosphate receptor 2 (Homo sapiens (Human)) | BDBM50250631 (CHEMBL4093489) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | >5.45E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ono Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Displacement of [33P]-S1P from human S1P2 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting method | J Med Chem 60: 9508-9530 (2017) Article DOI: 10.1021/acs.jmedchem.7b00785 BindingDB Entry DOI: 10.7270/Q2J968SK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sphingosine 1-phosphate receptor 3 (Homo sapiens (Human)) | BDBM50250631 (CHEMBL4093489) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | >5.63E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ono Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Displacement of [33P]-S1P from human S1P3 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting method | J Med Chem 60: 9508-9530 (2017) Article DOI: 10.1021/acs.jmedchem.7b00785 BindingDB Entry DOI: 10.7270/Q2J968SK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285779 (CHEMBL4165205) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.160 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cell membranes pretreated for 24 hrs prior to Fura-2-AM dye addition for 1 hr followed... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285779 (CHEMBL4165205) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.190 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cell membranes pretreated for 24 hrs prior to Fura-2-AM dye addition for 1 hr followed... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195700 (CHEMBL3975893) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.5 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195694 (CHEMBL3976876) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.90 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285789 (CHEMBL4169559) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195690 (CHEMBL3917128) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285788 (CHEMBL4162680) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285787 (CHEMBL4170604) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285780 (CHEMBL4164105) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 29 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285781 (CHEMBL4165714) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285790 (CHEMBL4169137) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285936 (CHEMBL4172946) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285935 (CHEMBL4171981) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 38 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285783 (CHEMBL4162273) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195693 (CHEMBL3947597) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 42 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285786 (CHEMBL4175424) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 45 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285784 (CHEMBL4167552) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 61 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285922 (CHEMBL4159560) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 61 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195778 (CHEMBL3971582) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 71 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285779 (CHEMBL4165205) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 86 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50373831 (CHEMBL272087) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 89 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195546 (CHEMBL3956307) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195691 (CHEMBL3986868) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285782 (CHEMBL4177410) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195776 (CHEMBL3932828) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195779 (CHEMBL3984953) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195701 (CHEMBL3956293) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195695 (CHEMBL3941037) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195695 (CHEMBL3941037) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285937 (CHEMBL4176330) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195773 (CHEMBL3901754) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195689 (CHEMBL3959223) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195552 (CHEMBL3944344) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 220 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195772 (CHEMBL3896148) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195620 (CHEMBL3930834) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195558 (CHEMBL3890162) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195771 (CHEMBL3950523) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 390 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285785 (CHEMBL4167471) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 460 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50285830 (CHEMBL4161219) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 520 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195563 (CHEMBL3913038) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 680 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 2 (Homo sapiens (Human)) | BDBM50195700 (CHEMBL3975893) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 790 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Inhibition of LPA2 (unknown origin) | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195571 (CHEMBL3973793) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195692 (CHEMBL3905099) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 receptor expressed in CHO cells assessed as reduction in LPA-induced intracellular Ca2+ concentration pretreated wi... | ACS Med Chem Lett 7: 913-918 (2016) Article DOI: 10.1021/acsmedchemlett.6b00225 BindingDB Entry DOI: 10.7270/Q2X350FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50195571 (CHEMBL3973793) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
ONO Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll... | ACS Med Chem Lett 8: 1281-1286 (2017) Article DOI: 10.1021/acsmedchemlett.7b00383 BindingDB Entry DOI: 10.7270/Q2PG1V8Z | |||||||||||
More data for this Ligand-Target Pair |
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