Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet-activating factor receptor (Mus musculus) | BDBM50118202 (6-(4-azido-2,3,5,6-tetrafluorobenzyloxy)-8-(tert-b...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123637 (6-benzyloxy-8-(tert-butyl)-9-flouro-12,17-dihydrox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123639 (8-(tert-butyl)-9-chloro-6,12,17-trihydroxy-16-meth...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123644 (6-benzyloxy-8-(tert-butyl)-12,17-dihydroxy-16-meth...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 120 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118204 (6-(4-benzoylphenylcarbonyloxy)-8-(tert-butyl)-12,1...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118194 (8-(tert-butyl)-12,17-dihydroxy-16-methyl-6-[4-(3-t...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 150 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118201 (6-(4-benzoylbenzyloxy)-8-(tert-butyl)-12,17-dihydr...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 150 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118203 (8-(tert-butyl)-9,12,17-trihydroxy-16-methyl-6-[4-(...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 470 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123638 (9-azido-8-(tert-butyl)-6,12,17-trihydroxy-16-methy...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 550 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118195 (3'-(tert-butyl)-4,9',14'-trihydroxy-2-methoxy-10'-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 560 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118196 (6-(4-benzoylbenzyloxy)-8-(tert-butyl)-9,12,17-trih...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 580 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123643 (6-benzyloxy-8-(tert-butyl)-9,12,17-trihydroxy-16-m...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123633 (8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-9-meth...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 610 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118200 (6-(4-azido-2,3,5,6-tetrafluorobenzyloxy)-8-(tert-b...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 790 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50251276 (BN 52021 | CHEMBL514432 | GINKOLIDE B | Gingkolide...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | 880 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123642 (8-(tert-butyl)-9-flouro-6,12,17-trihydroxy-16-meth...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 990 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118205 (3'-(tert-butyl)-4,9'-dihydroxy-2-methoxy-10'-methy...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.46E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123631 (8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-9-ethy...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.62E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123632 (6-benzyloxy-8-(tert-butyl)-9,12,17-trihydroxy-16-m...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.67E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123645 (CHEMBL348623 | benzyl (6R,9R,12R,16S,17R)-8-tert-b...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123635 (8-(tert-butyl)-6,9,12,17-tetrahydroxy-16-methyl-(6...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.26E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123636 (8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-5,15,1...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.84E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123640 (8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-9-amin...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.64E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118193 (3'-(tert-butyl)-4,4',9'-trihydroxy-2-methoxy-10'-m...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 9.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118197 (3'-(tert-butyl)-4,4',9',14'-tetrahydroxy-2-methoxy...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.26E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50123641 (8-(tert-butyl)-6,9,12,17-tetrahydroxy-16-methyl-(6...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.26E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membrane | J Med Chem 46: 601-8 (2003) Article DOI: 10.1021/jm0203985 BindingDB Entry DOI: 10.7270/Q2CC1023 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118199 (9-tert-Butyl-8,9-dihydroxy-dihydro-furo[2,3-b]furo...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Mus musculus) | BDBM50118198 (3'-(tert-butyl)-4,4',14'-trihydroxy-2-methoxy-10'-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF) | J Med Chem 45: 4038-46 (2002) BindingDB Entry DOI: 10.7270/Q29G5M5T | |||||||||||
More data for this Ligand-Target Pair |