Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sterol O-acyltransferase 2 (Chlorocebus aethiops) | BDBM50204552 (CHEMBL3959948) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT2 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Chlorocebus aethiops) | BDBM50204547 (CHEMBL3923673) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT2 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Chlorocebus aethiops) | BDBM50204550 (CHEMBL3916935) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT2 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Chlorocebus aethiops) | BDBM50204547 (CHEMBL3923673) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT1 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Chlorocebus aethiops) | BDBM50204553 (CHEMBL3971022) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 9.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT2 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Chlorocebus aethiops) | BDBM50204545 (CHEMBL3898917) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 9.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT2 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Chlorocebus aethiops) | BDBM50204553 (CHEMBL3971022) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT1 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Chlorocebus aethiops) | BDBM50204558 (CHEMBL3960874) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT2 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Chlorocebus aethiops) | BDBM50204551 (CHEMBL3958875) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT1 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Chlorocebus aethiops) | BDBM50204552 (CHEMBL3959948) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT1 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Chlorocebus aethiops) | BDBM50204551 (CHEMBL3958875) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT2 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Chlorocebus aethiops) | BDBM50204548 (CHEMBL3932453) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT1 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Chlorocebus aethiops) | BDBM50204558 (CHEMBL3960874) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT1 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Chlorocebus aethiops) | BDBM50204555 (CHEMBL3983935) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT2 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Chlorocebus aethiops) | BDBM50204556 (CHEMBL3941429) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT1 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Chlorocebus aethiops) | BDBM50204556 (CHEMBL3941429) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT2 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Chlorocebus aethiops) | BDBM50204545 (CHEMBL3898917) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT1 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Chlorocebus aethiops) | BDBM50204550 (CHEMBL3916935) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT1 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Chlorocebus aethiops) | BDBM50204555 (CHEMBL3983935) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >3.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT1 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 2 (Chlorocebus aethiops) | BDBM50204548 (CHEMBL3932453) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of African green monkey SOAT2 expressed in CHO cells assessed as reduction in [14C]cholesteryl ester formation from [1-14C]oleic acid meas... | Bioorg Med Chem Lett 26: 5899-5901 (2016) Article DOI: 10.1016/j.bmcl.2016.11.008 BindingDB Entry DOI: 10.7270/Q2D220KD | |||||||||||
More data for this Ligand-Target Pair |