Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229577 (CHEMBL63818) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | PubMed | 0.0450 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Hebrew University Curated by ChEMBL | Assay Description Compound was evaluated for the competitive inhibition of [3H]3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[... | J Med Chem 35: 2065-9 (1992) BindingDB Entry DOI: 10.7270/Q2Z60R9H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50000727 ((R)-3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl-6,6-di...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 0.181 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Hebrew University Curated by ChEMBL | Assay Description Compound was evaluated for the competitive inhibition of [3H]3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[... | J Med Chem 35: 2065-9 (1992) BindingDB Entry DOI: 10.7270/Q2Z60R9H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229579 (CHEMBL65475) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | PubMed | 0.190 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Hebrew University Curated by ChEMBL | Assay Description Compound was evaluated for the competitive inhibition of [3H]3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[... | J Med Chem 35: 2065-9 (1992) BindingDB Entry DOI: 10.7270/Q2Z60R9H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM50214798 (CHEMBL330379) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | 0.460 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Assay Description The affinity of compound for the cannabinoid brain receptor was determined by measuring its ability to displace [3H]CP-55940 from its binding site in... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ63Q7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM50214795 (CHEMBL317086) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Assay Description The affinity of compound for the cannabinoid brain receptor was determined by measuring its ability to displace [3H]CP-55940 from its binding site in... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ63Q7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM50067499 ((6aR,10aR)-3(1,1-dimethylheptyl)-9-hydroxymethyl)-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | 0.730 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Assay Description The affinity of compound for the cannabinoid brain receptor was determined by measuring its ability to displace [3H]CP-55940 from its binding site in... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ63Q7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM50067735 ((6aR,10aR)-3-(1,1-Dimethyl-heptyl)-6,6,9-trimethyl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | 0.770 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Assay Description The affinity of compound for the cannabinoid brain receptor was determined by measuring its ability to displace [3H]CP-55940 from its binding site in... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ63Q7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM50214797 (CHEMBL328588) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | 0.810 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Assay Description The affinity of compound for the cannabinoid brain receptor was determined by measuring its ability to displace [3H]CP-55940 from its binding site in... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ63Q7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM50214796 (CHEMBL328108) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | 0.840 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Assay Description The affinity of compound for the cannabinoid brain receptor was determined by measuring its ability to displace [3H]CP-55940 from its binding site in... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ63Q7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM50072775 (2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PDB Article | 0.924 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940 | Citation and Details Article DOI: 10.1016/S0960-894X(01)80155-4 BindingDB Entry DOI: 10.7270/Q24M978Z | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50471438 (CHEMBL122884) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Binding affinity towards cannabinoid receptor using [3H]CP-55940 as radioligand in rat brain membrane | J Med Chem 40: 3626-34 (1997) Article DOI: 10.1021/jm9702950 BindingDB Entry DOI: 10.7270/Q261131W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50471436 (CHEMBL123120) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Binding affinity towards cannabinoid receptor using [3H]CP-55940 as radioligand in rat brain membrane | J Med Chem 40: 3626-34 (1997) Article DOI: 10.1021/jm9702950 BindingDB Entry DOI: 10.7270/Q261131W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50060605 ((5Z,8Z,11Z,14Z)-16,16-Dimethyl-docosa-5,8,11,14-te...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Binding affinity towards cannabinoid receptor using [3H]CP-55940 as radioligand in rat brain membrane | J Med Chem 40: 3626-34 (1997) Article DOI: 10.1021/jm9702950 BindingDB Entry DOI: 10.7270/Q261131W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM239073 (US9416103, CP-55,940) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | PubMed | 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Hebrew University Curated by ChEMBL | Assay Description Compound was evaluated for the competitive inhibition of [3H]3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[... | J Med Chem 35: 2065-9 (1992) BindingDB Entry DOI: 10.7270/Q2Z60R9H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50056468 ((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid pr...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Binding affinity towards cannabinoid receptor using [3H]CP-55940 as radioligand in rat brain membrane | J Med Chem 40: 3626-34 (1997) Article DOI: 10.1021/jm9702950 BindingDB Entry DOI: 10.7270/Q261131W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50353747 (CHEMBL561013 | JWH-018) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Biological Research Centre of the Hungarian Academy of Sciences Curated by ChEMBL | Assay Description Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysis | Eur J Med Chem 178: 571-588 (2019) Article DOI: 10.1016/j.ejmech.2019.05.037 BindingDB Entry DOI: 10.7270/Q2Z60SD8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50353747 (CHEMBL561013 | JWH-018) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Biological Research Centre of the Hungarian Academy of Sciences Curated by ChEMBL | Assay Description Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysis | Eur J Med Chem 178: 571-588 (2019) Article DOI: 10.1016/j.ejmech.2019.05.037 BindingDB Entry DOI: 10.7270/Q2Z60SD8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50471437 (CHEMBL121384) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 3.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Binding affinity towards cannabinoid receptor using [3H]CP-55940 as radioligand in rat brain membrane | J Med Chem 40: 3626-34 (1997) Article DOI: 10.1021/jm9702950 BindingDB Entry DOI: 10.7270/Q261131W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50471435 (CHEMBL120428) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Binding affinity towards cannabinoid receptor using [3H]CP-55940 as radioligand in rat brain membrane | J Med Chem 40: 3626-34 (1997) Article DOI: 10.1021/jm9702950 BindingDB Entry DOI: 10.7270/Q261131W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM21281 ((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 7.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Biological Research Centre of the Hungarian Academy of Sciences Curated by ChEMBL | Assay Description Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysis | Eur J Med Chem 178: 571-588 (2019) Article DOI: 10.1016/j.ejmech.2019.05.037 BindingDB Entry DOI: 10.7270/Q2Z60SD8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50515047 (CHEMBL4526969) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 9.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Biological Research Centre of the Hungarian Academy of Sciences Curated by ChEMBL | Assay Description Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysis | Eur J Med Chem 178: 571-588 (2019) Article DOI: 10.1016/j.ejmech.2019.05.037 BindingDB Entry DOI: 10.7270/Q2Z60SD8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM50284000 ((2-Methyl-1-pentyl-1H-indol-3-yl)-naphthalen-1-yl-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article | 9.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940 | Citation and Details Article DOI: 10.1016/S0960-894X(01)80155-4 BindingDB Entry DOI: 10.7270/Q24M978Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50515051 (CHEMBL4439431) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Biological Research Centre of the Hungarian Academy of Sciences Curated by ChEMBL | Assay Description Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysis | Eur J Med Chem 178: 571-588 (2019) Article DOI: 10.1016/j.ejmech.2019.05.037 BindingDB Entry DOI: 10.7270/Q2Z60SD8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50054472 ((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid ((...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Connecticut Curated by ChEMBL | Assay Description Binding affinity for the cannabinoid receptor in the presence of phenylmethanesulfonyl fluoride (PMSF) was determined in rat fore brain membranes | J Med Chem 37: 1889-93 (1994) Article DOI: 10.1021/jm00038a020 BindingDB Entry DOI: 10.7270/Q2JQ13QV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50054472 ((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid ((...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 22 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Binding affinity towards cannabinoid receptor using [3H]CP-55940 as radioligand in rat brain membrane | J Med Chem 40: 3626-34 (1997) Article DOI: 10.1021/jm9702950 BindingDB Entry DOI: 10.7270/Q261131W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM50469722 (CHEMBL348654) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article | 22 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940 | Citation and Details Article DOI: 10.1016/S0960-894X(01)80155-4 BindingDB Entry DOI: 10.7270/Q24M978Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM21281 ((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PDB Article | 24 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940 | Citation and Details Article DOI: 10.1016/S0960-894X(01)80155-4 BindingDB Entry DOI: 10.7270/Q24M978Z | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM22988 ((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Binding affinity towards cannabinoid receptor using [3H]CP-55940 as radioligand in rat brain membrane | J Med Chem 40: 3626-34 (1997) Article DOI: 10.1021/jm9702950 BindingDB Entry DOI: 10.7270/Q261131W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50060622 ((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid ((...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Connecticut Curated by ChEMBL | Assay Description Binding affinity for the cannabinoid receptor in the presence of phenylmethanesulfonyl fluoride (PMSF) was determined in rat fore brain membranes | J Med Chem 37: 1889-93 (1994) Article DOI: 10.1021/jm00038a020 BindingDB Entry DOI: 10.7270/Q2JQ13QV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50160434 ((6-iodo-2-methyl-1-(2-morpholinoethyl)-1H-indol-3-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 27 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Biological Research Centre of the Hungarian Academy of Sciences Curated by ChEMBL | Assay Description Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysis | Eur J Med Chem 178: 571-588 (2019) Article DOI: 10.1016/j.ejmech.2019.05.037 BindingDB Entry DOI: 10.7270/Q2Z60SD8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50054472 ((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid ((...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 28 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Connecticut Curated by ChEMBL | Assay Description Binding affinity for the cannabinoid receptor in the absence of phenylmethanesulfonyl fluoride (PMSF) was determined in rat fore brain membranes | J Med Chem 37: 1889-93 (1994) Article DOI: 10.1021/jm00038a020 BindingDB Entry DOI: 10.7270/Q2JQ13QV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50471438 (CHEMBL122884) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 31 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Binding affinity towards cannabinoid receptor using [3H]SR-141,716A as radioligand in rat brain membrane | J Med Chem 40: 3626-34 (1997) Article DOI: 10.1021/jm9702950 BindingDB Entry DOI: 10.7270/Q261131W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM50469724 (CHEMBL152187) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article | 33 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940 | Citation and Details Article DOI: 10.1016/S0960-894X(01)80155-4 BindingDB Entry DOI: 10.7270/Q24M978Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50515051 (CHEMBL4439431) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 34 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Biological Research Centre of the Hungarian Academy of Sciences Curated by ChEMBL | Assay Description Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysis | Eur J Med Chem 178: 571-588 (2019) Article DOI: 10.1016/j.ejmech.2019.05.037 BindingDB Entry DOI: 10.7270/Q2Z60SD8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (MOUSE-Mus musculus (Mouse)) | BDBM85675 (Anandamide + PMSF | CHEMBL321585) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 34 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Hebrew University Curated by ChEMBL | Assay Description Ability to displace [3H]HU-243 binding to cannabinoid receptor in synaptosomal membrane | J Med Chem 36: 3032-4 (1993) Article DOI: 10.1021/jm00072a026 BindingDB Entry DOI: 10.7270/Q2D220V0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM60994 ((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL DrugBank KEGG PC cid PC sid PDB UniChem Similars | Article | 41 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940 | Citation and Details Article DOI: 10.1016/S0960-894X(01)80155-4 BindingDB Entry DOI: 10.7270/Q24M978Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM21278 (5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 43 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Biological Research Centre of the Hungarian Academy of Sciences Curated by ChEMBL | Assay Description Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysis | Eur J Med Chem 178: 571-588 (2019) Article DOI: 10.1016/j.ejmech.2019.05.037 BindingDB Entry DOI: 10.7270/Q2Z60SD8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50056461 ((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid (2...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 44 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Binding affinity towards cannabinoid receptor using [3H]CP-55940 as radioligand in rat brain membrane | J Med Chem 40: 3626-34 (1997) Article DOI: 10.1021/jm9702950 BindingDB Entry DOI: 10.7270/Q261131W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM50067734 ((-)-(6aR-trans)-6,6,9-trimethyl-3-pentyl-6a,7,10,1...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid UniChem Patents Similars | 44 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Assay Description The affinity of compound for the cannabinoid brain receptor was determined by measuring its ability to displace [3H]CP-55940 from its binding site in... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ63Q7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM50469721 (CHEMBL348715) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article | 46 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940 | Citation and Details Article DOI: 10.1016/S0960-894X(01)80155-4 BindingDB Entry DOI: 10.7270/Q24M978Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM60994 ((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL DrugBank KEGG PC cid PC sid PDB UniChem Similars | PubMed | 46 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Hebrew University Curated by ChEMBL | Assay Description Compound was evaluated for the competitive inhibition of [3H]3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[... | J Med Chem 35: 2065-9 (1992) BindingDB Entry DOI: 10.7270/Q2Z60R9H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM50469729 (CHEMBL436268) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article | 48 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940 | Citation and Details Article DOI: 10.1016/S0960-894X(01)80155-4 BindingDB Entry DOI: 10.7270/Q24M978Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (MOUSE-Mus musculus (Mouse)) | BDBM22988 ((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 52 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Hebrew University Curated by ChEMBL | Assay Description Ability to displace [3H]HU-243 binding to cannabinoid receptor in synaptosomal membrane | J Med Chem 36: 3032-4 (1993) Article DOI: 10.1021/jm00072a026 BindingDB Entry DOI: 10.7270/Q2D220V0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (MOUSE-Mus musculus (Mouse)) | BDBM50231338 (CHEMBL105429) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 53 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Hebrew University Curated by ChEMBL | Assay Description Ability to displace [3H]HU-243 binding to cannabinoid receptor in synaptosomal membrane | J Med Chem 36: 3032-4 (1993) Article DOI: 10.1021/jm00072a026 BindingDB Entry DOI: 10.7270/Q2D220V0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50471437 (CHEMBL121384) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 54 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Binding affinity towards cannabinoid receptor using [3H]SR-141,716A as radioligand in rat brain membrane | J Med Chem 40: 3626-34 (1997) Article DOI: 10.1021/jm9702950 BindingDB Entry DOI: 10.7270/Q261131W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50060622 ((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid ((...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 57 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Binding affinity towards cannabinoid receptor using [3H]CP-55940 as radioligand in rat brain membrane | J Med Chem 40: 3626-34 (1997) Article DOI: 10.1021/jm9702950 BindingDB Entry DOI: 10.7270/Q261131W | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50515056 (CHEMBL4544265) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 59 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Biological Research Centre of the Hungarian Academy of Sciences Curated by ChEMBL | Assay Description Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysis | Eur J Med Chem 178: 571-588 (2019) Article DOI: 10.1016/j.ejmech.2019.05.037 BindingDB Entry DOI: 10.7270/Q2Z60SD8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM21279 (1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 69 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Biological Research Centre of the Hungarian Academy of Sciences Curated by ChEMBL | Assay Description Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysis | Eur J Med Chem 178: 571-588 (2019) Article DOI: 10.1016/j.ejmech.2019.05.037 BindingDB Entry DOI: 10.7270/Q2Z60SD8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Homo sapiens (Human)) | BDBM50469726 (CHEMBL152801) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article | 72 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940 | Citation and Details Article DOI: 10.1016/S0960-894X(01)80155-4 BindingDB Entry DOI: 10.7270/Q24M978Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1/2 (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM22988 ((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 78 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Connecticut Curated by ChEMBL | Assay Description Binding affinity for the cannabinoid receptor in the presence of phenylmethanesulfonyl fluoride (PMSF) was determined in rat fore brain membranes | J Med Chem 37: 1889-93 (1994) Article DOI: 10.1021/jm00038a020 BindingDB Entry DOI: 10.7270/Q2JQ13QV | |||||||||||
More data for this Ligand-Target Pair |
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